prefName Afnty1 Afnty2 Uniprot1 Uniprot2 molregno molweight targetClass ref1 ref2 actType1 actType2 Alpha-1d adrenergic receptor 9.49485002168 9.10237290871 P25100 P23944 97 383.401 Membrane receptor 13032 13032 Ki Ki Alpha-1b adrenergic receptor 9.49485002168 10.0 P35368 P15823 97 383.401 Membrane receptor 13032 31554 Ki Ki Alpha-2a adrenergic receptor 5.67100914455 5.7778039537 P08913 P22909 97 383.401 Membrane receptor 13032 13032 Ki Ki Alpha-1a adrenergic receptor 9.2924298239 9.63827216398 P35348 P43140 97 383.401 Membrane receptor 13032 31554 Ki Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.61978875829 6.34678748622 P36544 Q05941 115 162.232 Ion channel 36679,36679,46997 3343,31624,34889,36701,38541,38731,38939,45545,46997 Ki,Ki,IC50 IC50,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki Cyclooxygenase-2 6.30102999566 8.0 P35354 P35355 173 357.788 Enzyme 1881,3180,3169,3249,16897,37249,42810,41863,51519,51519,51838 2020 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Cyclooxygenase-1 6.79588001734 8.22184874962 P23219 Q63921 173 357.788 Enzyme 1881,3169,16897,35598,37249,41863,46605,51519,51519 2020 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Serotonin transporter 6.34678748622 6.90739896741 P31645 P31652 423 181.298 Transporter 50103 50103,50103 Ki IC50,IC50 Serotonin 2a (5-HT2a) receptor 7.70335696649 7.72124639905 P28223 P14842 436 321.155 Membrane receptor 42137,42137,42137,42137 41933 Ki,Ki,Ki,Ki Ki Monoamine oxidase A 4.8416375079 4.91364016933 P21397 P21396 543 135.206 Enzyme 49639 45995,49639 Ki Ki,Ki Serotonin transporter 6.32057210339 6.16115638248 P31645 P31652 592 179.216 Transporter 51535 50103,50103 IC50 IC50,IC50 Serotonin 2a (5-HT2a) receptor 8.48228513091 8.45593195565 P28223 P14842 601 323.432 Membrane receptor 42137,42137,42137,42137 13278,17133,31390 Ki,Ki,Ki,Ki Ki,Ki,Ki Monoamine oxidase B 4.58502665203 5.24052599132 P27338 P19643 711 186.21 Enzyme 46621 46621,46621 Ki Ki,IC50 Muscarinic acetylcholine receptor M1 5.29672990978 7.50863830617 P11229 P08482 892 None Membrane receptor 14237,15502 14434,14434 IC50,Ki Ki,Ki Muscarinic acetylcholine receptor M2 7.42021640338 6.88605664769 P08172 P10980 892 None Membrane receptor 14434,14434,14434,15502,15502 14434,14434,14434 IC50,IC50,Ki,Ki,Ki IC50,IC50,Ki Muscarinic acetylcholine receptor M4 5.58502665203 5.58502665203 P08173 P08485 892 None Membrane receptor 14434,15502,15502 14434 Ki,Ki,Ki Ki Muscarinic acetylcholine receptor M1 5.5631944015 3.69637974808 P11229 P08482 1022 155.194 Membrane receptor 4543,4543,14237,15502 42623,42623,48714,48714,50847,50847 IC50,IC50,IC50,Ki Ki,IC50,Ki,IC50,Ki,IC50 Muscarinic acetylcholine receptor M2 7.39794000867 6.17827366176 P08172 P10980 1022 155.194 Membrane receptor 14434,15502 9770,14434 Ki,Ki IC50,Ki Muscarinic acetylcholine receptor M4 5.61978875829 5.61978875829 P08173 P08485 1022 155.194 Membrane receptor 14434,15502,15502 14434 Ki,Ki,Ki Ki Histamine H3 receptor 7.5376020021 8.06048074738 Q9Y5N1 Q9QYN8 611887 253.341 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.3767507096 7.92081875395 Q9Y5N1 Q9QYN8 611889 253.341 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.88605664769 8.2924298239 Q9Y5N1 Q9QYN8 611891 253.341 Membrane receptor 50228 50228 Ki Ki Aldose reductase 6.25963731051 6.60205999133 P15121 P07943 2029 236.199 Enzyme 30209,38948,51711 10832,42594,49754,50326,53890 IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50 Muscarinic acetylcholine receptor M2 6.97500357154 6.06651271215 P08172 P10980 2076 206.284 Membrane receptor 15502,15502 316 Ki,Ki IC50 Dihydrofolate reductase 6.36664901656 5.63827216398 P00374 Q920D2 2080 248.711 Enzyme 43976,53022 12673 IC50,Ki IC50 Aldose reductase 7.88605664769 6.02227639471 P15121 P07943 2084 357.347 Enzyme 21693,38948,51711 10832,38646,50326 IC50,IC50,IC50 IC50,IC50,IC50 Serotonin 2c (5-HT2c) receptor 8.08092190762 7.6883753548 P28335 P08909 2214 176.215 Membrane receptor 17200,6857,30538,30606,30606,39082,40781,42924,46215,48846 10444,14178 Ki,Ki,Ki,IC50,Ki,IC50,Ki,Ki,IC50,IC50 Ki,IC50 Serotonin 1b (5-HT1b) receptor 7.7447274949 8.33724216832 P28222 P28564 2214 176.215 Membrane receptor 45320,45320,42202 14178 IC50,Ki,Ki IC50 Serotonin 4 (5-HT4) receptor 6.30102999566 6.83268266525 Q13639 Q62758 2214 176.215 Membrane receptor 42924,46295,46295 14178 Ki,Ki,IC50 IC50 Serotonin 2a (5-HT2a) receptor 7.03786035697 6.45469288353 P28223 P14842 2214 176.215 Membrane receptor 6857,30538,30606,30606,39082,40781,42924,42137,42137,42137,42137,46215 17200,17200,14178,17200,30538,46737,48520 Ki,Ki,IC50,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,IC50 IC50,IC50,IC50,Ki,IC50,Ki,Ki Serotonin 1a (5-HT1a) receptor 8.60205999133 8.55395269865 P08908 P19327 2214 176.215 Membrane receptor 17200,17200,13051 14178,12028,43958,43771,46737,48520 IC50,IC50,Ki IC50,Ki,IC50,Ki,Ki,Ki Norepinephrine transporter 5.80687540165 6.75448733219 P23975 Q9WTR4 2223 309.326 Transporter 30228,30184,31495,31619,44487,47195,44158,44579,46012,46012,44983,44983 15861 Ki,Ki,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,Ki,IC50 Ki Serotonin transporter 8.0268721464 8.40893539297 P31645 P31652 2223 309.326 Transporter 30228,30184,31450,31495,31619,36227,36915,37349,37465,43754,44487,47195,44158,44579,44692,46012,46012,44898,44983,44983,48123,48706,48811,49880,49648,51128,51343,52510 5371,15861,3775,31450,36227,36474,36915,37349,37465,43800,44692,45021,47621,49889,52510 Ki,Ki,IC50,IC50,IC50,Ki,Ki,Ki,Ki,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50 Dopamine transporter 5.22184874962 5.22184874962 Q01959 P23977 2223 309.326 Transporter 30228,30184,31495,31619,44487,44158,46012,46012,44983,44983 45021 Ki,Ki,IC50,IC50,IC50,IC50,Ki,IC50,Ki,IC50 IC50 Serotonin 2a (5-HT2a) receptor 7.82390874094 8.02090709936 P28223 P14842 2232 218.295 Membrane receptor 30538 30538 Ki IC50 Serotonin 2c (5-HT2c) receptor 7.76955107862 7.95860731484 P28335 P08909 2261 326.823 Membrane receptor 43952 14229 Ki IC50 Dopamine D3 receptor 6.53017798402 6.30102999566 P35462 P19020 2261 326.823 Membrane receptor 13379,13378,13910,31339,43952,46646,47889 12771 Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki Histamine H1 receptor 8.68407526892 7.94981472744 P35367 P31390 2261 326.823 Membrane receptor 43952,46646 16647,39442 Ki,Ki Ki,IC50 Dopamine D2 receptor 7.13076828027 6.5869950111 P14416 P61169 2261 326.823 Membrane receptor 2541,13379,13378,13910,15727,30228,31339,31339,31631,31663,43952,46646,47889,47889 10451,14229,13134,2100,45067,51830 Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki IC50,IC50,Ki,Ki,Ki,Ki Dopamine D1 receptor 6.87942606879 6.69723973828 P21728 P18901 2261 326.823 Membrane receptor 31631,31663,43952,46646 10451,14229,45067,51830 Ki,Ki,Ki,Ki IC50,IC50,Ki,Ki Dopamine D4 receptor 7.53190403817 7.49485002168 P21917 P30729 2261 326.823 Membrane receptor 13378,13910,13379,20195,20195,30228,31339,43952 13427 Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki Ki Serotonin 2a (5-HT2a) receptor 8.05060999336 8.0 P28223 P14842 2261 326.823 Membrane receptor 43952 14229,45067,46353,49687,51830 Ki IC50,Ki,Ki,Ki,Ki Serotonin 1a (5-HT1a) receptor 6.85387196432 6.79588001734 P08908 P19327 2261 326.823 Membrane receptor 43952 11049,12771,45067,49687,51830 Ki IC50,Ki,Ki,Ki,Ki P2X purinoceptor 7 6.33724216832 4.72124639905 Q99572 Q64663 437302 449.545 Ion channel 38841 38841 IC50 IC50 Dopamine D2 receptor 6.70190385075 6.36407919673 P14416 P61169 2724 219.323 Membrane receptor 49693,49693 10465,10465 Ki,Ki IC50,IC50 Monoglyceride lipase 4.72124639905 4.45593195565 Q99685 Q8R431 567488 279.332 Enzyme 47831 47831 IC50 IC50 Serotonin 1a (5-HT1a) receptor 8.22184874962 8.25963731051 P08908 P19327 3587 401.483 Membrane receptor 31185 43958 Ki Ki Serotonin 1a (5-HT1a) receptor 7.73426054148 8.03249842427 P08908 P19327 3599 385.503 Membrane receptor 31185,31374,46667,46667 14331,13825,11642,43958,46068,46353 Ki,Ki,Ki,IC50 Ki,Ki,Ki,Ki,Ki,Ki Sucrase-isomaltase 4.45593195565 3.9345116542 P14410 P23739 3665 270.237 Enzyme 40101 38800,40101 IC50 IC50,IC50 Aldose reductase 6.74365780189 5.38828837519 P15121 P07943 3666 302.236 Enzyme 38948,44762 10832,10832,36696,41934 IC50,IC50 IC50,IC50,IC50,IC50 Serotonin 2a (5-HT2a) receptor 8.24405831951 9.19019249713 P28223 P14842 3683 395.427 Membrane receptor 43854,45320,45320,47190 1559,36609,37090,48634 IC50,Ki,IC50,IC50 IC50,Ki,Ki,Ki Arachidonate 5-lipoxygenase 6.88605664769 8.0 P09917 P12527 3784 302.365 Enzyme 35598,44465,51447 961 IC50,IC50,IC50 IC50 Dopamine D2 receptor 7.59691001301 7.91267940367 P14416 P61169 3854 267.322 Membrane receptor 16372,34751,37919,38679,43771,41947,49693,49693 10383,10587,38182,38524,41947,41947,47870,47870 Ki,Ki,IC50,IC50,Ki,Ki,Ki,Ki IC50,Ki,Ki,Ki,Ki,Ki,Ki,IC50 Dopamine D1 receptor 6.91079932923 6.62708799703 P21728 P18901 3854 267.322 Membrane receptor 38679,43771 10383,10587,8741,38182,38524 IC50,Ki IC50,Ki,Ki,Ki,Ki Sigma opioid receptor 7.48775716615 8.00683811147 Q99720 Q9R0C9 3859 375.864 Membrane receptor 12347,50595 16719,16655,11576,12885,15667,38870,46059,47758 Ki,IC50 Ki,Ki,IC50,IC50,Ki,Ki,Ki,Ki Dopamine D3 receptor 8.19382002602 8.07133375178 P35462 P19020 3859 375.864 Membrane receptor 12121,13379,13378,12032,21038,30313,36383,36703,43952,45899,51800,53158 12771,30552 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Histamine H1 receptor 6.35654732351 6.41566877563 P35367 P31390 3859 375.864 Membrane receptor 43952 16647 Ki Ki Dopamine D2 receptor 8.78755918168 8.73975823363 P14416 P61169 3859 375.864 Membrane receptor 12121,2541,13379,13378,13910,13670,21038,30252,43952,45355,45366,44623,45253,45899,49693,49693,51064,51800,53158,53158 9174,14509,14229,9205,3070,14389,12032,2100,21218,45067 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki IC50,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki Dopamine D1 receptor 7.00350245078 7.44369749923 P21728 P18901 3859 375.864 Membrane receptor 21038,43952 14229,3070,45067 Ki,Ki IC50,Ki,Ki Serotonin 2a (5-HT2a) receptor 6.92081875395 7.02239673123 P28223 P14842 3859 375.864 Membrane receptor 43952 14229,45067 Ki IC50,Ki Serotonin 1a (5-HT1a) receptor 5.44369749923 5.7447274949 P08908 P19327 3859 375.864 Membrane receptor 43952 45067 Ki Ki Metabotropic glutamate receptor 5 8.69897000434 8.28066871302 P41594 P31424 306513 277.344 Membrane receptor 20024 46751 IC50 IC50 Dopamine D2 receptor 7.06550154876 7.06550154876 P14416 P61169 4149 247.376 Membrane receptor 12249 2331 Ki Ki Serotonin 1a (5-HT1a) receptor 8.67778070527 8.92081875395 P08908 P19327 4149 247.376 Membrane receptor 2331,36609,38784,43854,45355,45320,45320,44692,44692,45253 14331,17136,17331,12058,35308,37090,44570,48634 Ki,Ki,Ki,IC50,Ki,Ki,IC50,Ki,IC50,Ki Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Serotonin 1a (5-HT1a) receptor 9.22184874962 9.24074303006 P08908 P19327 4181 393.479 Membrane receptor 48700 13825,15247 Ki Ki,Ki Dopamine D2 receptor 8.29904137474 8.44369749923 P14416 P61169 4259 361.52 Membrane receptor 2541,43854,45320,45320 10263,15453,21218 Ki,IC50,Ki,IC50 Ki,Ki,Ki Monoamine oxidase B 4.21218543294 3.39696394375 P27338 P19643 4381 272.17 Enzyme 47084,44148,44874,46413,49935,50304,51147,52183,52782,52818,52882 35878,45377,45377,44921 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,Ki,IC50,IC50 Monoamine oxidase A 8.35066514129 5.68824613894 P21397 P21396 4381 272.17 Enzyme 43854,47084,44148,44874,46413,49935,50304,51147,52183,52782,52818,52882 35878,45377,45377,44921 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,Ki,IC50 Cannabinoid CB1 receptor 8.15357654036 7.38721614328 P21554 P20272 4496 314.462 Membrane receptor 36793,44405 39196,52192,53907 Ki,Ki Ki,Ki,Ki P2X purinoceptor 7 6.50863830617 6.85387196432 Q99572 Q64663 437669 487.595 Ion channel 38841 38841 IC50 IC50 Dopamine D1 receptor 7.57745097999 6.46040937698 P21728 P18901 4584 153.178 Membrane receptor 38679,52488 8741,10581 IC50,IC50 Ki,IC50 Dopamine D2 receptor 6.67985371389 5.96017878052 P14416 P61169 4584 153.178 Membrane receptor 13670,15817,15817,38128,38679,42030,44689,44689,47595,49130,49693,49693,49668,52843 10581,10263,47870,47870 Ki,Ki,Ki,IC50,IC50,IC50,Ki,Ki,IC50,IC50,Ki,Ki,IC50,IC50 IC50,Ki,Ki,IC50 Serotonin 7 (5-HT7) receptor 6.95860731484 7.69897000434 P34969 P32305 4634 395.47 Membrane receptor 17066 17066 Ki Ki Dopamine D2 receptor 9.35654732351 10.1003297253 P14416 P61169 4634 395.47 Membrane receptor 43771 10263,21218 Ki Ki,Ki Cannabinoid CB1 receptor 7.54515513999 7.32239304728 P21554 P20272 4750 314.462 Membrane receptor 44424,46129 5256,30893,45300 Ki,Ki Ki,Ki,Ki Dopamine D1 receptor 9.09691001301 9.0 P21728 P18901 4778 287.784 Membrane receptor 43854,43771,45320,45320,48842 13090,14693,10581 IC50,Ki,IC50,Ki,Ki IC50,IC50,IC50 Histamine H3 receptor 9.14266750357 8.79588001734 Q9Y5N1 Q9QYN8 350352 330.507 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.34678748622 8.4921441283 Q9Y5N1 Q9QYN8 267366 330.423 Membrane receptor 21227,30224,36041,37121,37121,37369,43979,44709,47387,51341 37121,37121,37121,37369,47387,51341 Ki,Ki,Ki,Ki,IC50,Ki,Ki,IC50,Ki,Ki Ki,Ki,IC50,Ki,Ki,Ki Histamine H3 receptor 7.93554201077 7.311580178 Q9Y5N1 Q9QYN8 350419 330.464 Membrane receptor 31381 31381 Ki Ki Adenosine A1 receptor 6.06098022355 5.90974194707 P30542 P25099 267552 385.417 Membrane receptor 3027 3027 IC50 IC50 Cholecystokinin A receptor 9.30980391997 10.0 P32238 P30551 5535 408.452 Membrane receptor 43854 11697,604,9864 IC50 Ki,IC50,IC50 Mu opioid receptor 8.39794000867 7.84620919762 P35372 P33535 6005 285.338 Membrane receptor 30571,31576,36720,39273,39273,39273,39273,46008,48670 11019,13393,6196,11861,39391,49432,49432,51243 Ki,Ki,Ki,IC50,IC50,IC50,Ki,IC50,Ki IC50,IC50,Ki,Ki,IC50,Ki,IC50,IC50 Delta opioid receptor 6.85387196432 6.39361863489 P41143 P33533 6005 285.338 Membrane receptor 30571,31576,36720,46008 11019,13393,39391,49432,51243 Ki,Ki,Ki,IC50 IC50,IC50,IC50,Ki,IC50 Vasopressin V2 receptor 6.65757731918 7.61978875829 P30518 Q00788 268323 442.533 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V1a receptor 5.75945075172 5.69680394258 P37288 P30560 268323 442.533 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V2 receptor 6.85387196432 6.46852108296 P30518 Q00788 268324 466.915 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V2 receptor 7.14874165128 7.16115090926 P30518 Q00788 268352 446.497 Membrane receptor 4138 4138 IC50 IC50 Dopamine D1 receptor 7.01772876696 8.66756154008 P21728 P18901 6216 318.864 Membrane receptor 46646 13090 Ki IC50 Vasopressin V2 receptor 8.56863623584 8.82390874094 P30518 Q00788 268557 518.005 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V1a receptor 6.43179827593 7.79588001734 P37288 P30560 268557 518.005 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V2 receptor 6.88605664769 6.92081875395 P30518 Q00788 268602 428.506 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V1a receptor 6.61978875829 5.67778070527 P37288 P30560 268602 428.506 Membrane receptor 4138 4138 IC50 IC50 Cytochrome P450 24A1 6.50584540598 4.69897000434 Q07973 Q09128 6514 531.431 Enzyme 35331 52858 IC50 IC50 Cytochrome P450 17A1 5.55595520408 5.49996525922 P05093 P11715 6514 531.431 Enzyme 13523,13523,38222,38400,44172,44174,44186,45200,47824,51275,51866,52270 10691,10691,48065,48065,52424,52424 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50,IC50 Vasopressin V2 receptor 6.82390874094 7.42021640338 P30518 Q00788 268666 497.396 Membrane receptor 4138 4138 IC50 IC50 Vasopressin V1a receptor 5.38721614328 