About the Authors

Elena Dolghih

lena.dolgikh@ucsf.edu

Affiliation Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California, United States of America

Clifford Bryant

Affiliation Small Molecule Discovery Center, University of California, San Francisco, San Francisco, California, United States of America

Adam R. Renslo

Affiliations Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California, United States of America, Small Molecule Discovery Center, University of California, San Francisco, San Francisco, California, United States of America

Matthew P. Jacobson

Affiliation Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California, United States of America

Competing Interests

I have read the journal's policy and have the following conflicts: MPJ is a consultant to Schrodinger LLC.

Author Contributions

Conceived and designed the experiments: ED CB ARR MPJ. Performed the experiments: ED CB. Analyzed the data: ED CB ARR MPJ. Contributed reagents/materials/analysis tools: ARR MPJ. Wrote the paper: ED CB ARR MPJ.