5.67778070527 P37288 P30560 268666 497.396 Membrane receptor 4138 4138 IC50 IC50 Alpha-1d adrenergic receptor 7.16767901222 7.45593195565 P25100 P23944 6593 354.443 Membrane receptor 13061,13032 13032 Ki,Ki Ki Dopamine transporter 6.39794000867 6.20551195334 Q01959 P23977 6643 329.365 Transporter 30184 14615 Ki IC50 Serotonin transporter 9.42021640338 9.2757241304 P31645 P31652 6643 329.365 Transporter 30184,37090,44082,44082,44570,44579,42172,42172 5371,3775,14615 Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki Ki,Ki,IC50 Muscarinic acetylcholine receptor M1 7.62893213773 8.28357946653 P11229 P08482 6772 351.402 Membrane receptor 21052,30369,37078,43854,45320,45320 10799,2520 Ki,Ki,Ki,IC50,IC50,Ki Ki,Ki Histamine H3 receptor 9.2757241304 9.01322826573 Q9Y5N1 Q9QYN8 350692 384.598 Membrane receptor 31381 31381 Ki Ki Serotonin 1a (5-HT1a) receptor 6.63827216398 6.63827216398 P08908 P19327 350712 456.578 Membrane receptor 31374 46353 Ki Ki Alpha-2a adrenergic receptor 7.16749108729 8.5376020021 P08913 P22909 44906 232.345 Membrane receptor 15822 15822,15882 Ki Ki,Ki Dihydrofolate reductase 3.69897000434 3.87614835903 P00374 Q920D2 1216 290.318 Enzyme 15984,36076,43976,45337,48431,49279,50606 12673,17495,14276,14893,36076,36100,43976,45205,49279,49957 IC50,IC50,IC50,IC50,IC50,Ki,IC50 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50 Serotonin transporter 6.0985416786 6.62342304294 P31645 P31652 438128 404.505 Transporter 38371 38371 Ki Ki Serotonin 2a (5-HT2a) receptor 5.33629907461 5.24412514433 P28223 P14842 7646 197.276 Membrane receptor 49240 4664 Ki Ki Histamine H1 receptor 7.72124639905 7.09691001301 P35367 P31390 7714 410.484 Membrane receptor 43952 39442 Ki IC50 Dopamine D2 receptor 8.65757731918 8.42021640338 P14416 P61169 7714 410.484 Membrane receptor 43952 3070,21218,45067 Ki Ki,Ki,Ki Dopamine D1 receptor 6.23657200644 7.47930365742 P21728 P18901 7714 410.484 Membrane receptor 43952 3070,45067 Ki Ki,Ki Serotonin 2a (5-HT2a) receptor 9.5376020021 9.82390874094 P28223 P14842 7714 410.484 Membrane receptor 43952 45067 Ki Ki Serotonin 1a (5-HT1a) receptor 6.67778070527 6.72124639905 P08908 P19327 7714 410.484 Membrane receptor 43952 45067 Ki Ki Coagulation factor X 10.0 8.87942606879 P00742 Q63207 497828 565.955 Enzyme 46394 46394 IC50 IC50 Serotonin 1a (5-HT1a) receptor 7.76955107862 7.76955107862 P08908 P19327 350960 484.631 Membrane receptor 31374 46353 Ki Ki Serotonin 1a (5-HT1a) receptor 6.46344155743 5.9829666607 P08908 P19327 9128 247.376 Membrane receptor 2331 12058 Ki Ki Dopamine D2 receptor 7.38510278397 7.59859945922 P14416 P61169 9128 247.376 Membrane receptor 47595,49130,49130 12058,2331,47595,52843 IC50,Ki,IC50 Ki,Ki,Ki,Ki Dopamine D3 receptor 8.8882779901 8.86646109163 P35462 P19020 9128 247.376 Membrane receptor 2331,47595,49130,49130 47595,52843 Ki,IC50,Ki,IC50 Ki,Ki Arachidonate 5-lipoxygenase 6.09691001301 6.09474395125 P09917 P12527 9217 236.29 Enzyme 20275,20777,46825,46825,44797,47888,50733,51519,51519,51519 14427,338,35997 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50 Butyrylcholinesterase 7.55284196866 7.87872928585 P06276 Q9JKC1 9277 275.346 Enzyme 14083,10673,10673,10673,10673,21324,21519,30919,30919,34898,45281,49147,51782 14639,50487 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50 Acetylcholinesterase 7.45593195565 8.84948500217 P22303 P37136 9277 275.346 Enzyme 1308,14083,10673,10673,10673,10673,21324,21519,30919,30919,34898,51782,52762 14639,50487 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50 Butyrylcholinesterase 7.44369749923 7.03621217265 P06276 Q9JKC1 9333 198.264 Enzyme 16061,21244,21435,21519,30445,30919,31257,31842,34767,35354,35892,36705,37091,37270,43975,45783,47082,44067,42156,42214,50243,51864,53122 3267,31775,41889,42214 IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,Ki,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Acetylcholinesterase 6.68824613894 6.65169513695 P22303 P37136 9333 198.264 Enzyme 16061,15335,11387,21244,21435,21519,30445,30919,31257,31842,36705,37091,37164,37270,38283,43975,45783,47082,44067,42156,47991,49254,50243,51286,51864,52762,53122 327,3267,31775,41889,42214,48633 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50,IC50 Butyrylcholinesterase 5.12959609472 5.33068311943 P06276 Q9JKC1 9372 379.492 Enzyme 16061,21519,30919,35892,36705,45877,47136,42214,49723 44140,41889,46056,42214,49233 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50 Acetylcholinesterase 7.67291172906 7.92081875395 P22303 P37136 9372 379.492 Enzyme 16061,15335,21519,30919,35297,36705,38283,45877,47136,49723,51286,52762 44140,41889,45908,46056,42214,49233 IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50,IC50 Serotonin 1a (5-HT1a) receptor 7.7447274949 8.04575749056 P08908 P19327 351128 496.642 Membrane receptor 31374 36406,46353 Ki Ki,Ki Acetylcholinesterase 6.49757288002 6.48811663902 P22303 P37136 569641 287.806 Enzyme 48391 48391 IC50 IC50 Acetylcholinesterase 7.04575749056 7.12493873661 P22303 P37136 569642 322.251 Enzyme 48391 48391 IC50 IC50 Acetylcholinesterase 6.339134522 6.33441900898 P22303 P37136 569647 309.467 Enzyme 48391 48391 IC50 IC50 Histamine H3 receptor 7.79588001734 6.79588001734 Q9Y5N1 Q9QYN8 438653 219.323 Membrane receptor 38490 38490 Ki Ki Serotonin 7 (5-HT7) receptor 7.49485002168 7.50031291738 P34969 P32305 10841 338.508 Membrane receptor 17066 16372 Ki Ki Muscarinic acetylcholine receptor M1 7.25181197299 7.56863623584 P11229 P08482 11015 174.261 Membrane receptor 15502 14434,14434 Ki Ki,Ki Muscarinic acetylcholine receptor M2 7.12493873661 6.30980391997 P08172 P10980 11015 174.261 Membrane receptor 14434,14434,14434,15502,15502 14434,14434,14434 IC50,IC50,Ki,Ki,Ki IC50,IC50,Ki Muscarinic acetylcholine receptor M4 6.74607206415 5.85387196432 P08173 P08485 11015 174.261 Membrane receptor 15502,15502 14434 Ki,Ki Ki Dipeptidyl peptidase IV 7.39794000867 7.23657200644 P27487 P14740 438778 378.492 Enzyme 38801,38801 38801 IC50,IC50 IC50 Glutamate receptor ionotropic kainate 5 6.75202673364 7.82390874094 Q16478 Q63273 11671 213.23 Ion channel 14175 43825 Ki Ki Glutamate receptor ionotropic, AMPA 1 5.12784372725 4.63827216398 P42261 P19490 11671 213.23 Ion channel 14175 45271,47617,50876,50876 Ki Ki,IC50,IC50,IC50 Glutamate receptor ionotropic, AMPA 2 4.91364016933 3.42021640338 P42262 P19491 11671 213.23 Ion channel 14175 45271,47617,50876 Ki Ki,IC50,IC50 Glutamate receptor ionotropic, AMPA 4 5.76700388961 4.32790214206 P48058 P19493 11671 213.23 Ion channel 14175 45271,47617,50876 Ki Ki,IC50,IC50 Mu opioid receptor 6.45345733652 5.24321180123 P35372 P33535 12225 449.628 Membrane receptor 48996 12391,12391,13393 Ki IC50,IC50,IC50 Delta opioid receptor 8.42154378715 7.65874695703 P41143 P33533 12225 449.628 Membrane receptor 37896,39029,45228,45228,46432,47540,48996,48996 13393,48465 IC50,Ki,Ki,IC50,IC50,IC50,Ki,IC50 IC50,IC50 Kappa opioid receptor 5.37996810487 5.44357687863 P41145 P34975 12225 449.628 Membrane receptor 48996 49186 Ki IC50 Calcitonin receptor 10.1611509093 9.6038006529 P30988 P32214 12836 3430.87 Membrane receptor 16855 16855 Ki IC50 Alpha-1a adrenergic receptor 6.60205999133 7.01 P35348 P43140 12872 385.5 Membrane receptor 4771,16909,20732 16909 Ki,IC50,Ki IC50 Alpha-1b adrenergic receptor 7.02548830726 7.48 P35368 P15823 12872 385.5 Membrane receptor 4771 16909 Ki IC50 Calcitonin receptor 7.37161106995 5.61083391564 P30988 P32214 12943 3376.84 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 9.25181197299 8.26841123481 P30988 P32214 12944 3354.81 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 10.638272164 9.48678239993 P30988 P32214 12997 3406.84 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 8.27736607747 7.10237290871 P30988 P32214 13017 3372.83 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 6.70996538864 7.22184874962 P30988 P32214 13021 3386.88 Membrane receptor 16855 16855 Ki IC50 Histamine H3 receptor 6.1402614338 7.37468754904 Q9Y5N1 Q9QYN8 13036 123.156 Membrane receptor 16985 16985 IC50 Ki Histamine H3 receptor 7.3767507096 8.36653154442 Q9Y5N1 Q9QYN8 13050 123.156 Membrane receptor 16985 16985 IC50 Ki Calcitonin receptor 5.91044811711 5.72010501999 P30988 P32214 13053 3345.78 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 10.2924298239 9.42365864979 P30988 P32214 13067 3433.87 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 10.3010299957 9.7447274949 P30988 P32214 13140 3444.9 Membrane receptor 16855 16855 Ki IC50 Calcitonin receptor 10.1611509093 9.38933983691 P30988 P32214 13141 3431.9 Membrane receptor 16855 16855 Ki IC50 Gamma-amino-N-butyrate transaminase 4.78251605579 4.78251605579 P80404 P50554 13328 122.121 Enzyme 30636 45659 IC50 IC50 Nitric-oxide synthase, brain 5.0 6.9761679027 P29475 P29476 613899 390.47 Enzyme 50330 50330,50330 IC50 IC50,Ki Acetylcholinesterase 6.7166987713 6.73048705578 P22303 P37136 570211 298.358 Enzyme 48391 48391 IC50 IC50 HMG-CoA reductase 7.55284196866 8.52287874528 P04035 P51639 140116 411.466 Enzyme 20770 47915 IC50 IC50 Mu opioid receptor 5.31515463836 5.71449516385 P35372 P33535 13693 369.329 Membrane receptor 39419 11861,52824 IC50 Ki,Ki Prostanoid EP4 receptor 8.91180965388 8.91634133263 P35408 P43114 14125 352.465 Membrane receptor 37631,37888,38798,38798,45320,45320 47314,47314 Ki,Ki,Ki,IC50,Ki,IC50 IC50,IC50 Prostanoid EP2 receptor 8.30980391997 8.99148333035 P43116 Q62928 14125 352.465 Membrane receptor 37631,37888,38798 47314,47314 Ki,Ki,Ki IC50,IC50 Serotonin transporter 8.3767507096 8.37571790416 P31645 P31652 14241 385.24 Transporter 17704 13641,13641,3817 Ki IC50,IC50,Ki Serotonin transporter 8.3585258895 8.71219827007 P31645 P31652 14367 324.392 Transporter 17704,44082,44082,42172,42172 3775,50103,52243 Ki,Ki,Ki,Ki,Ki Ki,IC50,Ki Histamine H3 receptor 8.80989437914 9.22184874962 Q9Y5N1 Q9QYN8 14559 308.83 Membrane receptor 50228,53396 3951 Ki,IC50 Ki Histamine H3 receptor 7.26895080943 9.30980391997 Q9Y5N1 Q9QYN8 14718 270.326 Membrane receptor 21227,50228 3951 Ki,Ki Ki Kappa opioid receptor 7.52775866392 9.20065945055 P41145 P34975 15149 356.502 Membrane receptor 37097,37097,44050,42671,42671,50996 2703 IC50,IC50,IC50,IC50,IC50,IC50 IC50 Alpha-1d adrenergic receptor 7.66749108729 7.28399665637 P25100 P23944 15191 354.443 Membrane receptor 13061,13032 13032 Ki,Ki Ki Sodium channel protein type X alpha subunit 4.25181197299 4.50863830617 Q9Y5Y9 Q62968 15958 179.259 Ion channel 42188 42188 IC50 IC50 Cannabinoid CB1 receptor 8.26760624018 8.34390179799 P21554 P20272 16088 463.787 Membrane receptor 21631,21571,20730,20855,30097,30560,30663,31883,31883,34762,35375,35980,36010,37225,37904,38502,38562,38562,38671,39325,43936,47186,47057,44206,45166,45166,45193,45193,45533,45533,45533,45499,42580,46986,46986,42209,42209,42209,42092,42092,45084,45084,46331,47927,47927,48435,48905,49460,49514,49532,49532,49532,49921,49829,50392,50392,50392,51101,51101,52280,53408,53408,53408 38929,45882,47034,45637,45637,46772,41874,42574,42580,42092,44990,45084,46418,47614,48261,49038,48905,49921,51963,52405,53408 Ki,Ki,IC50,IC50,Ki,Ki,Ki,Ki,Ki,IC50,Ki,IC50,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,IC50,Ki,Ki,IC50,IC50,IC50,Ki,IC50,Ki,IC50,Ki,IC50,IC50,IC50,Ki,Ki,IC50,Ki,IC50,Ki,Ki,Ki,Ki,IC50,Ki,Ki,IC50,IC50,IC50,IC50,IC50,IC50,Ki,Ki,IC50,IC50,Ki,IC50,Ki,Ki,Ki,IC50 IC50,IC50,IC50,IC50,Ki,Ki,IC50,IC50,IC50,Ki,IC50,Ki,IC50,Ki,IC50,IC50,Ki,IC50,IC50,IC50,IC50 Cannabinoid CB1 receptor 7.15490195999 6.87942606879 P21554 P20272 16217 347.535 Membrane receptor 21380,30511,30928,31470,35365,35863,45420,47070,46289 13682,40501,48741 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki,Ki Vanilloid receptor 6.69897000434 6.77211329539 Q8NER1 O35433 16217 347.535 Ion channel 47070 16255 IC50 Ki Serotonin 1a (5-HT1a) receptor 7.14266750357 6.37161106995 P08908 P19327 16396 497.588 Membrane receptor 2391,30095,30095 15796 Ki,Ki,Ki IC50 Histamine H3 receptor 9.02227639471 8.34678748622 Q9Y5N1 Q9QYN8 632088 419.605 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 10.0 9.60205999133 Q9Y5N1 Q9QYN8 631651 377.506 Membrane receptor 51341 51341 Ki Ki Adenosine A1 receptor 4.30980391997 4.58251957437 P30542 P25099 16485 194.191 Membrane receptor 38739,42591,47890 11687,11292,11292,37033,37600,41516,43227,49741 Ki,Ki,Ki Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Adenosine A2a receptor 4.74232142513 4.48811663902 P29274 P30543 16485 194.191 Membrane receptor 38739,42591,47890 37033,37600,41516,44553,43227,49741 Ki,Ki,Ki Ki,Ki,Ki,Ki,Ki,Ki Adenosine A2a receptor 7.69897000434 7.04575749056 P29274 P30543 279670 293.363 Membrane receptor 44049 6610 Ki Ki Vasopressin V2 receptor 7.23657200644 7.30102999566 P30518 Q00788 308814 422.52 Membrane receptor 44817 44817 IC50 IC50 Histamine H3 receptor 7.01772876696 8.60205999133 Q9Y5N1 Q9QYN8 94393 137.182 Membrane receptor 16985 16985 IC50 Ki Adenosine A3 receptor 7.07058107429 4.0 P33765 P28647 18409 285.689 Membrane receptor 15744,31432 13642 Ki,Ki Ki Adenosine A1 receptor 8.35166740487 7.67778070527 P30542 P25099 18409 285.689 Membrane receptor 13642,15744 13642,10574 Ki,Ki IC50,Ki Adenosine A2a receptor 9.1739251973 8.70115240704 P29274 P30543 18409 285.689 Membrane receptor 13642,17274,17274,17274,17274,17274,17274,14051,14051,14051,15744,44049,49760 13642,989 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki IC50,Ki Adenosine A1 receptor 6.24328405159 6.66307501133 P30542 P25099 18511 345.358 Membrane receptor 14441,50765 17447,35271 Ki,Ki Ki,Ki Adenosine A2a receptor 8.9343511017 8.03503521996 P29274 P30543 18511 345.358 Membrane receptor 16389,14441,20969,43756,43769,44049,48395,50765 17447,35271 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A2b receptor 8.70553377384 7.89279003035 P29275 P29276 18536 486.522 Membrane receptor 15856,16896,20724,31281,46829,51928 16424,46829 Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A1 receptor 6.39469495386 7.77469071827 P30542 P25099 18536 486.522 Membrane receptor 16896,20724,31281,46829,51928 16896,46829 Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A2a receptor 6.29843201494 6.21324857785 P29274 P30543 18536 486.522 Membrane receptor 16896,31281,46829,51928 16896,46829 Ki,Ki,Ki,Ki Ki,Ki Adenosine A2a receptor 8.82390874094 7.85387196432 P29274 P30543 440015 451.565 Membrane receptor 38555 38555 Ki Ki Adenosine A3 receptor 7.04431224969 5.56066730617 P33765 P28647 18693 414.455 Membrane receptor 15856 15856 Ki Ki Androgen Receptor 8.49485002168 7.22184874962 P10275 P15207 364998 307.303 Transcription Factor 34764,34764,35979,35979,36077,36077,36821 34764,34764,34764 Ki,Ki,IC50,Ki,Ki,IC50,Ki IC50,IC50,IC50 Dihydrofolate reductase 7.06890448447 8.52287874528 P00374 Q920D2 19101 369.418 Enzyme 15984,51527 17611,14096,12673,12062,14893,36076,43976,45205,49957 IC50,IC50 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 Dopamine D2 receptor 6.51712641639 5.57283859707 P14416 P61169 19316 260.375 Membrane receptor 14294,37919,49130,49668,52843 52843 Ki,IC50,IC50,IC50,IC50 Ki Dopamine D3 receptor 7.98716277529 7.53313237965 P35462 P19020 19316 260.375 Membrane receptor 14294,37919,49130,49668,52843 52843 Ki,IC50,IC50,IC50,IC50 Ki Glycine transporter 1 8.61978875829 8.49485002168 P48067 P28572 368857 506.443 Transporter 34944 34944 IC50 IC50 Peroxisome proliferator-activated receptor gamma 6.6883753548 6.15490195999 P37231 O88275 19737 356.439 Transcription Factor 50782,52221 42166 IC50,IC50 IC50 Mu opioid receptor 8.5376020021 8.22914798836 P35372 P33535 19915 336.471 Membrane receptor 6559 50686 Ki Ki Dihydrofolate reductase 4.48148606012 5.90308998699 P00374 Q920D2 489493 299.394 Enzyme 43976 43976 IC50 IC50 Alpha-2a adrenergic receptor 7.25258819211 8.32790214206 P08913 P22909 20131 281.352 Membrane receptor 30076 13032 Ki Ki C-X-C chemokine receptor type 4 6.61083391564 6.96657624451 P61073 O08565 20346 502.782 Membrane receptor 42523,42523,45946,45946,44811 44811 Ki,Ki,IC50,IC50,IC50 IC50 Neprilysin 7.70553377384 7.84466396253 P08473 P07861 352984 339.453 Enzyme 31362,31362,35497,35497,35497 31362,35497 IC50,IC50,IC50,IC50,IC50 IC50,IC50 Serotonin 2c (5-HT2c) receptor 8.16767901222 6.82390874094 P28335 P08909 20819 190.242 Membrane receptor 17200,30538 10444 Ki,Ki Ki Serotonin 2a (5-HT2a) receptor 7.92081875395 8.6399203483 P28223 P14842 20819 190.242 Membrane receptor 30538 17200,17200,17200,30538 Ki IC50,IC50,Ki,IC50 Adenosine A2a receptor 8.61978875829 7.38721614328 P29274 P30543 440405 437.538 Membrane receptor 38555 38555 Ki Ki Dopamine transporter 7.92081875395 8.28383610387 Q01959 P23977 21086 299.474 Transporter 43854,45320,45320 12267,12267 IC50,Ki,IC50 IC50,IC50 Adenosine A2a receptor 7.95860731484 7.46852108296 P29274 P30543 440433 437.538 Membrane receptor 38555 38555 Ki Ki Serotonin 3a (5-HT3a) receptor 8.43179827593 9.01772876696 P46098 P35563 21258 213.278 Ion channel 36679 46737,48520 Ki Ki,Ki Mu opioid receptor 8.1238028958 8.54363396687 P35372 P33535 509921 751.914 Membrane receptor 42132,42132 42132 Ki,IC50 Ki Histamine H3 receptor 8.72124639905 8.77642098433 Q9Y5N1 Q9QYN8 22385 170.235 Membrane receptor 16985,51165,51165 15187,15187 IC50,Ki,IC50 IC50,IC50 Serotonin transporter 7.0840727883 8.48148606012 P31645 P31652 353362 453.524 Transporter 31450 31450 IC50 Ki Serotonin transporter 6.52287874528 7.9829666607 P31645 P31652 353363 453.524 Transporter 31450 31450 IC50 Ki Alpha-1d adrenergic receptor 8.45593195565 7.45593195565 P25100 P23944 23093 387.433 Membrane receptor 13032 13032 Ki Ki Serotonin transporter 6.93554201077 7.82973828461 P31645 P31652 353433 399.434 Transporter 31450 31450 IC50 Ki Adenosine A3 receptor 7.87289520164 6.38721614328 P33765 P28647 178743 371.493 Membrane receptor 31432 15333 Ki Ki P2X purinoceptor 7 5.88605664769 4.79588001734 Q99572 Q64663 437250 463.572 Ion channel 38841 38841 IC50 IC50 Sigma opioid receptor 7.22184874962 7.0530567293 Q99720 Q9R0C9 24304 239.316 Membrane receptor 12347 16719,16655,46059,47758,48530 Ki Ki,Ki,Ki,Ki,Ki Serotonin transporter 7.59859945922 8.52287874528 P31645 P31652 353672 439.498 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Dopamine transporter 7.56863623584 7.97469413474 Q01959 P23977 24971 450.563 Transporter 43854 15202,4998,31402,31402,35266,37932,39086,39086,49889 IC50 IC50,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki Heme oxygenase 1 5.82390874094 6.09691001301 P09601 P06762 549383 306.787 Enzyme 31360 31360 IC50 IC50 Serotonin transporter 6.05403929642 7.22040350874 P31645 P31652 353738 399.434 Transporter 31450 31450 IC50 Ki Vasopressin V1b receptor 7.15490195999 7.79588001734 P47901 P48974 572208 619.836 Membrane receptor 48483 48483 Ki Ki Peroxisome proliferator-activated receptor alpha 6.96040937698 6.77989191196 Q07869 P37230 25512 492.622 Transcription Factor 17297,35939,46424,51326 38094 IC50,IC50,IC50,IC50 IC50 Vasopressin V1b receptor 6.91364016933 7.04095860768 P47901 P48974 572257 627.814 Membrane receptor 48483 48483 Ki Ki Histamine H3 receptor 8.08092190762 7.82390874094 Q9Y5N1 Q9QYN8 611890 253.341 Membrane receptor 50228 50228 Ki Ki Acetylcholinesterase 6.54637592641 6.69897000434 P22303 P37136 353878 401.493 Enzyme 31481 31481 IC50 IC50 Vasopressin V1b receptor 6.94309514866 5.35105481783 P47901 P48974 572340 560.128 Membrane receptor 48483 48483 Ki Ki Adenosine A3 receptor 3.91736596318 4.18708664336 P33765 P28647 26237 194.191 Membrane receptor 31281,46829 46829 Ki,Ki Ki Adenosine A1 receptor 4.36664901656 3.80687540165 P30542 P25099 26237 194.191 Membrane receptor 31281,46829 46829 Ki,Ki Ki Adenosine A2a receptor 4.29237973804 4.49485002168 P29274 P30543 26237 194.191 Membrane receptor 31281,46829 46829 Ki,Ki Ki Oxytocin receptor 7.55284196866 7.33483311575 P30559 P70536 703483 471.548 Membrane receptor 52842,52842 52842,52842 Ki,Ki Ki,IC50 Butyrylcholinesterase 6.76955107862 5.81533639965 P06276 Q9JKC1 27251 250.337 Enzyme 21188,21519,30919,34898,36705,42047,48400 46056,49233 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50 Acetylcholinesterase 5.45025463739 5.66592356822 P22303 P37136 27251 250.337 Enzyme 21188,21519,30919,34898,36705,38283,42047,52762 46056,49233 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50 Serotonin transporter 7.538637271 6.56685633046 P31645 P31652 27278 277.402 Transporter 43754,51128 43754,49842 IC50,IC50 IC50,IC50 Dopamine transporter 5.52287874528 5.69897000434 Q01959 P23977 27342 255.355 Transporter 38698,38837,44487,45878,44158,44164,44914 45021 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Serotonin transporter 6.7447274949 5.82390874094 P31645 P31652 27342 255.355 Transporter 38698,38837,44487,45878,47195,44158,44164,44579,44898,44914 45021 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 Ki Cannabinoid CB1 receptor 8.26760624018 8.91009488856 P21554 P20272 551643 463.787 Membrane receptor 30590,49138,49138 30590 Ki,Ki,IC50 Ki Alpha-2a adrenergic receptor 7.24463368611 9.40893539297 P08913 P22909 27609 230.094 Membrane receptor 13831,15822 15822,15882 Ki,Ki Ki,Ki Nischarin 7.25963731051 6.43628166003 Q9Y2I1 Q4G017 27609 230.094 Cytosolic other 44014 45562 Ki IC50 Butyrylcholinesterase 5.07572071394 5.22914798836 P06276 Q9JKC1 27639 287.354 Enzyme 21519,30919,34898,36705,42156 46338 IC50,IC50,IC50,IC50,IC50 IC50 Acetylcholinesterase 6.09691001301 5.98494312365 P22303 P37136 27639 287.354 Enzyme 21519,30919,31012,34898,36705,42909,42156,49125,51286 40916,46338 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50 Nitric-oxide synthase, brain 5.14266750357 5.06048074738 P29475 P29476 27660 94.1145 Enzyme 46991 46991 IC50 IC50 Norepinephrine transporter 6.49430749259 6.48811663902 P23975 Q9WTR4 28068 272.408 Transporter 21634,21309,45802 16872 Ki,Ki,Ki Ki Dopamine transporter 6.2740883677 5.38090666937 Q01959 P23977 28068 272.408 Transporter 21309 37723 Ki Ki Serotonin transporter 8.8534845472 8.78251605579 P31645 P31652 28068 272.408 Transporter 21634,21309,30817,44082,44082,49772 16872,37723,45802,45802 Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki Norepinephrine transporter 6.01227306632 6.16557929632 P23975 Q9WTR4 28220 384.278 Transporter 21634,21309 16872 Ki,Ki Ki Serotonin transporter 9.928336435 10.1419983282 P31645 P31652 28220 384.278 Transporter 21634,21309 5371,16872 Ki,Ki Ki,Ki Corticotropin releasing factor receptor 1 8.72124639905 9.58502665203 P34998 P35353 559603 377.865 Membrane receptor 47379 47378,47379 IC50 IC50,IC50 Monoamine oxidase B 5.7447274949 5.44409999655 P27338 P19643 28477 159.228 Enzyme 30041 35878,45377,45377,44921 Ki IC50,Ki,IC50,IC50 Gonadotropin-releasing hormone receptor 7.46852108296 5.65757731918 P30968 P30969 29311 520.57 Membrane receptor 20737 17718 Ki Ki Serotonin 1a (5-HT1a) receptor 7.5376020021 7.72124639905 P08908 P19327 351101 470.604 Membrane receptor 31374 36406,46353 Ki Ki,Ki Gonadotropin-releasing hormone receptor 8.43179827593 5.10237290871 P30968 P30969 29782 553.572 Membrane receptor 42049 17718 Ki Ki Muscarinic acetylcholine receptor M3 8.98088868082 8.60205999133 P20309 P08483 291960 426.55 Membrane receptor 16845,30486 37711 Ki,Ki Ki Muscarinic acetylcholine receptor M2 7.31446606886 7.20065945055 P08172 P10980 291960 426.55 Membrane receptor 16845,30486 37711 Ki,Ki Ki Gonadotropin-releasing hormone receptor 8.21648681692 5.12493873661 P30968 P30969 29824 501.541 Membrane receptor 39564,39564 17718 Ki,IC50 Ki Gonadotropin-releasing hormone receptor 8.95860731484 5.19382002602 P30968 P30969 29833 524.534 Membrane receptor 42049 17718 Ki Ki Metabotropic glutamate receptor 4 6.25181197299 6.67778070527 Q14833 P31423 554348 242.273 Membrane receptor 47355 47355 IC50 IC50 Metabotropic glutamate receptor 4 5.95860731484 6.13076828027 Q14833 P31423 554358 262.692 Membrane receptor 47355 47355 IC50 IC50 Histamine H3 receptor 7.36957212497 6.07007043992 Q9Y5N1 Q9QYN8 554446 331.454 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.14996674231 6.2700257143 Q9Y5N1 Q9QYN8 554447 331.454 Membrane receptor 47387 47387 Ki Ki Serotonin transporter 6.83863199777 8.63078414259 P31645 P31652 554815 411.496 Transporter 47621 47621 IC50 Ki Neurokinin 1 receptor 9.13667713988 6.88605664769 P25103 P14600 30818 472.38 Membrane receptor 11880,38754,45287,47632,49287,52184 38754,45287,47632,49287 IC50,Ki,Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki Renin 8.15490195999 5.85387196432 P00797 P08424 555811 552.746 Enzyme 48265,48265 48265 IC50,IC50 IC50 Vasopressin V2 receptor 8.30102999566 6.50863830617 P30518 Q00788 293983 452.567 Membrane receptor 17861 17861 IC50 IC50 Histamine H3 receptor 9.26760624018 8.34008379993 Q9Y5N1 Q9QYN8 556181 303.401 Membrane receptor 47387 47387 Ki Ki Dihydrofolate reductase 3.95860731484 4.60205999133 P00374 Q920D2 556333 472.539 Enzyme 47416 47416 IC50 IC50 Vasopressin V2 receptor 7.52287874528 7.52287874528 P30518 Q00788 294295 482.593 Membrane receptor 17861 17861 IC50 IC50 Delta opioid receptor 10.7447274949 9.72124639905 P41143 P33533 556500 396.524 Membrane receptor 47540 47540 IC50 Ki Cannabinoid CB1 receptor 9.53786035697 8.55284196866 P21554 P20272 556582 510.418 Membrane receptor 45084,45084 45084 Ki,Ki Ki Vasopressin V2 receptor 7.30102999566 7.30102999566 P30518 Q00788 295235 586.746 Membrane receptor 17861 17861 IC50 IC50 Vasopressin V2 receptor 7.22184874962 6.42021640338 P30518 Q00788 295257 449.544 Membrane receptor 17861 17861 IC50 IC50 Alpha-1d adrenergic receptor 8.92081875395 8.97 P25100 P23944 33373 451.475 Membrane receptor 13032 47620 Ki IC50 Alpha-1b adrenergic receptor 9.13076828027 9.51 P35368 P15823 33373 451.475 Membrane receptor 13032 47620 Ki IC50 Alpha-1a adrenergic receptor 8.58502665203 8.69 P35348 P43140 33373 451.475 Membrane receptor 13032 47620 Ki IC50 Oxytocin receptor 8.01810608633 7.72124639905 P30559 P70536 33420 507.578 Membrane receptor 44053,52842 52842 Ki,Ki Ki Vasopressin V1a receptor 5.49485002168 8.43179827593 P37288 P30560 33420 507.578 Membrane receptor 52842 52842 Ki Ki Dopamine D2 receptor 6.64397414281 6.64397414281 P14416 P61169 557741 465.945 Membrane receptor 30625 17394 IC50 Ki Alpha-1d adrenergic receptor 6.95860731484 6.21395878976 P25100 P23944 33466 347.453 Membrane receptor 13032 13032 Ki Ki Histamine H3 receptor 8.30980391997 7.53017798402 Q9Y5N1 Q9QYN8 557790 303.401 Membrane receptor 47387 47387 Ki Ki Metabotropic glutamate receptor 4 6.61978875829 6.95860731484 Q14833 P31423 557815 262.692 Membrane receptor 47355 47355 IC50 IC50 Vasopressin V2 receptor 7.52287874528 7.69897000434 P30518 Q00788 295716 495.635 Membrane receptor 17861 17861 IC50 IC50 Histamine H3 receptor 6.93930215965 6.37986394503 Q9Y5N1 Q9QYN8 557877 345.477 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 6.25963731051 6.05012229596 Q9Y5N1 Q9QYN8 557918 303.401 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.0 6.17005330406 Q9Y5N1 Q9QYN8 557919 281.191 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.69036983257 6.34008379993 Q9Y5N1 Q9QYN8 557933 346.441 Membrane receptor 47387 47387 Ki Ki Histamine H1 receptor 7.32790214206 6.82390874094 P35367 P31390 33664 412.936 Membrane receptor 43952 39442 Ki IC50 Alpha-1d adrenergic receptor 8.44369749923 8.45593195565 P25100 P23944 33667 389.449 Membrane receptor 13032 13032 Ki Ki Alpha-1d adrenergic receptor 9.09691001301 8.8 P25100 P23944 33675 345.39 Membrane receptor 13032 13032,16909,30512 Ki Ki,IC50,IC50 Alpha-1b adrenergic receptor 8.0043648054 8.18 P35368 P15823 33675 345.39 Membrane receptor 13032 16909,30512 Ki IC50,IC50 Alpha-2a adrenergic receptor 8.45593195565 7.33724216832 P08913 P22909 33675 345.39 Membrane receptor 13032 13032 Ki Ki Alpha-1a adrenergic receptor 9.43179827593 9.51 P35348 P43140 33675 345.39 Membrane receptor 13032 16909,16909,30512 Ki IC50,IC50,IC50 Steroid 5-alpha-reductase 2 8.30102999566 7.95860731484 P31213 P31214 33679 372.544 Enzyme 14360,15700,16544 16544 IC50,IC50,IC50 IC50 Steroid 5-alpha-reductase 1 6.54575749056 8.0 P18405 P24008 33679 372.544 Enzyme 15700,14360 16544 IC50,Ki IC50 Neurokinin 1 receptor 11.9586073148 8.82390874094 P25103 P14600 558019 1327.33 Membrane receptor 47632 47632 Ki Ki Dopamine D3 receptor 8.86996430601 7.69464863055 P35462 P19020 33870 417.543 Membrane receptor 30313,31276,37020,45366 52373 Ki,Ki,Ki,Ki Ki Alpha-2a adrenergic receptor 8.56066730617 7.05060999336 P08913 P22909 33870 417.543 Membrane receptor 52373 17167 Ki Ki Serotonin 1a (5-HT1a) receptor 6.92548286642 8.30980391997 P08908 P19327 33870 417.543 Membrane receptor 31276,52373 17167 Ki,Ki Ki Delta opioid receptor 9.00438696215 8.8416375079 P41143 P33533 558225 358.476 Membrane receptor 47540,47540 47540 IC50,IC50 Ki Adenosine A3 receptor 7.88605664769 7.08196966322 P33765 P28647 558341 440.679 Membrane receptor 47561 47561 Ki Ki Adenosine A3 receptor 8.85387196432 9.06048074738 P33765 P28647 296217 488.924 Membrane receptor 39543 39543 Ki Ki Adenosine A3 receptor 9.16115090926 8.0 P33765 P28647 296226 518.995 Membrane receptor 39543 39543 Ki Ki Adenosine A3 receptor 8.44369749923 8.40893539297 P33765 P28647 296227 554.769 Membrane receptor 39543 39543 Ki Ki Adenosine A3 receptor 8.5376020021 8.79588001734 P33765 P28647 296233 482.92 Membrane receptor 39543 39543 Ki Ki Dopamine D3 receptor 7.34678748622 7.40893539297 P35462 P19020 34197 312.432 Membrane receptor 43952 16647 Ki Ki Histamine H1 receptor 8.55284196866 8.70446769649 P35367 P31390 34197 312.432 Membrane receptor 43952 16647,39442 Ki Ki,IC50 Dopamine D2 receptor 7.69897000434 7.55395269865 P14416 P61169 34197 312.432 Membrane receptor 43952,49693,49693 45067,51830 Ki,Ki,Ki Ki,Ki Dopamine D1 receptor 7.28399665637 7.65051499783 P21728 P18901 34197 312.432 Membrane receptor 43952 45067,51830 Ki Ki,Ki Serotonin 2a (5-HT2a) receptor 8.48148606012 8.39794000867 P28223 P14842 34197 312.432 Membrane receptor 43952 45067,51830 Ki Ki,Ki Serotonin 1a (5-HT1a) receptor 5.67778070527 6.21467016499 P08908 P19327 34197 312.432 Membrane receptor 43952 45067,51830 Ki Ki,Ki Metabotropic glutamate receptor 1 8.09691001301 7.85498269432 Q13255 P23385 296357 325.445 Membrane receptor 21599 21599,21599 IC50 IC50,IC50 Metabotropic glutamate receptor 1 7.2076083105 7.88605664769 Q13255 P23385 296370 423.288 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 6.75945075172 7.95860731484 Q13255 P23385 296371 322.401 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.04575749056 8.39794000867 Q13255 P23385 296376 315.382 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 5.19997064076 5.46495918675 Q13255 P23385 296391 383.481 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 9.0 8.15490195999 Q13255 P23385 296392 312.406 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.39794000867 7.56983099671 Q13255 P23385 296424 331.836 Membrane receptor 21599 21599,21599 IC50 IC50,IC50 Metabotropic glutamate receptor 1 7.36292107537 6.67324902652 Q13255 P23385 296428 327.417 Membrane receptor 21599,21599 21599,21599 IC50,IC50 IC50,IC50 Metabotropic glutamate receptor 1 5.36051351073 6.49485002168 Q13255 P23385 296437 341.447 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.15490195999 7.08092190762 Q13255 P23385 296458 333.38 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 7.77030375612 7.0 Q13255 P23385 296466 337.455 Membrane receptor 21599,21599 21599,21599 IC50,IC50 IC50,IC50 Metabotropic glutamate receptor 1 7.13076828027 8.15490195999 Q13255 P23385 296467 309.382 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.11716572262 7.93483311575 Q13255 P23385 296487 325.402 Membrane receptor 21599,21599 21599,21599 IC50,IC50 IC50,IC50 Metabotropic glutamate receptor 1 7.5376020021 8.09691001301 Q13255 P23385 296488 338.443 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 6.79588001734 7.07058107429 Q13255 P23385 296490 317.381 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 7.85387196432 8.22184874962 Q13255 P23385 296491 303.354 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 7.07058107429 7.79588001734 Q13255 P23385 296508 325.445 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 9.25181197299 8.39794000867 Q13255 P23385 296515 309.402 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.52287874528 8.30102999566 Q13255 P23385 296533 311.418 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.69897000434 8.69897000434 Q13255 P23385 296534 327.441 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 5.92996213339 7.25181197299 Q13255 P23385 296550 315.408 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 8.22184874962 8.15490195999 Q13255 P23385 296555 325.445 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 7.09691001301 7.30102999566 Q13255 P23385 296570 297.391 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 7.2924298239 8.0 Q13255 P23385 296571 289.371 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 7.07058107429 7.82390874094 Q13255 P23385 296575 313.391 Membrane receptor 21599 21599 IC50 IC50 Metabotropic glutamate receptor 1 6.34678748622 7.34678748622 Q13255 P23385 296576 338.404 Membrane receptor 21599 21599 IC50 IC50 Histamine H3 receptor 9.18326577221 8.55284196866 Q9Y5N1 Q9QYN8 558746 431.545 Membrane receptor 47928,47928 47928 IC50,Ki Ki Anandamide amidohydrolase 8.0 7.7447274949 O00519 P97612 296684 410.592 Enzyme 21573,21573,38830 38830,44028 Ki,IC50,Ki Ki,Ki Anandamide amidohydrolase 8.04575749056 8.32790214206 O00519 P97612 296748 334.412 Enzyme 21573,21573,38447,38830,44028,48011 36082,38493,38830,45114,44028,44028,44843,44843,45059,48011,48011,49095 Ki,IC50,IC50,Ki,Ki,IC50 Ki,IC50,Ki,Ki,Ki,Ki,Ki,IC50,Ki,IC50,IC50,Ki Anandamide amidohydrolase 9.5134360732 8.87236374745 O00519 P97612 296769 294.348 Enzyme 21573,38830 38830,49818 IC50,Ki Ki,IC50 Anandamide amidohydrolase 7.79588001734 10.5528419687 O00519 P97612 296770 308.374 Enzyme 21573,45059,45059,45059,45059 45059 IC50,IC50,IC50,IC50,IC50 Ki Cannabinoid CB1 receptor 8.85387196432 9.23657200644 P21554 P20272 559235 376.573 Membrane receptor 30511,36602,37845,39045,45320,45320,44149,44207,44207,45096,46425,50392,52442 39196,44207,46425 Ki,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,Ki,IC50,Ki Ki,IC50,Ki Cannabinoid CB2 receptor 9.07584384819 9.46852108296 P34972 Q9QZN9 559235 376.573 Membrane receptor 30511,30560,36602,37845,37845,39045,39045,39196,39196,44149,44149,44207,44207,45096,46425,52442 44207 Ki,Ki,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,Ki,IC50,IC50,IC50,Ki,Ki IC50 Corticotropin releasing factor receptor 1 8.30980391997 9.0 P34998 P35353 559570 424.657 Membrane receptor 47378 47378 IC50 IC50 Histamine H3 receptor 7.80966830183 6.83863199777 Q9Y5N1 Q9QYN8 559655 345.477 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.05012229596 6.69897000434 Q9Y5N1 Q9QYN8 559685 289.374 Membrane receptor 47387 47387 Ki Ki Gonadotropin-releasing hormone receptor 8.69897000434 5.63827216398 P30968 P30969 297647 559.359 Membrane receptor 20604 20604 Ki Ki Gonadotropin-releasing hormone receptor 7.7447274949 5.0268721464 P30968 P30969 297650 546.47 Membrane receptor 20604 20604 Ki Ki Histamine H3 receptor 8.76955107862 7.48148606012 Q9Y5N1 Q9QYN8 490011 431.451 Membrane receptor 43963,43963,43963 43963 IC50,Ki,IC50 Ki Serotonin transporter 5.67985371389 6.20551195334 P31645 P31652 35586 414.582 Transporter 15623 14301 Ki IC50 Serotonin 2a (5-HT2a) receptor 7.76955107862 7.93930215965 P28223 P14842 35617 244.332 Membrane receptor 17200 17200,17200,17200 Ki IC50,IC50,Ki Gonadotropin-releasing hormone receptor 7.88605664769 4.88605664769 P30968 P30969 297769 487.482 Membrane receptor 20604 20604 Ki Ki Serotonin 7 (5-HT7) receptor 8.05164872753 8.05164872753 P34969 P32305 35706 350.456 Membrane receptor 17066,17066 16372,16372 Ki,Ki Ki,Ki Serotonin 1a (5-HT1a) receptor 6.47836602931 4.97539098866 P08908 P19327 35706 350.456 Membrane receptor 16372,16372 38182,38182 Ki,Ki Ki,Ki Dopamine D2 receptor 5.95503685199 5.9515449935 P14416 P61169 35706 350.456 Membrane receptor 16372,16372 38182,38182 Ki,Ki Ki,Ki Adenosine A2a receptor 9.0 9.0 P29274 P30543 35757 412.482 Membrane receptor 15707,16115,16115 2252 Ki,IC50,Ki Ki Serotonin 2a (5-HT2a) receptor 8.08618614762 8.55284196866 P28223 P14842 35905 230.306 Membrane receptor 17200 17200,17200,17200 Ki IC50,IC50,Ki Adenosine A3 receptor 8.82390874094 8.95860731484 P33765 P28647 36005 554.769 Membrane receptor 39543,44562 39543 Ki,Ki Ki Adenosine A1 receptor 6.86646109163 7.07623803917 P30542 P25099 36005 554.769 Membrane receptor 39543,44562 39543 Ki,Ki Ki Adenosine A2a receptor 6.10568393732 5.77989191196 P29274 P30543 36005 554.769 Membrane receptor 39543,44562 39543 Ki,Ki Ki Monoglyceride lipase 6.0 5.72124639905 Q99685 Q8R431 560359 389.555 Enzyme 47831 47831 IC50 IC50 Serotonin 2a (5-HT2a) receptor 8.30980391997 8.7447274949 P28223 P14842 36132 216.279 Membrane receptor 17200 17200,17200,17200 Ki IC50,IC50,Ki Serotonin 1a (5-HT1a) receptor 6.90389474747 3.91634133263 P08908 P19327 36144 341.446 Membrane receptor 16372,16372 38182,38182 Ki,Ki Ki,Ki Adenosine A3 receptor 8.65757731918 6.79588001734 P33765 P28647 36146 352.776 Membrane receptor 39543 39543 Ki Ki Adenosine A1 receptor 5.67778070527 6.09420411963 P30542 P25099 36146 352.776 Membrane receptor 39543 39543 Ki Ki Serotonin 7 (5-HT7) receptor 8.00966114521 8.00966114521 P34969 P32305 36324 311.42 Membrane receptor 17066 16372 Ki Ki Serotonin 7 (5-HT7) receptor 7.7447274949 7.7447274949 P34969 P32305 36357 262.349 Membrane receptor 17066 16372 Ki Ki Serotonin 1a (5-HT1a) receptor 6.44977164694 6.44369749923 P08908 P19327 36357 262.349 Membrane receptor 16372 38182 Ki Ki Dopamine D2 receptor 5.64781748189 5.64781748189 P14416 P61169 36357 262.349 Membrane receptor 16372 38182 Ki Ki Histamine H3 receptor 8.5484550065 8.52287874528 Q9Y5N1 Q9QYN8 560871 372.524 Membrane receptor 48124,48124 48124 Ki,Ki Ki Histamine H3 receptor 8.76143937264 8.69897000434 Q9Y5N1 Q9QYN8 560885 414.561 Membrane receptor 48124,48124 48124 Ki,Ki Ki Androgen Receptor 8.73992861201 8.55284196866 P10275 P15207 36705 290.44 Transcription Factor 34749,34764,35644,35644,35972,35972,36333,36333,36717,36717,37738,38697,38697,38697,39522,39522,48062,48062,51594 34749,34764,45812 IC50,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50,IC50,Ki,IC50,IC50,Ki,IC50,IC50,Ki IC50,IC50,Ki Serotonin 7 (5-HT7) receptor 8.88605664769 8.89962945488 P34969 P32305 36730 352.492 Membrane receptor 17066 16372 Ki Ki Gonadotropin-releasing hormone receptor 8.76955107862 5.36877445513 P30968 P30969 299187 495.493 Membrane receptor 20414,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,30461,39564,45332,45332,42049 45332,42049 Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,Ki,IC50,Ki Ki,Ki Histamine H3 receptor 7.60032627852 7.03011835625 Q9Y5N1 Q9QYN8 561379 294.391 Membrane receptor 47387 47387 Ki Ki Metabotropic glutamate receptor 4 6.10790539731 6.43179827593 Q14833 P31423 561418 246.237 Membrane receptor 47355 47355 IC50 IC50 Metabotropic glutamate receptor 4 5.82390874094 6.0 Q14833 P31423 561426 284.209 Membrane receptor 47355 47355 IC50 IC50 Histamine H3 receptor 7.83863199777 7.34008379993 Q9Y5N1 Q9QYN8 561492 328.45 Membrane receptor 47387 47387 Ki Ki Neurokinin 1 receptor 9.06048074738 9.09691001301 P25103 P14600 37245 403.361 Membrane receptor 1477,13886 2360 IC50,IC50 IC50 Serotonin 1a (5-HT1a) receptor 8.29670862188 8.2924298239 P08908 P19327 37476 261.361 Membrane receptor 15874 38182 Ki Ki Serotonin 1a (5-HT1a) receptor 7.50723961097 7.50863830617 P08908 P19327 37553 261.361 Membrane receptor 15874 38182 Ki Ki Delta opioid receptor 10.2218487496 9.72124639905 P41143 P33533 561848 398.54 Membrane receptor 47540 47540 IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 8.09691001301 6.00877392431 P28845 P16232 561936 348.48 Enzyme 47580 47580 IC50 IC50 Serotonin 7 (5-HT7) receptor 8.32790214206 7.67778070527 P34969 P32305 299949 361.48 Membrane receptor 20615,36534,46399 20615 Ki,Ki,Ki Ki Serotonin 7 (5-HT7) receptor 8.26760624018 7.72124639905 P34969 P32305 300042 372.463 Membrane receptor 20615,36534 20615 Ki,Ki Ki Anandamide amidohydrolase 6.98088868082 6.13082340682 O00519 P97612 562466 420.332 Enzyme 48011,48011 48011,48011 IC50,IC50 IC50,IC50 Anandamide amidohydrolase 7.91009488856 5.43179827593 O00519 P97612 38208 356.465 Enzyme 48666 49818 IC50 IC50 Sodium channel protein type X alpha subunit 4.01772876696 4.60205999133 Q9Y5Y9 Q62968 38727 256.091 Ion channel 42188 42188 IC50 IC50 Sodium channel protein type II alpha subunit 5.0 4.45593195565 Q99250 P04775 38727 256.091 Ion channel 42188 49996 IC50 IC50 Histamine H3 receptor 7.87942606879 6.83863199777 Q9Y5N1 Q9QYN8 563105 278.391 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.97061622231 6.95078197733 Q9Y5N1 Q9QYN8 563112 296.382 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.25963731051 6.40011692793 Q9Y5N1 Q9QYN8 563211 343.465 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 7.79860287568 7.21968268786 Q9Y5N1 Q9QYN8 563219 289.374 Membrane receptor 47387 47387 Ki Ki Neurokinin 1 receptor 10.1135092748 7.85387196432 P25103 P14600 563307 1327.33 Membrane receptor 47632 47632 Ki Ki Neurokinin 1 receptor 10.2839966564 7.46852108296 P25103 P14600 563308 1438.51 Membrane receptor 47632 47632 Ki Ki Delta opioid receptor 10.3279021421 9.85387196432 P41143 P33533 563507 356.46 Membrane receptor 47540 47540 IC50 Ki Anandamide amidohydrolase 8.92081875395 9.5376020021 O00519 P97612 301697 335.4 Enzyme 44028 38830,44028,44028 Ki Ki,Ki,Ki Metabotropic glutamate receptor 1 6.95860731484 7.61978875829 Q13255 P23385 564196 366.496 Membrane receptor 48030 48030 Ki Ki Histamine H3 receptor 7.58004425151 6.8601209136 Q9Y5N1 Q9QYN8 564861 292.418 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 8.48945498979 7.65955588516 Q9Y5N1 Q9QYN8 564862 320.428 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 8.82102305271 7.6090648929 Q9Y5N1 Q9QYN8 564873 308.417 Membrane receptor 47387 47387 Ki Ki Histamine H3 receptor 8.17979854051 7.44977164694 Q9Y5N1 Q9QYN8 564967 317.427 Membrane receptor 47387 47387 Ki Ki Serotonin transporter 8.69250396209 5.97469413474 P31645 P31652 66613 193.242 Transporter 42172,42172,51535 50103 Ki,Ki,IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 8.09691001301 7.50863830617 P28845 P16232 565394 375.505 Enzyme 47580 47580 IC50 IC50 Dopamine D1 receptor 7.34678748622 6.15552282425 P21728 P18901 41198 279.376 Membrane receptor 44602 38182,38524,43841,45044 Ki Ki,Ki,Ki,Ki Gonadotropin-releasing hormone receptor 6.40893539297 6.16115090926 P30968 P30969 304426 437.53 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.76955107862 6.95860731484 P30968 P30969 304427 555.639 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 7.24412514433 7.2924298239 P30968 P30969 304428 605.647 Membrane receptor 20757 20757 IC50 IC50 Delta opioid receptor 8.79588001734 8.48168555232 P41143 P33533 42299 645.79 Membrane receptor 30746,31109,35601,35662,38101,38754,43854,44050,42904,45287,47632,47632,50978,52184 2703,2703,41786,52824 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,Ki IC50,IC50,IC50,Ki Gonadotropin-releasing hormone receptor 7.18045606446 7.2757241304 P30968 P30969 304445 575.629 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 8.3767507096 8.40893539297 P30968 P30969 304454 554.103 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.82390874094 7.10237290871 P30968 P30969 304468 523.622 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.16115090926 6.42021640338 P30968 P30969 304490 509.596 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 7.08092190762 7.30102999566 P30968 P30969 304491 592.083 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.92081875395 6.85387196432 P30968 P30969 304508 532.652 Membrane receptor 20756,20757,42049 20757 IC50,IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 7.32878865959 7.72184874962 P30968 P30969 304513 537.649 Membrane receptor 20757,20757 20757,20757 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 6.30980391997 6.50863830617 P30968 P30969 304516 519.658 Membrane receptor 20757 20757 IC50 IC50 Histamine H3 receptor 8.22988470521 7.40011692793 Q9Y5N1 Q9QYN8 566678 320.428 Membrane receptor 47387 47387 Ki Ki Gonadotropin-releasing hormone receptor 6.39794000867 6.63827216398 P30968 P30969 304558 536.661 Membrane receptor 20757 20757 IC50 IC50 Solute carrier family 22 member 12 5.47002905597 4.7447274949 Q96S37 Q3ZAV1 42426 302.236 NA 39400,39400 39400 IC50,Ki IC50 Metabotropic glutamate receptor 4 5.95860731484 6.5376020021 Q14833 P31423 566715 232.666 Membrane receptor 47355 47355 IC50 IC50 Metabotropic glutamate receptor 4 5.67778070527 5.76955107862 Q14833 P31423 566716 300.664 Membrane receptor 47355 47355 IC50 IC50 Gonadotropin-releasing hormone receptor 7.65757731918 7.85387196432 P30968 P30969 304593 588.548 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.13076828027 6.26760624018 P30968 P30969 304610 538.634 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.46852108296 6.69897000434 P30968 P30969 304618 549.684 Membrane receptor 20757 20757 IC50 IC50 Norepinephrine transporter 6.18837276973 6.07831352452 P23975 Q9WTR4 566765 277.334 Transporter 35284,35284 13641,13641,14202,12788,13096 IC50,Ki IC50,IC50,IC50,IC50,Ki Dopamine transporter 7.91583966724 7.74094052643 Q01959 P23977 566765 277.334 Transporter 35284,52167 13641,13641,3964,3964,14202,12788,16247,13096 IC50,Ki IC50,IC50,IC50,IC50,IC50,IC50,Ki,Ki Serotonin transporter 6.68027667804 6.11947231591 P31645 P31652 566765 277.334 Transporter 35284,35284 13641,13641,3964,3964,14202,12788,3964,3964 IC50,Ki IC50,IC50,IC50,IC50,IC50,IC50,Ki,Ki Gonadotropin-releasing hormone receptor 5.58502665203 6.07572071394 P30968 P30969 304633 536.661 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 5.72124639905 5.79588001734 P30968 P30969 304653 435.514 Membrane receptor 20757 20757 IC50 IC50 Neurokinin 1 receptor 11.5528419687 8.16749108729 P25103 P14600 566897 1191.27 Membrane receptor 47632 47632 Ki Ki Dopamine D2 receptor 7.38510278397 6.80410034759 P14416 P61169 567168 460.611 Membrane receptor 47595 47595 IC50 Ki Dopamine D3 receptor 8.91009488856 8.64397414281 P35462 P19020 567168 460.611 Membrane receptor 47595 47595 IC50 Ki Prostanoid EP1 receptor 7.38734535914 7.92081875395 P34995 P70597 305607 421.896 Membrane receptor 20789,20789 20789 Ki,Ki Ki Serotonin 2a (5-HT2a) receptor 8.33724216832 8.52775866392 P28223 P14842 43567 204.268 Membrane receptor 30538 17200,17200,17200,30538 Ki IC50,IC50,Ki,IC50 Histamine H3 receptor 8.57745097999 8.69897000434 Q9Y5N1 Q9QYN8 568042 428.587 Membrane receptor 48124,48124 48124 Ki,Ki Ki Metabotropic glutamate receptor 5 7.38721614328 8.51570016065 P41594 P31424 306526 275.368 Membrane receptor 20024 46751 IC50 IC50 Metabotropic glutamate receptor 5 9.30102999566 8.91721462968 P41594 P31424 306598 276.356 Membrane receptor 20024 46751 IC50 IC50 Dipeptidyl peptidase IV 7.58374554365 7.30980391997 P27487 P14740 438493 408.518 Enzyme 38801,38801 38801 IC50,IC50 IC50 P2X purinoceptor 7 8.0 8.0 Q99572 Q64663 569153 317.364 Ion channel 48423 48423 IC50 IC50 Alpha-2a adrenergic receptor 6.64975198167 8.52287874528 P08913 P22909 44885 202.275 Membrane receptor 15822 15822,15882 Ki Ki,Ki Alpha-2a adrenergic receptor 6.55752023094 8.58502665203 P08913 P22909 44977 200.26 Membrane receptor 15822 15822,15882 Ki Ki,Ki Alpha-2a adrenergic receptor 6.59516628338 8.82390874094 P08913 P22909 44978 202.275 Membrane receptor 15822 15822,15882 Ki Ki,Ki Alpha-2a adrenergic receptor 7.56863623584 9.25181197299 P08913 P22909 44979 204.291 Membrane receptor 15822 15822,15882 Ki Ki,Ki Serotonin transporter 7.55395269865 7.48148606012 P31645 P31652 400087 422.391 Transporter 36915,37465 37465 Ki,Ki Ki Metabotropic glutamate receptor 7 3.72584215074 3.51427857352 Q14831 P35400 45058 183.1 Membrane receptor 36453 36677,50682,50682 IC50 IC50,IC50,IC50 Metabotropic glutamate receptor 4 6.79588001734 6.84096833252 Q14833 P31423 45058 183.1 Membrane receptor 45031 30522,36453,36453,36677,50682,50682 Ki Ki,IC50,Ki,IC50,IC50,IC50 Alpha-2a adrenergic receptor 7.60205999133 11.0655015488 P08913 P22909 45217 230.329 Membrane receptor 15822 15822,15882 Ki Ki,Ki Acetylcholinesterase 7.12493873661 7.07058107429 P22303 P37136 569640 191.291 Enzyme 48391 48391 IC50 IC50 Acetylcholinesterase 6.40671393298 6.44129142947 P22303 P37136 569645 253.36 Enzyme 48391 48391 IC50 IC50 Acetylcholinesterase 6.43415218133 6.44129142947 P22303 P37136 569646 267.387 Enzyme 48391 48391 IC50 IC50 Acetylcholinesterase 6.7328282716 6.70996538864 P22303 P37136 570210 298.358 Enzyme 48391 48391 IC50 IC50 Acetylcholinesterase 5.93930215965 5.92081875395 P22303 P37136 570212 298.358 Enzyme 48391 48391 IC50 IC50 Adenosine A3 receptor 8.62342304294 7.1771783547 P33765 P28647 570475 538.983 Membrane receptor 48662 48662 Ki Ki Dipeptidyl peptidase IV 6.85387196432 6.10790539731 P27487 P14740 308440 297.315 Enzyme 45969 45969 IC50 IC50 Serotonin 4 (5-HT4) receptor 8.30102999566 8.97061622231 Q13639 Q62758 46814 312.792 Membrane receptor 30200,36639,36639,46295,46295 809 Ki,Ki,Ki,Ki,IC50 Ki Dihydrofolate reductase 5.07058107429 7.24412514433 P00374 Q920D2 47163 340.38 Enzyme 13858 45205 IC50 IC50 Dihydrofolate reductase 4.88605664769 6.45593195565 P00374 Q920D2 47403 326.353 Enzyme 13858 45205 IC50 IC50 Mu opioid receptor 8.20065945055 7.43483311575 P35372 P33535 572021 414.496 Membrane receptor 17097,17097,35310,46432,48048 14517,6070,46044,47540 IC50,Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki Delta opioid receptor 9.69897000434 9.5376020021 P41143 P33533 572021 414.496 Membrane receptor 17097,17097,16664,35310,46432,46432,48048 14517,14517,14517,6070,46044,47540,48048 IC50,Ki,Ki,Ki,Ki,IC50,Ki Ki,Ki,Ki,Ki,Ki,Ki,Ki Kappa opioid receptor 7.99567862622 7.52287874528 P41145 P34975 572021 414.496 Membrane receptor 17097,17097,35310,46432,48048 46044 Ki,IC50,Ki,Ki,Ki Ki Vasopressin V1b receptor 5.94423953531 5.48891915446 P47901 P48974 572188 572.182 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 5.98464024459 5.40439356513 P47901 P48974 572189 608.235 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.38404994834 6.25414480483 P47901 P48974 572206 577.756 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 9.22184874962 9.0 P47901 P48974 572209 630.108 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 7.18045606446 7.63827216398 P47901 P48974 572250 619.816 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 7.01772876696 6.83863199777 P47901 P48974 572251 619.816 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.9829666607 7.08092190762 P47901 P48974 572252 613.788 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.6615435064 6.80134291305 P47901 P48974 572253 631.778 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.02733440773 6.19586056766 P47901 P48974 572254 643.814 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.55439579673 6.56863623584 P47901 P48974 572255 643.814 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.14448084433 6.00043451177 P47901 P48974 572256 627.814 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 5.14290884533 5.01831727263 P47901 P48974 572264 530.145 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.22184874962 6.08990945441 P47901 P48974 572280 594.209 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.81815641206 6.64397414281 P47901 P48974 572281 565.745 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 5.92664829761 5.55658053822 P47901 P48974 572318 544.171 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 6.12609840214 5.57024772 P47901 P48974 572363 580.182 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 7.45593195565 7.56863623584 P47901 P48974 572364 593.798 Membrane receptor 48483 48483 Ki Ki Vasopressin V1b receptor 7.10790539731 7.2076083105 P47901 P48974 572365 577.756 Membrane receptor 48483 48483 Ki Ki Corticotropin releasing factor receptor 1 8.72124639905 9.06550154876 P34998 P35353 572860 425.817 Membrane receptor 48629 48629 IC50 IC50 Oxytocin receptor 8.56863623584 9.05060999336 P30559 P70536 48705 1007.19 Membrane receptor 36382 10675 IC50 Ki Vasopressin V2 receptor 5.45593195565 7.13509374642 P30518 Q00788 48705 1007.19 Membrane receptor 16468 10675,10675 Ki Ki,Ki Dihydrofolate reductase 7.65757731918 8.60205999133 P00374 Q920D2 49931 454.439 Enzyme 15984,13858,21405,30626,35323,35335,35353,36076,36100,38127,38176,43976,41861,45252,46340,47619,49279,49957,50832,50606 17126,14893,49279 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,Ki,IC50,IC50,IC50 IC50,IC50,Ki Adenosine A1 receptor 5.0 5.95860731484 P30542 P25099 312150 482.85 Membrane receptor 21051 35271 Ki Ki Adenosine A2a receptor 7.0 7.85387196432 P29274 P30543 312150 482.85 Membrane receptor 21051 35271 Ki Ki Adenosine A3 receptor 8.67778070527 8.06148027482 P33765 P28647 574305 595.092 Membrane receptor 48662 48662 Ki Ki Adenosine A3 receptor 8.36352252758 8.01682492796 P33765 P28647 574309 1126.78 Membrane receptor 48662,48662 48662 Ki,IC50 Ki Adenosine A3 receptor 8.30980391997 7.69250396209 P33765 P28647 574313 371.821 Membrane receptor 48662 48662 Ki Ki Bradykinin B1 receptor 10.4443687432 6.786482243 P46663 P97583 312179 586.49 Membrane receptor 20349,31083,31083,31083,31083,31083,44181,44181,52840,52840 52840 Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,IC50 IC50 Rho-associated protein kinase 2 6.55395269865 6.09691001301 O75116 Q62868 50239 247.336 Enzyme 49811,49811 52567 Ki,IC50 IC50 Adenosine A3 receptor 8.92693598216 9.48148606012 P33765 P28647 312680 544.731 Membrane receptor 17161,20156 17161,6127 Ki,Ki Ki,Ki Adenosine A1 receptor 6.28011267019 6.08618614762 P30542 P25099 312680 544.731 Membrane receptor 17161,20156 17161,14546 Ki,Ki Ki,Ki Adenosine A2a receptor 5.27083521031 6.32790214206 P29274 P30543 312680 544.731 Membrane receptor 17161,20156 17161,14546 Ki,Ki Ki,Ki Rho-associated protein kinase 2 6.18045606446 5.72124639905 O75116 Q62868 50822 291.369 Enzyme 49811 52567 IC50 IC50 Anandamide amidohydrolase 7.5618910797 7.99740974375 O00519 P97612 312994 338.4 Enzyme 45322,45059,45059,45059,45059,48011 31306,45114,42205,45059,47831,48011,48011,49818 IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50 Monoamine oxidase B 7.69897000434 5.8696662315 P27338 P19643 96021 187.281 Enzyme 30041,47084,44148,44874,46413,49935,50304,51147,52183,52379,52782,52818,52882 11483,45377,45377,44921,49220,49220,49443 Ki,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,Ki,IC50,IC50,IC50,Ki,Ki Monoamine oxidase A 4.17230771133 3.97608939365 P21397 P21396 96021 187.281 Enzyme 47084,44148,44874,46413,48800,49935,50304,51147,52183,52379,52782,52818,52882 11483,45377,45377,44921,49220,49220,49443 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,Ki,IC50,IC50,Ki,Ki Cannabinoid CB1 receptor 10.0 8.7447274949 P21554 P20272 576353 521.868 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.04575749056 8.24412514433 P21554 P20272 576361 459.799 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.11918640772 8.2757241304 P21554 P20272 576404 411.327 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.32790214206 8.06550154876 P21554 P20272 576416 485.836 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.30102999566 8.0 P21554 P20272 576430 457.783 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.04575749056 8.30980391997 P21554 P20272 576437 445.772 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 10.0 8.95860731484 P21554 P20272 576438 487.423 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.10237290871 8.13076828027 P21554 P20272 576446 409.311 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.42021640338 7.72124639905 P21554 P20272 576447 445.343 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.28399665637 8.02227639471 P21554 P20272 576453 445.772 Membrane receptor 48905 48905 Ki Ki Cannabinoid CB1 receptor 8.02227639471 8.14266750357 P21554 P20272 576466 445.772 Membrane receptor 48905 48905 Ki Ki Serotonin 2a (5-HT2a) receptor 9.13667713988 9.12493873661 P28223 P14842 358277 272.138 Membrane receptor 31732 31732 Ki Ki Serotonin transporter 8.3622291558 8.34678748622 P31645 P31652 401995 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Adenosine A3 receptor 7.37365963262 6.62525165399 P33765 P28647 52938 369.803 Membrane receptor 6714,30314,38198 15464,30314 Ki,Ki,Ki Ki,Ki Adenosine A1 receptor 9.08092190762 9.05395269865 P30542 P25099 52938 369.803 Membrane receptor 17473,6714,30314,38198,45180 10854,13048 IC50,Ki,Ki,Ki,Ki Ki,Ki Adenosine A2a receptor 5.64397414281 6.20266563435 P29274 P30543 52938 369.803 Membrane receptor 6714,30314,38198 15464,13048 Ki,Ki,Ki Ki,Ki Serotonin transporter 6.62708799703 7.40893539297 P31645 P31652 438226 397.486 Transporter 38371 38371 Ki Ki Anandamide amidohydrolase 9.48148606012 7.63827216398 O00519 P97612 183694 370.482 Enzyme 48666 49818 IC50 IC50 Kappa opioid receptor 8.64878473178 7.75696195131 P41145 P34975 316021 432.464 Membrane receptor 31702,31702,34894,37097,38874,38874,39419,39419,39419,45669,45669,42671,42671,53086 35985,35985,38503 Ki,Ki,Ki,IC50,Ki,IC50,Ki,Ki,IC50,Ki,IC50,IC50,IC50,IC50 Ki,Ki,Ki Lysophosphatidic acid receptor Edg-2 6.2924298239 6.79588001734 Q92633 P61794 316115 474.957 Membrane receptor 37582 37582 IC50 IC50 Metabotropic glutamate receptor 5 7.52287874528 6.65086271166 P41594 P31424 317037 353.416 Membrane receptor 21179 31236,31236 IC50 Ki,IC50 Cannabinoid CB2 receptor 9.01322826573 10.15490196 P34972 Q9QZN9 579544 354.443 Membrane receptor 49092,49092,49092 49092 Ki,IC50,IC50 IC50 Vasopressin V2 receptor 10.2839966564 9.34678748622 P30518 Q00788 55330 1084.23 Membrane receptor 30695 35041 IC50 Ki Vasopressin V1a receptor 8.9164891021 8.81247927916 P37288 P30560 55330 1084.23 Membrane receptor 36698,36698,36698,36698,36698,36698,36698,36698 35041 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki Cannabinoid CB1 receptor 5.78919803657 5.75448733219 P21554 P20272 55384 395.577 Membrane receptor 30511,44808 13682 Ki,Ki Ki Endothelin receptor ET-A 4.12493873661 3.39794000867 P25101 P26684 446141 430.491 Membrane receptor 41260 41260 IC50 IC50 Anandamide amidohydrolase 6.52287874528 7.0 O00519 P97612 55550 333.508 Enzyme 21573,21573 4252,38830,44028 Ki,IC50 Ki,Ki,Ki Dopamine D2 receptor 6.75289486539 6.57024772 P14416 P61169 579864 450.643 Membrane receptor 49130,49130 52843 Ki,IC50 Ki Dopamine D3 receptor 8.96784589666 8.65169513695 P35462 P19020 579864 450.643 Membrane receptor 49130,49130 52843 Ki,IC50 Ki Anandamide amidohydrolase 6.06833856994 6.62785350844 O00519 P97612 55597 383.567 Enzyme 21573,38830 4252,38830 IC50,Ki Ki,Ki Niemann-Pick C1-like protein 1 8.39794000867 8.39794000867 Q9UHC9 Q6T3U3 580274 701.647 Membrane other 48809,48809 48809,48809 IC50,IC50 IC50,IC50 Niemann-Pick C1-like protein 1 6.76143937264 6.82907508796 Q9UHC9 Q6T3U3 580275 571.543 Membrane other 48809,48809 48809,48809 IC50,IC50 IC50,IC50 Cholecystokinin A receptor 6.71547113441 7.23709678856 P32238 P30551 708487 605.64 Membrane receptor 53436,53436 53436,53436 IC50,IC50 IC50,IC50 Urotensin II receptor 6.79588001734 6.88605664769 Q9UKP6 P49684 580910 499.601 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.50863830617 6.7447274949 Q9UKP6 P49684 580918 513.627 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.15490195999 6.52287874528 Q9UKP6 P49684 580919 514.615 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.36653154442 6.92081875395 Q9UKP6 P49684 580920 614.731 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.5376020021 7.12493873661 Q9UKP6 P49684 580921 660.803 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.26760624018 6.95860731484 Q9UKP6 P49684 580922 628.758 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.56863623584 6.92081875395 Q9UKP6 P49684 580923 674.829 Membrane receptor 48952 48952 Ki IC50 Cholecystokinin A receptor 6.74879668304 7.0690536548 P32238 P30551 708490 600.666 Membrane receptor 53436,53436 53436,53436 IC50,IC50 IC50,IC50 Urotensin II receptor 6.50863830617 6.0 Q9UKP6 P49684 580930 507.528 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.79588001734 6.82390874094 Q9UKP6 P49684 580946 471.548 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 5.98268577169 7.07572071394 Q9UKP6 P49684 580957 485.574 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 5.49485002168 6.69897000434 Q9UKP6 P49684 580958 542.669 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.69897000434 6.69897000434 Q9UKP6 P49684 580959 642.784 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.96479633913 7.5376020021 Q9UKP6 P49684 580962 688.856 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 5.85387196432 6.95860731484 Q9UKP6 P49684 580964 620.759 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.5624693683 7.39794000867 Q9UKP6 P49684 580988 584.707 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.1399203483 8.31875876262 Q9UKP6 P49684 580990 612.76 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.08534811358 8.45593195565 Q9UKP6 P49684 580991 626.787 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.19045333469 7.69897000434 Q9UKP6 P49684 580992 687.805 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 6.50262152771 7.95860731484 Q9UKP6 P49684 580993 651.751 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.60697939488 7.95860731484 Q9UKP6 P49684 580994 700.847 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.24613951166 7.95860731484 Q9UKP6 P49684 580995 664.793 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.22672866826 7.85387196432 Q9UKP6 P49684 580996 700.847 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 8.24742501084 9.0 Q9UKP6 P49684 580998 598.776 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.83683206954 8.52287874528 Q9UKP6 P49684 580999 612.803 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 6.50863830617 7.15490195999 Q9UKP6 P49684 581014 499.601 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.63827216398 6.82390874094 Q9UKP6 P49684 581025 499.601 Membrane receptor 48952 48952 Ki IC50 Urotensin II receptor 6.69897000434 8.49485002168 Q9UKP6 P49684 319196 450.401 Membrane receptor 43815,43815,51448,51448 51448 Ki,IC50,Ki,Ki Ki Fructose-1,6-bisphosphatase 6.7447274949 5.88605664769 P09467 P19112 581633 447.372 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.04575749056 5.69897000434 P09467 P19112 581634 463.826 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.60205999133 4.69897000434 P09467 P19112 581641 375.359 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.39794000867 4.69897000434 P09467 P19112 581648 375.339 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.0 5.642065153 P09467 P19112 581649 353.285 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.25963731051 6.25963731051 P09467 P19112 581650 381.339 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.48811663902 4.69897000434 P09467 P19112 581664 389.385 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.82390874094 6.07058107429 P09467 P19112 581665 381.339 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.25963731051 5.6615435064 P09467 P19112 581674 351.269 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.0 6.18708664336 P09467 P19112 581675 395.365 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.30102999566 4.69897000434 P09467 P19112 581683 369.311 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.02227639471 4.69897000434 P09467 P19112 581684 425.417 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.0 5.69897000434 P09467 P19112 581685 493.087 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.34678748622 5.69897000434 P09467 P19112 581686 404.185 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.60205999133 4.69897000434 P09467 P19112 581691 363.348 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.52287874528 4.69897000434 P09467 P19112 581692 377.375 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.15490195999 5.69897000434 P09467 P19112 581693 365.321 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.67778070527 5.79588001734 P09467 P19112 581694 437.445 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.30102999566 4.69897000434 P09467 P19112 581702 351.294 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.0 5.67778070527 P09467 P19112 581703 437.445 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.64781748189 4.39794000867 P09467 P19112 581709 307.242 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.95860731484 5.69897000434 P09467 P19112 581730 321.268 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.82390874094 5.39794000867 P09467 P19112 581731 335.295 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.88605664769 5.67985371389 P09467 P19112 581732 432.181 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.64781748189 5.69897000434 P09467 P19112 581733 387.73 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.09691001301 4.69897000434 P09467 P19112 581742 333.279 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.15490195999 4.69897000434 P09467 P19112 581743 437.309 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.69897000434 5.69897000434 P09467 P19112 581744 369.74 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.09691001301 5.69897000434 P09467 P19112 581749 347.306 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.60205999133 4.69897000434 P09467 P19112 581750 445.407 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.04575749056 5.69897000434 P09467 P19112 581751 369.74 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.55284196866 6.04575749056 P09467 P19112 581763 379.323 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.09691001301 6.34678748622 P09467 P19112 581764 411.364 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.3767507096 4.69897000434 P09467 P19112 581771 359.273 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.25963731051 6.39794000867 P09467 P19112 581773 438.433 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.15490195999 6.30102999566 P09467 P19112 581774 443.837 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 5.82390874094 5.69897000434 P09467 P19112 581782 361.332 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 7.04575749056 6.04575749056 P09467 P19112 581784 429.381 Enzyme 49142 49142 IC50 IC50 Melanin-concentrating hormone receptor 1 7.88477553931 8.05551732785 Q99705 P97639 582361 494.533 Membrane receptor 48902,48902 48902 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.88605664769 7.88605664769 P34972 Q9QZN9 582409 331.452 Membrane receptor 48957 48957 Ki IC50 Cannabinoid CB2 receptor 8.15490195999 8.05551732785 P34972 Q9QZN9 582410 345.479 Membrane receptor 48957 48957 Ki IC50 Cannabinoid CB2 receptor 8.72124639905 8.55284196866 P34972 Q9QZN9 582441 345.479 Membrane receptor 48957 48957 Ki IC50 Urotensin II receptor 7.29929972961 8.15490195999 Q9UKP6 P49684 582480 562.723 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.48693774163 8.22184874962 Q9UKP6 P49684 582489 548.739 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.05551732785 8.15490195999 Q9UKP6 P49684 582490 612.803 Membrane receptor 48952 48952 IC50 IC50 Urotensin II receptor 6.84851003163 7.40893539297 Q9UKP6 P49684 582506 584.75 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.12981865525 8.69897000434 Q9UKP6 P49684 582508 626.83 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 6.57498337116 7.88605664769 Q9UKP6 P49684 582509 624.814 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 6.82448857371 8.39794000867 Q9UKP6 P49684 582510 638.84 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.42233198127 7.79588001734 Q9UKP6 P49684 582511 574.714 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 7.44724490762 7.63827216398 Q9UKP6 P49684 582513 582.714 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Cannabinoid CB2 receptor 7.61978875829 7.38721614328 P34972 Q9QZN9 582523 305.415 Membrane receptor 48957 48957 Ki IC50 Cannabinoid CB2 receptor 7.1739251973 6.58502665203 P34972 Q9QZN9 582532 305.415 Membrane receptor 48957 48957 Ki IC50 Urotensin II receptor 7.65225916175 8.39794000867 Q9UKP6 P49684 582545 560.687 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Cannabinoid CB2 receptor 8.10237290871 8.01772876696 P34972 Q9QZN9 582547 319.442 Membrane receptor 48957 48957 Ki IC50 Cannabinoid CB2 receptor 7.09151498112 7.15490195999 P34972 Q9QZN9 582584 291.389 Membrane receptor 48957 48957 Ki IC50 Urotensin II receptor 7.19382002602 8.02726570743 Q9UKP6 P49684 582611 435.559 Membrane receptor 48952,51448,51448 48952,51448 Ki,Ki,Ki IC50,Ki Cannabinoid CB2 receptor 8.2757241304 8.38721614328 P34972 Q9QZN9 582615 319.442 Membrane receptor 48957 48957 Ki IC50 Cannabinoid CB2 receptor 7.34678748622 6.85387196432 P34972 Q9QZN9 582617 317.426 Membrane receptor 48957 48957 Ki IC50 Mu opioid receptor 8.0 7.43179827593 P35372 P33535 58836 513.586 Membrane receptor 37896,39273,39273,39419,43854,45320,45320,44050,42044,46647,45005,46432 2703,30746,31109,36495,38119,38754,43813,45287,47632,49184,49287,49287,52184,52184,52824 IC50,IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50,Ki,IC50,Ki,IC50,Ki Delta opioid receptor 9.18045606446 5.85597716389 P41143 P33533 58836 513.586 Membrane receptor 49287 36495,52824 Ki IC50,Ki Matrix metalloproteinase 13 9.07572071394 5.14266750357 P45452 P23097 368760 538.508 Enzyme 34887 34887 IC50 IC50 Metabotropic glutamate receptor 5 6.35457773065 6.29417331455 P41594 P31424 359473 350.437 Membrane receptor 31805,35368 31805,35368 IC50,IC50 IC50,Ki Metabotropic glutamate receptor 1 8.52287874528 8.30102999566 Q13255 P23385 359473 350.437 Membrane receptor 31805,35368 31805,35368,44256 IC50,IC50 IC50,Ki,IC50 Neprilysin 8.04575749056 8.04575749056 P08473 P07861 59756 408.535 Enzyme 49077 4050 Ki IC50 Cannabinoid CB1 receptor 6.64589156085 7.1771783547 P21554 P20272 446975 460.439 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.35556141053 6.73048705578 P21554 P20272 446988 480.858 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.13727247168 7.04963514562 P21554 P20272 446989 494.884 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 7.72124639905 6.9829666607 P21554 P20272 447017 480.858 Membrane receptor 42580,50392,50392 42580 IC50,Ki,IC50 IC50 Vanilloid receptor 7.31678852139 6.79857710917 Q8NER1 O35433 323063 337.412 Ion channel 38185,38185 36134,36134,38185,38185 IC50,IC50 IC50,IC50,IC50,IC50 Histamine H3 receptor 8.2700257143 7.61083391564 Q9Y5N1 Q9QYN8 323303 356.588 Membrane receptor 44314,47387 38812,44314,47387 Ki,Ki Ki,Ki,Ki Adenosine A2a receptor 7.92081875395 7.63827216398 P29274 P30543 709246 420.464 Membrane receptor 53459 53459 Ki Ki Vanilloid receptor 7.88605664769 7.45593195565 Q8NER1 O35433 323453 324.397 Ion channel 38526 38526 IC50 IC50 Serotonin transporter 7.43179827593 7.79588001734 P31645 P31652 438496 433.467 Transporter 38371 38371 Ki Ki Anandamide amidohydrolase 7.42829116819 7.92081875395 O00519 P97612 447268 307.35 Enzyme 48666 45322,42654,45059 IC50 IC50,IC50,Ki Adenosine A3 receptor 9.42021640338 9.11918640772 P33765 P28647 324339 507.768 Membrane receptor 39543 39543 Ki Ki Serotonin 2b (5-HT2b) receptor 8.36653154442 8.49 P41595 P30994 62720 292.335 Membrane receptor 53923 13735,12936 Ki IC50,IC50 Vitamin D receptor 9.0484550065 9.69897000434 P11473 P13053 63252 416.636 Transcription Factor 34758,35163,37132,38881,38881,38881,39177,39177,46249,46249 37189,37189,39177,46705,44545,44545,45922,45922,49330,49330 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,Ki,Ki,IC50,Ki,IC50,Ki,IC50 Sodium channel protein type X alpha subunit 8.0 6.88605664769 Q9Y5Y9 Q62968 709229 407.893 Ion channel 53444 53444 IC50 IC50 Serotonin transporter 7.55284196866 7.7447274949 P31645 P31652 438630 397.511 Transporter 38371 38371 Ki Ki Neuropeptide Y receptor type 5 9.16115090926 8.88605664769 Q15761 Q63634 501480 423.849 Membrane receptor 46791 46791 IC50 IC50 Metabotropic glutamate receptor 5 7.72124639905 6.71229060439 P41594 P31424 316795 407.388 Membrane receptor 21179 31236,31236 IC50 Ki,IC50 Cannabinoid CB2 receptor 7.85387196432 5.85387196432 P34972 Q9QZN9 590136 394.528 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 8.04575749056 7.65757731918 P34972 Q9QZN9 590143 380.545 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 8.07572071394 7.69897000434 P34972 Q9QZN9 590149 416.555 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 7.04575749056 7.13667713988 P34972 Q9QZN9 590154 368.491 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 7.18045606446 6.8696662315 P34972 Q9QZN9 590156 352.492 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 7.36653154442 7.00877392431 P34972 Q9QZN9 590172 382.517 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 8.16115090926 7.92081875395 P34972 Q9QZN9 590177 370.53 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 7.92081875395 5.76955107862 P34972 Q9QZN9 590179 380.502 Membrane receptor 49415 49415 Ki IC50 Serotonin transporter 5.85387196432 6.55752023094 P31645 P31652 66246 271.354 Transporter 44487,44158,44579 45021 IC50,IC50,IC50 Ki Serotonin 6 (5-HT6) receptor 6.75956553816 6.92445303861 P50406 P31388 590783 319.443 Membrane receptor 49446,50854,50854,50854 50854 IC50,Ki,Ki,IC50 Ki Calcitonin gene-related peptide type 1 receptor 6.79948500217 4.15181088301 Q16602 Q63118 328724 789.557 Membrane receptor 30176,30176 30176 IC50,IC50 IC50 Calcitonin gene-related peptide type 1 receptor 9.89948500217 7.24641694111 Q16602 Q63118 328729 855.619 Membrane receptor 30176,30176 30176 IC50,IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 4.92922353716 6.99139982824 P36544 Q05941 591009 391.897 Ion channel 49457 49457 IC50 Ki Delta opioid receptor 8.32697909287 6.73518217699 P41143 P33533 66780 783.868 Membrane receptor 16024 11019 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 4.8894102897 7.3767507096 P36544 Q05941 591079 387.478 Ion channel 49457 49457 IC50 Ki Serotonin transporter 8.08092190762 8.11350927483 P31645 P31652 329090 323.353 Transporter 37541 37541 Ki Ki C5a anaphylatoxin chemotactic receptor 6.22184874962 5.50863830617 P21730 P97520 591363 371.473 Membrane receptor 49491,49491,49491 49491 IC50,IC50,IC50 IC50 Serotonin 2a (5-HT2a) receptor 7.69897000434 7.69897000434 P28223 P14842 67202 209.286 Membrane receptor 45779,49240 4664 Ki,Ki Ki Corticotropin releasing factor receptor 1 8.76955107862 8.64878473178 P34998 P35353 67244 410.298 Membrane receptor 15791 47072,47378 Ki IC50,IC50 Nitric-oxide synthase, brain 7.30102999566 8.15490195999 P29475 P29476 592050 372.48 Enzyme 53397 53397 Ki Ki Glucagon receptor 7.65428242393 7.63827216398 P47871 P30082 330027 563.608 Membrane receptor 30062,45153 45153 IC50,IC50 IC50 Gastric inhibitory polypeptide receptor 7.54821356448 7.3767507096 P48546 P43219 330027 563.608 Membrane receptor 45153 45153 IC50 IC50 Metabotropic glutamate receptor 5 7.30102999566 6.26916071495 P41594 P31424 317154 364.399 Membrane receptor 21179,54098 31236,31236 IC50,Ki Ki,IC50 Metabotropic glutamate receptor 5 7.39794000867 6.03566384016 P41594 P31424 317192 339.39 Membrane receptor 21179 31236,31236 IC50 Ki,IC50 Metabotropic glutamate receptor 5 7.42021640338 7.52287874528 P41594 P31424 592470 358.865 Membrane receptor 49423,49423,49423 49423 IC50,IC50,Ki Ki Sodium channel protein type X alpha subunit 7.19382002602 6.2924298239 Q9Y5Y9 Q62968 710455 386.367 Ion channel 53444 53444 IC50 IC50 Renin 7.84391132178 5.0 P00797 P08424 331011 675.879 Enzyme 9146,9146 9146 IC50,IC50 IC50 Neuropeptide Y receptor type 5 8.35654732351 8.76955107862 Q15761 Q63634 593355 388.419 Membrane receptor 49253 49253 IC50 IC50 Neuropeptide Y receptor type 5 9.03621217265 8.67778070527 Q15761 Q63634 593357 406.41 Membrane receptor 49253 49253 IC50 IC50 Neuropeptide Y receptor type 5 8.63827216398 8.65757731918 Q15761 Q63634 593415 388.419 Membrane receptor 49253 49253 IC50 IC50 Serotonin transporter 6.17979854051 5.28399665637 P31645 P31652 593611 313.391 Transporter 45054 44451 Ki IC50 Cannabinoid CB1 receptor 5.72561120445 5.68256350346 P21554 P20272 579539 313.434 Membrane receptor 49092 49092 IC50 IC50 Cannabinoid CB2 receptor 8.65757731918 8.35654732351 P34972 Q9QZN9 579539 313.434 Membrane receptor 49092,49092,49092 49092 Ki,IC50,IC50 IC50 Adenosine A3 receptor 7.88272870434 7.99139982824 P33765 P28647 331595 372.422 Membrane receptor 30314 30314 Ki Ki Adenosine A3 receptor 8.43179827593 8.23657200644 P33765 P28647 331610 406.867 Membrane receptor 30314 30314 Ki Ki Adenosine A1 receptor 7.73754891027 7.75945075172 P30542 P25099 331610 406.867 Membrane receptor 30314 30314 Ki Ki Adenosine A3 receptor 7.83564714422 8.01772876696 P33765 P28647 331611 432.904 Membrane receptor 30314 30314 Ki Ki Anandamide amidohydrolase 7.64199832818 8.63827216398 O00519 P97612 54688 384.555 Enzyme 21573,38830 4252,38830 IC50,Ki Ki,Ki Adenosine A3 receptor 6.64016451766 6.98716277529 P33765 P28647 331688 361.396 Membrane receptor 30314 30314 Ki Ki Sodium channel protein type X alpha subunit 8.04575749056 7.06048074738 Q9Y5Y9 Q62968 710668 336.815 Ion channel 53444 53444 IC50 IC50 Dihydrofolate reductase 5.29051808465 5.03503521996 P00374 Q920D2 594518 296.324 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 4.47407658084 4.81585655755 P00374 Q920D2 594519 340.419 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Neurokinin 1 receptor 9.28399665637 7.34678748622 P25103 P14600 594526 1211.3 Membrane receptor 49287 49287 Ki Ki Dihydrofolate reductase 6.01113819736 5.47521656542 P00374 Q920D2 594536 296.324 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 5.35476009333 5.3070182147 P00374 Q920D2 594537 324.377 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 4.73922829478 4.89117907961 P00374 Q920D2 594538 340.419 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 4.85648003624 4.9300604568 P00374 Q920D2 594539 340.419 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 5.63907409117 5.40525484315 P00374 Q920D2 594554 324.377 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Oxytocin receptor 7.73235293998 7.60205999133 P30559 P70536 332412 597.085 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Dihydrofolate reductase 4.92204365546 5.00958941668 P00374 Q920D2 594584 338.404 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 4.51079560369 4.84271881091 P00374 Q920D2 594585 338.404 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 5.09438011362 4.99646767181 P00374 Q920D2 594591 326.393 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Oxytocin receptor 8.60032972527 8.09691001301 P30559 P70536 332464 598.07 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Dihydrofolate reductase 5.70339574625 5.3767507096 P00374 Q920D2 594627 326.393 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 5.74362445874 5.47714297053 P00374 Q920D2 594628 324.377 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Oxytocin receptor 8.52047930384 9.1739251973 P30559 P70536 332627 625.138 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Oxytocin receptor 6.50751143679 6.85387196432 P30559 P70536 332645 571.048 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Oxytocin receptor 8.40623963958 8.33724216832 P30559 P70536 332655 570.06 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Oxytocin receptor 7.95346434681 7.82390874094 P30559 P70536 332911 556.033 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Cannabinoid CB2 receptor 8.18045606446 7.95860731484 P34972 Q9QZN9 595137 462.407 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 8.01322826573 7.67778070527 P34972 Q9QZN9 595145 382.517 Membrane receptor 49415 49415 Ki IC50 Oxytocin receptor 7.6883753548 7.60205999133 P30559 P70536 333024 494.563 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Oxytocin receptor 8.33889035263 7.92081875395 P30559 P70536 333032 587.044 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Oxytocin receptor 8.1259059865 7.48148606012 P30559 P70536 333065 542.991 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Serotonin 1a (5-HT1a) receptor 7.03590452598 7.63827216398 P08908 P19327 333436 460.594 Membrane receptor 30374,30374 30374 Ki,IC50 Ki Serotonin 1a (5-HT1a) receptor 7.41410752972 7.7878123956 P08908 P19327 333574 460.594 Membrane receptor 30374,30374 30374 Ki,IC50 Ki Serotonin 2a (5-HT2a) receptor 7.06048074738 9.0 P28223 P14842 596207 329.824 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 5.88239730831 7.38721614328 P28223 P14842 596218 329.824 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 5.84527179256 7.79588001734 P28223 P14842 596219 359.413 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 6.23807216158 8.69897000434 P28223 P14842 596228 343.85 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 5.65718268536 7.67778070527 P28223 P14842 596232 217.31 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 7.15490195999 9.15490195999 P28223 P14842 596241 343.85 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 6.62708799703 8.42021640338 P28223 P14842 596242 329.824 Membrane receptor 49402 49402 IC50 Ki Serotonin 2a (5-HT2a) receptor 6.76895080943 8.35654732351 P28223 P14842 596247 355.449 Membrane receptor 49402,49402 49402 IC50,IC50 Ki Adenosine A1 receptor 5.92628164965 6.58670023592 P30542 P25099 72303 217.27 Membrane receptor 16931 16931,11175,16931 Ki Ki,Ki,Ki Vanilloid receptor 4.85387196432 7.76955107862 Q8NER1 O35433 492724 479.396 Ion channel 44549,44549,44549 44549 IC50,IC50,IC50 IC50 Prostanoid EP4 receptor 8.60205999133 9.15490195999 P35408 P43114 597224 473.507 Membrane receptor 49707,49707,49707,49707,49707 49707 Ki,IC50,Ki,IC50,IC50 Ki Prostanoid EP2 receptor 5.22914798836 5.14266750357 P43116 Q62928 597224 473.507 Membrane receptor 49707 49707 Ki Ki Adenosine A3 receptor 9.42021640338 9.08618614762 P33765 P28647 335105 560.796 Membrane receptor 30572,36081,38563,45270,47561,49365,49365,52928 45270 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki Mu opioid receptor 8.85387196432 8.85387196432 P35372 P33535 335107 908.998 Membrane receptor 30482 30482,35835,38754,45287,47632,49287,52184 IC50 IC50,Ki,Ki,Ki,Ki,Ki,Ki Mu opioid receptor 9.22184874962 9.69897000434 P35372 P33535 335209 971.112 Membrane receptor 30482 30482 IC50 IC50 Adenosine A1 receptor 7.26520017041 7.59516628338 P30542 P25099 597422 374.412 Membrane receptor 49741 49741,49741,49741 Ki Ki,IC50,IC50 Adenosine A2a receptor 6.45842075605 6.17914201056 P29274 P30543 597422 374.412 Membrane receptor 49741 49741 Ki Ki Mu opioid receptor 6.88605664769 6.92081875395 P35372 P33535 335287 971.112 Membrane receptor 30482 30482 IC50 IC50 Cannabinoid CB1 receptor 7.63397650496 6.16941133131 P21554 P20272 335312 312.489 Membrane receptor 46742,45100 53907 Ki,Ki Ki Vanilloid receptor 7.98940535047 6.55752023094 Q8NER1 O35433 632467 432.482 Ion channel 51336,51336 51336 IC50,IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 6.98168555232 7.40893539297 P28845 P16232 369067 460.396 Enzyme 34972,34972 34972 Ki,IC50 Ki Adenosine A1 receptor 9.0 8.60032627852 P30542 P25099 597839 308.378 Membrane receptor 49741 49741 Ki Ki Adenosine A2a receptor 6.40011692793 6.30016227413 P29274 P30543 597839 308.378 Membrane receptor 49741 49741 Ki Ki Serotonin 2a (5-HT2a) receptor 7.61383914664 8.71896663275 P28223 P14842 335712 205.256 Membrane receptor 30538,39082 30538 Ki,Ki IC50 Serotonin 2a (5-HT2a) receptor 8.7447274949 9.13076828027 P28223 P14842 335713 205.256 Membrane receptor 30538 30538 Ki IC50 Serotonin 2a (5-HT2a) receptor 8.23657200644 9.13667713988 P28223 P14842 335714 209.22 Membrane receptor 30538 30538 Ki IC50 Serotonin 2a (5-HT2a) receptor 7.69897000434 9.11350927483 P28223 P14842 335729 177.203 Membrane receptor 30538 30538 Ki IC50 Serotonin 2a (5-HT2a) receptor 7.92081875395 9.23657200644 P28223 P14842 335730 191.23 Membrane receptor 30538 30538 Ki IC50 Endothelin receptor ET-A 10.8239087409 9.48148606012 P25101 P26684 187027 614.511 Membrane receptor 16144 16144 Ki IC50 Serotonin 2a (5-HT2a) receptor 7.92081875395 9.26760624018 P28223 P14842 335908 225.675 Membrane receptor 30538 30538 Ki IC50 Serotonin 2a (5-HT2a) receptor 7.67778070527 8.77469071827 P28223 P14842 335909 317.126 Membrane receptor 30538 30538 Ki IC50 Serotonin 2c (5-HT2c) receptor 8.61828600322 7.21467016499 P28335 P08909 599085 231.294 Membrane receptor 49854,49854 49854 Ki,IC50 IC50 Cannabinoid CB1 receptor 6.04335142079 5.7584535194 P21554 P20272 336949 476.15 Membrane receptor 30590 30590 Ki Ki Cannabinoid CB1 receptor 5.72653572738 5.58203035779 P21554 P20272 337066 431.699 Membrane receptor 30590 30590 Ki Ki Metabotropic glutamate receptor 5 8.99869906698 9.14874165128 P41594 P31424 337091 226.297 Membrane receptor 30615 30615 Ki Ki Cannabinoid CB1 receptor 6.45222529461 6.60730304674 P21554 P20272 337176 397.254 Membrane receptor 30590 30590 Ki Ki Metabotropic glutamate receptor 5 9.43179827593 9.60205999133 P41594 P31424 337510 224.281 Membrane receptor 30615 30615 Ki Ki Cannabinoid CB1 receptor 7.54975089168 8.85387196432 P21554 P20272 599995 675.201 Membrane receptor 49921 49921 IC50 IC50 Cannabinoid CB1 receptor 8.60032627852 8.95860731484 P21554 P20272 600148 640.756 Membrane receptor 49921 49921 IC50 IC50 Adenosine A1 receptor 9.09691001301 8.84466396253 P30542 P25099 75895 344.408 Membrane receptor 13965,13965,13965 13965,13965,13965 Ki,Ki,Ki Ki,Ki,Ki Adenosine A3 receptor 7.5376020021 6.54363396687 P33765 P28647 338715 558.757 Membrane receptor 30715,36081,38563,44562 30715 Ki,Ki,Ki,Ki Ki Adenosine A3 receptor 7.80966830183 6.4934949676 P33765 P28647 338778 574.823 Membrane receptor 30715,36081,38563,45270 30715,38563,45270 Ki,Ki,Ki,Ki Ki,Ki,Ki Dihydrofolate reductase 5.39794000867 4.68824613894 P00374 Q920D2 600929 445.449 Enzyme 49957 49957 IC50 IC50 Histamine H3 receptor 7.52287874528 6.6038006529 Q9Y5N1 Q9QYN8 339073 408.172 Membrane receptor 30729 30729 Ki Ki Histamine H3 receptor 7.44369749923 6.49620931694 Q9Y5N1 Q9QYN8 339074 394.145 Membrane receptor 30729 30729 Ki Ki Histamine H3 receptor 7.7447274949 6.59345981957 Q9Y5N1 Q9QYN8 339075 236.353 Membrane receptor 30729 30729 Ki Ki Histamine H3 receptor 8.52287874528 7.34678748622 Q9Y5N1 Q9QYN8 339086 276.417 Membrane receptor 30729 30729 Ki Ki Delta opioid receptor 8.31695296176 6.70333480974 P41143 P33533 77021 345.519 Membrane receptor 36965,36965,37230 14428 Ki,Ki,Ki Ki Histamine H3 receptor 8.22184874962 7.05060999336 Q9Y5N1 Q9QYN8 339236 250.38 Membrane receptor 30729 30729 Ki Ki Histamine H3 receptor 7.39794000867 6.46218090493 Q9Y5N1 Q9QYN8 339244 236.353 Membrane receptor 30729 30729 Ki Ki Histamine H3 receptor 7.85387196432 7.30102999566 Q9Y5N1 Q9QYN8 339472 276.417 Membrane receptor 30729 30729 Ki Ki Histamine H3 receptor 9.30102999566 8.30102999566 Q9Y5N1 Q9QYN8 339481 290.444 Membrane receptor 30729 30729 Ki Ki Adenosine A1 receptor 5.73992861201 6.52870828894 P30542 P25099 500131 512.557 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 7.03621217265 7.39577394692 P29274 P30543 500131 512.557 Membrane receptor 46829 46829 Ki Ki Cathepsin K 9.0268721464 6.88605664769 P43235 O35186 339579 404.503 Enzyme 30702 30702 IC50 IC50 Adenosine A1 receptor 9.30980391997 7.76447155309 P30542 P25099 77702 375.464 Membrane receptor 49741 16115,1775,3214,49741 Ki IC50,IC50,IC50,IC50 Adenosine A2a receptor 5.4164891021 4.95276443568 P29274 P30543 77702 375.464 Membrane receptor 16115,16115 3214,49741 IC50,Ki IC50,IC50 Urotensin II receptor 6.75292270299 7.16115090926 Q9UKP6 P49684 580961 688.856 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Urotensin II receptor 6.55237162343 6.85387196432 Q9UKP6 P49684 580997 624.751 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Bradykinin B1 receptor 9.22914798836 9.03621217265 P46663 P97583 78762 601.741 Membrane receptor 44560 44560 Ki Ki Monoamine oxidase B 4.77211329539 5.46852108296 P27338 P19643 603564 237.318 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 4.22184874962 4.91009488856 P21397 P21396 603564 237.318 Enzyme 49639 49639 Ki Ki Monoamine oxidase B 6.33724216832 6.79588001734 P27338 P19643 603654 265.371 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 5.0 4.29328221766 P21397 P21396 603654 265.371 Enzyme 49639 49639 Ki Ki Monoamine oxidase B 7.31875876262 7.13076828027 P27338 P19643 603655 299.387 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 4.79048498546 5.19449914184 P21397 P21396 603657 209.308 Enzyme 49639 49639 Ki Ki Monoamine oxidase B 6.88605664769 6.00877392431 P27338 P19643 603659 237.361 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 5.17914201056 5.43297363384 P21397 P21396 603659 237.361 Enzyme 49639 49639 Ki Ki Monoamine oxidase B 7.16749108729 6.56863623584 P27338 P19643 603660 251.388 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 5.60205999133 4.85078088734 P21397 P21396 603660 251.388 Enzyme 49639 49639 Ki Ki Monoamine oxidase B 7.42021640338 6.88605664769 P27338 P19643 603661 285.404 Enzyme 49639 49639 Ki Ki Acetylcholinesterase 7.36700181475 7.42693598216 P22303 P37136 79557 None Enzyme 37075,43854,48391,50471 37075,48391 IC50,IC50,IC50,IC50 IC50,IC50 Adenosine A3 receptor 6.5376020021 7.0 P33765 P28647 605198 267.241 Membrane receptor 51669 15464 IC50 Ki Adenosine A1 receptor 6.50863830617 7.89279003035 P30542 P25099 605198 267.241 Membrane receptor 51669 127 IC50 Ki Adenosine A2a receptor 6.15490195999 7.52287874528 P29274 P30543 605198 267.241 Membrane receptor 51669 15464 IC50 Ki Dopamine D1 receptor 8.72124639905 10.096910013 P21728 P18901 100867 290.402 Membrane receptor 30791,31902,31902,37386 15453 Ki,Ki,Ki,Ki Ki Dopamine D2 receptor 7.35163998902 8.22184874962 P14416 P61169 100867 290.402 Membrane receptor 30791,31902,31902,37386 15453 Ki,Ki,Ki,Ki Ki Cholecystokinin A receptor 6.70553377384 6.70553377384 P32238 P30551 343119 427.452 Membrane receptor 30939 46412,48402 IC50 IC50,IC50 Cholecystokinin A receptor 5.55284196866 5.48945498979 P32238 P30551 343120 351.356 Membrane receptor 30939 46412 IC50 IC50 Cholecystokinin A receptor 5.39794000867 5.39685562738 P32238 P30551 343173 414.453 Membrane receptor 30939 48402 IC50 IC50 Dopamine D2 receptor 6.69464863055 6.46852108296 P14416 P61169 81407 247.376 Membrane receptor 38128,49130 12058 Ki,Ki Ki Fructose-1,6-bisphosphatase 5.7328282716 4.69897000434 P09467 P19112 581642 385.31 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.0 5.69897000434 P09467 P19112 581672 387.369 Enzyme 49142 49142 IC50 IC50 Fructose-1,6-bisphosphatase 6.07058107429 5.60205999133 P09467 P19112 581673 367.312 Enzyme 49142 49142 IC50 IC50 Adenosine A1 receptor 6.37778597703 8.28755918168 P30542 P25099 82353 470.588 Membrane receptor 16931 16931,16931 Ki Ki,Ki Cathepsin S 6.74957999769 5.61243222058 P25774 Q02765 344540 481.531 Enzyme 30943,30943,37689 37689 IC50,IC50,IC50 IC50 Cathepsin L 6.57839607313 7.04575749056 P07711 P07154 344540 481.531 Enzyme 37689 37689 IC50 IC50 Cathepsin B 5.29943873971 6.03385826726 P07858 P00787 344540 481.531 Enzyme 30943,37689 37689 IC50,IC50 IC50 Fructose-1,6-bisphosphatase 7.0 5.69897000434 P09467 P19112 581716 387.73 Enzyme 49142 49142 IC50 IC50 Adenosine A1 receptor 6.20065945055 8.24919653879 P30542 P25099 82433 486.587 Membrane receptor 16931 16931,16931 Ki Ki,Ki Fructose-1,6-bisphosphatase 6.39794000867 5.69897000434 P09467 P19112 581772 414.191 Enzyme 49142 49142 IC50 IC50 Anandamide amidohydrolase 6.59006687667 6.7878123956 O00519 P97612 450703 399.897 Enzyme 45114 45114 IC50 IC50 Fructose-1,6-bisphosphatase 7.22184874962 6.45593195565 P09467 P19112 581783 393.349 Enzyme 49142 49142 IC50 IC50 Branched-chain-amino-acid transferase 6.09691001301 6.11092437481 P54687 P54690 345575 417.79 Enzyme 31047 31047,31047 IC50 IC50,IC50 Adenosine A1 receptor 4.0 5.99139982824 P30542 P25099 607751 384.389 Membrane receptor 3027 3027 IC50 Ki Dihydrofolate reductase 7.99139982824 7.55284196866 P00374 Q920D2 232379 359.81 Enzyme 53022 12673 Ki IC50 Serotonin 1a (5-HT1a) receptor 8.30102999566 8.31247103879 P08908 P19327 84146 371.475 Membrane receptor 30228 11049 IC50 IC50 Dopamine D2 receptor 7.35654732351 7.42021640338 P14416 P61169 84146 371.475 Membrane receptor 30228 11049 IC50 IC50 Anandamide amidohydrolase 6.59687947882 6.72584215074 O00519 P97612 450991 392.438 Enzyme 45114 45114 IC50 IC50 Adenosine A1 receptor 4.97109090278 4.95860731484 P30542 P25099 84584 299.311 Membrane receptor 16975,45208,49281,50809 45180 IC50,IC50,IC50,IC50 Ki HMG-CoA reductase 7.63827216398 7.39794000867 P04035 P51639 84814 390.513 Enzyme 20770 47915 IC50 IC50 Anandamide amidohydrolase 5.93292914395 6.90308998699 O00519 P97612 451060 355.417 Enzyme 45114 45114 IC50 IC50 Norepinephrine transporter 7.54468779756 7.42829116819 P23975 Q9WTR4 609219 293.789 Transporter 35284,35284 12788 IC50,Ki IC50 Dopamine transporter 8.95860731484 8.87333099734 Q01959 P23977 609219 293.789 Transporter 35284 11608,12788,12997,12997 IC50 IC50,IC50,Ki,Ki Serotonin transporter 7.87478999885 7.35163998902 P31645 P31652 609219 293.789 Transporter 35284,35284 12788 IC50,Ki IC50 Anandamide amidohydrolase 6.49485002168 7.38721614328 O00519 P97612 451133 357.394 Enzyme 45114 45114 IC50 IC50 Histamine H3 receptor 7.30980391997 7.03621217265 Q9Y5N1 Q9QYN8 494859 334.453 Membrane receptor 45718 45718 Ki Ki Serotonin 1a (5-HT1a) receptor 8.2924298239 7.76955107862 P08908 P19327 347877 450.638 Membrane receptor 31185 31185 Ki Ki Histamine H3 receptor 9.65757731918 9.30980391997 Q9Y5N1 Q9QYN8 451251 455.719 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 8.79048498546 8.17005330406 Q9Y5N1 Q9QYN8 451262 497.756 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 9.55284196866 9.14266750357 Q9Y5N1 Q9QYN8 713478 353.501 Membrane receptor 53911 53911 Ki Ki Adenosine A2a receptor 7.79588001734 7.22914798836 P29274 P30543 709953 434.491 Membrane receptor 53459 53459 Ki Ki Urotensin II receptor 6.46852108296 7.79588001734 Q9UKP6 P49684 582507 598.777 Membrane receptor 48952 48952 IC50 IC50 Urotensin II receptor 7.15937938131 8.22184874962 Q9UKP6 P49684 582512 637.768 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Gonadotropin-releasing hormone receptor 9.39794000867 9.39794000867 P30968 P30969 349376 565.661 Membrane receptor 31239 31239 Ki Ki Urotensin II receptor 6.75431915308 9.0 Q9UKP6 P49684 582544 565.106 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Cannabinoid CB2 receptor 7.0 6.69897000434 P34972 Q9QZN9 582548 316.398 Membrane receptor 48957 48957 Ki IC50 Histamine H3 receptor 7.30980391997 7.69897000434 Q9Y5N1 Q9QYN8 611818 225.287 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.92081875395 7.72124639905 Q9Y5N1 Q9QYN8 611819 225.287 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.50863830617 7.63827216398 Q9Y5N1 Q9QYN8 611820 225.287 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.67778070527 7.60205999133 Q9Y5N1 Q9QYN8 611821 239.314 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.82390874094 7.92081875395 Q9Y5N1 Q9QYN8 611822 239.314 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 8.32790214206 7.7447274949 Q9Y5N1 Q9QYN8 611823 239.314 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.72124639905 7.72124639905 Q9Y5N1 Q9QYN8 611888 253.341 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.28399665637 7.7447274949 Q9Y5N1 Q9QYN8 611894 267.367 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.38721614328 7.63827216398 Q9Y5N1 Q9QYN8 611976 267.367 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.13076828027 7.7447274949 Q9Y5N1 Q9QYN8 611977 267.367 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.12493873661 7.65757731918 Q9Y5N1 Q9QYN8 611978 281.394 Membrane receptor 50228 50228 Ki Ki Histamine H3 receptor 7.04095860768 7.7447274949 Q9Y5N1 Q9QYN8 611980 281.394 Membrane receptor 50228 50228 Ki Ki Anandamide amidohydrolase 6.62090753092 7.11350927483 O00519 P97612 612112 300.309 Enzyme 50231,50231 50231 IC50,IC50 IC50 Acetyl-CoA carboxylase 1 6.38721614328 7.26768072045 Q13085 P11497 350255 485.617 Enzyme 31354,34929,50235 31354,45547,50235,50688 IC50,IC50,IC50 IC50,IC50,IC50,IC50 Histamine H3 receptor 9.46852108296 9.19382002602 Q9Y5N1 Q9QYN8 350309 302.454 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.45593195565 9.33724216832 Q9Y5N1 Q9QYN8 350310 370.571 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 7.91721462968 7.41907502432 Q9Y5N1 Q9QYN8 350388 366.518 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.76955107862 9.05060999336 Q9Y5N1 Q9QYN8 350420 316.481 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 8.30980391997 7.40230481407 Q9Y5N1 Q9QYN8 350450 359.506 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 7.62342304294 7.12784372725 Q9Y5N1 Q9QYN8 350451 352.492 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 7.71219827007 7.43533393575 Q9Y5N1 Q9QYN8 350506 316.438 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.46852108296 9.25181197299 Q9Y5N1 Q9QYN8 350596 316.481 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.69897000434 9.09691001301 Q9Y5N1 Q9QYN8 350597 378.55 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.69897000434 8.8894102897 Q9Y5N1 Q9QYN8 350628 330.507 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 7.76700388961 7.48811663902 Q9Y5N1 Q9QYN8 350629 373.532 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 8.5376020021 7.15428198203 Q9Y5N1 Q9QYN8 350663 366.518 Membrane receptor 31381 31381 Ki Ki Histamine H3 receptor 9.58502665203 8.95860731484 Q9Y5N1 Q9QYN8 350665 316.481 Membrane receptor 31381 31381 Ki Ki Serotonin 1a (5-HT1a) receptor 7.20065945055 7.20065945055 P08908 P19327 350741 508.652 Membrane receptor 31374 46353 Ki Ki Serotonin 1a (5-HT1a) receptor 7.16115090926 7.16115090926 P08908 P19327 350742 402.487 Membrane receptor 31374 46353 Ki Ki Serotonin 1a (5-HT1a) receptor 7.39794000867 7.63827216398 P08908 P19327 350773 456.578 Membrane receptor 31374 36406 Ki Ki Serotonin 1a (5-HT1a) receptor 7.39794000867 7.39794000867 P08908 P19327 350921 482.615 Membrane receptor 31374 46353 Ki Ki Serotonin 1a (5-HT1a) receptor 6.31875876262 6.31875876262 P08908 P19327 350922 388.461 Membrane receptor 31374 46353 Ki Ki Dopamine D2 receptor 7.67778070527 8.50863830617 P14416 P61169 88815 211.327 Membrane receptor 21630,21630,21630,21630,30162,30162,30162,30162,38679 45224 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50 Ki Dopamine D3 receptor 8.82390874094 9.10790539731 P35462 P19020 88815 211.327 Membrane receptor 21630,21630,21630,30162,30162,30162 45224 Ki,Ki,IC50,Ki,Ki,IC50 Ki Serotonin 1a (5-HT1a) receptor 7.56863623584 7.72124639905 P08908 P19327 351005 470.647 Membrane receptor 31374 46353 Ki Ki Aldose reductase 6.29043534613 7.41022410442 P15121 P07943 88882 319.399 Enzyme 51711,53097 14299,41469 IC50,IC50 IC50,IC50 Aldehyde reductase 5.58502665203 5.82390874094 P14550 P51635 88882 319.399 Enzyme 51711 14299 IC50 IC50 Serotonin 1a (5-HT1a) receptor 8.39794000867 8.52287874528 P08908 P19327 351080 522.722 Membrane receptor 31374 46353 Ki Ki Gonadotropin-releasing hormone receptor 8.0 8.15490195999 P30968 P30969 351140 1125.24 Membrane receptor 31350 31350 IC50 IC50 Gonadotropin-releasing hormone receptor 10.0 6.69897000434 P30968 P30969 351157 628.731 Membrane receptor 31350 31350 IC50 IC50 Serotonin 1a (5-HT1a) receptor 7.82390874094 8.39794000867 P08908 P19327 351161 522.679 Membrane receptor 31374 36406,46353 Ki Ki,Ki Gonadotropin-releasing hormone receptor 10.0 6.82390874094 P30968 P30969 351207 657.769 Membrane receptor 31350 31350 IC50 IC50 Ghrelin receptor 8.04095860768 8.69897000434 Q92847 O08725 613362 441.497 Membrane receptor 50448 50448 IC50 IC50 Mu opioid receptor 9.33724216832 9.33724216832 P35372 P33535 351610 514.615 Membrane receptor 31329 46616 Ki Ki Delta opioid receptor 7.95860731484 7.95860731484 P41143 P33533 351610 514.615 Membrane receptor 31329 46616 Ki Ki Mu opioid receptor 9.04 7.99139982824 P35372 P33535 613764 760.92 Membrane receptor 50453 50453 IC50 Ki Mu opioid receptor 8.54 7.79317412397 P35372 P33535 613765 875.023 Membrane receptor 50453 50453 IC50 Ki Mu opioid receptor 8.31 8.82390874094 P35372 P33535 613769 815.011 Membrane receptor 50453 50453 IC50 Ki Mu opioid receptor 7.48 8.10902040301 P35372 P33535 613770 1197.47 Membrane receptor 50453 50453 IC50 Ki Mu opioid receptor 6.95 8.09366495819 P35372 P33535 613771 1368.62 Membrane receptor 50453 50453 IC50 Ki G protein-coupled receptor 44 9.8210325765 8.12493873661 Q9Y5Y4 Q6XKD3 613847 434.41 Membrane receptor 50457,50457 50457 IC50,IC50 IC50 Nitric-oxide synthase, brain 4.72124639905 6.6259059865 P29475 P29476 613900 408.46 Enzyme 50330 50330,50330 IC50 IC50,Ki Serotonin 2a (5-HT2a) receptor 9.18045606446 9.05551732785 P28223 P14842 89669 260.128 Membrane receptor 31732 31732 Ki Ki Cannabinoid CB1 receptor 8.2924298239 8.65757731918 P21554 P20272 89797 372.541 Membrane receptor 52442 53169 Ki Ki Oxytocin receptor 7.56863623584 7.11918640772 P30559 P70536 352319 994.189 Membrane receptor 30371,30371,38537 30371 Ki,IC50,Ki Ki Alpha-1d adrenergic receptor 7.67778070527 6.73048705578 P25100 P23944 146114 401.503 Membrane receptor 13032 13032 Ki Ki Adenosine A1 receptor 5.68465952337 6.58502665203 P30542 P25099 352423 508.593 Membrane receptor 31364,46829,46829,51928 31364,46829,46829 Ki,Ki,Ki,Ki Ki,Ki,Ki Adenosine A2a receptor 6.31515463836 7.02826040911 P29274 P30543 352423 508.593 Membrane receptor 31364,46829,46829,51928 31364,46829,46829 Ki,Ki,Ki,Ki Ki,Ki,Ki Adenosine A1 receptor 6.7328282716 7.92081875395 P30542 P25099 352455 439.488 Membrane receptor 31364 31364 Ki Ki Adenosine A2a receptor 7.48678239993 6.94692155652 P29274 P30543 352455 439.488 Membrane receptor 31364 31364 Ki Ki Adenosine A1 receptor 7.26121944152 8.33724216832 P30542 P25099 352681 439.488 Membrane receptor 31364,51928 31364 Ki,Ki Ki Adenosine A2a receptor 6.79048498546 7.57348873864 P29274 P30543 352681 439.488 Membrane receptor 31364,51928 31364 Ki,Ki Ki Adenosine A1 receptor 6.73754891027 8.0 P30542 P25099 352715 453.514 Membrane receptor 31364 31364 Ki Ki Adenosine A2a receptor 6.1140736602 6.52724355068 P29274 P30543 352715 453.514 Membrane receptor 31364 31364 Ki Ki Mu opioid receptor 9.79588001734 9.79588001734 P35372 P33535 495699 514.615 Membrane receptor 31329 44204,46616 Ki Ki,Ki Delta opioid receptor 10.5086383062 10.5086383062 P41143 P33533 495699 514.615 Membrane receptor 31329 44204,46616 Ki Ki,Ki Neuronal acetylcholine receptor protein alpha-7 subunit 8.15490195999 8.05063740921 P36544 Q05941 352807 271.314 Ion channel 39478 31361,39478 Ki Ki,Ki Histamine H3 receptor 6.95860731484 6.59006687667 Q9Y5N1 Q9QYN8 452026 384.598 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 7.91009488856 7.42021640338 Q9Y5N1 Q9QYN8 452100 446.667 Membrane receptor 44314 44314 Ki Ki Serotonin transporter 6.66354026615 7.91364016933 P31645 P31652 353308 441.513 Transporter 31450 31450 IC50 Ki Serotonin transporter 7.36957212497 8.46852108296 P31645 P31652 353469 413.46 Transporter 31450 31450 IC50 Ki Serotonin transporter 7.42829116819 8.44369749923 P31645 P31652 353470 413.46 Transporter 31450 31450 IC50 Ki Serotonin transporter 6.89279003035 8.14874165128 P31645 P31652 353497 427.487 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.74232142513 8.09691001301 P31645 P31652 353498 427.487 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 7.22257317761 8.32790214206 P31645 P31652 353529 427.487 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 7.27164621798 8.45593195565 P31645 P31652 353530 439.498 Transporter 31450 31450 IC50 Ki Histamine H3 receptor 8.48017200622 7.95078197733 Q9Y5N1 Q9QYN8 452156 466.722 Membrane receptor 44314 44314 Ki Ki Serotonin transporter 7.22402566887 8.40893539297 P31645 P31652 353649 439.498 Transporter 31450 31450 IC50 Ki Serotonin transporter 7.44009337496 8.3767507096 P31645 P31652 353671 439.498 Transporter 31450 31450 IC50 Ki Serotonin transporter 7.82390874094 8.16749108729 P31645 P31652 353716 368.444 Transporter 31450 31450 IC50 Ki Serotonin transporter 7.72815839346 8.82390874094 P31645 P31652 353717 439.498 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 7.75945075172 8.2757241304 P31645 P31652 353718 439.498 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 7.3705904009 8.36653154442 P31645 P31652 353765 408.508 Transporter 31450 31450 IC50 Ki Serotonin transporter 6.39794000867 7.88605664769 P31645 P31652 353766 408.508 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.13548891894 7.38510790108 P31645 P31652 353788 408.508 Transporter 31450,44692 31450,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.70553377384 7.69036983257 P31645 P31652 353789 385.407 Transporter 31450 31450 IC50 Ki Acetylcholinesterase 6.89859664944 7.0280287236 P22303 P37136 353879 399.52 Enzyme 31481 31481 IC50 IC50 Acetylcholinesterase 7.67778070527 7.72699872794 P22303 P37136 353882 385.493 Enzyme 31481 31481 IC50 IC50 Acetylcholinesterase 7.13312218566 7.42596873227 P22303 P37136 353895 479.563 Enzyme 31481 31481 IC50 IC50 Acetylcholinesterase 7.55078002745 7.42596873227 P22303 P37136 353902 None Enzyme 31481,51782 31481 IC50,IC50 IC50 Vanilloid receptor 7.5484550065 6.55913653231 Q8NER1 O35433 91783 305.412 Ion channel 36194,47070,49452,53995 17091,45405,45405,53995 IC50,IC50,IC50,Ki Ki,IC50,Ki,IC50 Glutamate receptor ionotropic, AMPA 2 5.64975198167 5.11918640772 P42262 P19491 92458 389.878 Ion channel 50876 45271 IC50 IC50 Androgen Receptor 8.76955107862 6.56863623584 P10275 P15207 364997 311.292 Transcription Factor 34764 34764 Ki IC50 Nitric-oxide synthase, brain 7.0 7.0 P29475 P29476 93362 122.168 Enzyme 46991 46991 IC50 IC50 Dopamine D2 receptor 6.93930215965 8.25963731051 P14416 P61169 146638 268.353 Membrane receptor 2789,49693,49693 2789 Ki,Ki,Ki Ki Dopamine D2 receptor 7.32790214206 7.57186520597 P14416 P61169 146648 370.286 Membrane receptor 2789 2789 Ki Ki Dopamine D2 receptor 7.05898575629 8.3767507096 P14416 P61169 146683 308.378 Membrane receptor 2789 2789 Ki Ki Histamine H3 receptor 5.63264407897 7.04000516167 Q9Y5N1 Q9QYN8 94225 123.156 Membrane receptor 16985 16985 IC50 Ki Histamine H3 receptor 8.0 8.88272870434 Q9Y5N1 Q9QYN8 94285 151.209 Membrane receptor 16985 16985 IC50 Ki Histamine H3 receptor 5.85078088734 8.32057210339 Q9Y5N1 Q9QYN8 94453 151.209 Membrane receptor 16985 16985 IC50 Ki Fatty acid synthase 6.68402965454 7.13667713988 P49327 P12785 356737 316.696 Enzyme 31790 31790 IC50 IC50 Histamine H3 receptor 9.14794000867 7.89431811792 Q9Y5N1 Q9QYN8 627435 403.49 Membrane receptor 51148,51148 51148,51148 Ki,IC50 IC50,Ki Fatty acid synthase 5.85294232897 6.25963731051 P49327 P12785 356993 282.251 Enzyme 31790 31790 IC50 IC50 Alpha-1d adrenergic receptor 10.3979400087 10.5228787453 P25100 P23944 190581 395.452 Membrane receptor 13032 13032 Ki Ki Oxytocin receptor 6.76955107862 6.63827216398 P30559 P70536 96086 435.515 Membrane receptor 52842 52842 Ki Ki Vasopressin V1a receptor 4.28399665637 7.49485002168 P37288 P30560 96086 435.515 Membrane receptor 52842 52842 Ki Ki Serotonin 2a (5-HT2a) receptor 9.45593195565 9.58502665203 P28223 P14842 358567 272.138 Membrane receptor 31732 31732 Ki Ki Serotonin 2a (5-HT2a) receptor 7.82390874094 7.3767507096 P28223 P14842 358569 272.138 Membrane receptor 31732 31732 Ki Ki Serotonin 2a (5-HT2a) receptor 7.2757241304 7.32790214206 P28223 P14842 358640 286.165 Membrane receptor 31732 31732 Ki Ki Serotonin 2a (5-HT2a) receptor 6.76955107862 7.13076828027 P28223 P14842 358641 312.202 Membrane receptor 31732 31732 Ki Ki Gonadotropin-releasing hormone receptor 7.23657200644 6.5376020021 P30968 P30969 621029 457.614 Membrane receptor 50731 50731 IC50 IC50 Gonadotropin-releasing hormone receptor 7.61531133696 6.73400522429 P30968 P30969 621031 456.626 Membrane receptor 50731,50731 50731,50731 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.78057067029 7.14878473178 P30968 P30969 621101 456.626 Membrane receptor 50731,50731 50731,50731 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 8.03275077438 6.18941185911 P30968 P30969 621175 458.555 Membrane receptor 50731,50731 50731,50731 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 8.46965107982 7.41457589818 P30968 P30969 621176 486.609 Membrane receptor 50731,50731 50731,50731 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.38274135824 6.68075537152 P30968 P30969 621177 476.615 Membrane receptor 50731,50731 50731,50731 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.18682981631 6.28001803204 P30968 P30969 621178 476.615 Membrane receptor 50731,50731 50731,50731 IC50,IC50 IC50,IC50 Melanocortin receptor 3 6.25265143844 6.00130484169 P41968 P32244 621194 600.182 Membrane receptor 50673,50673 50673 IC50,IC50 IC50 Melanocortin receptor 4 8.09793028383 8.69897000434 P32245 P70596 621194 600.182 Membrane receptor 50673,50673 50673 IC50,IC50 IC50 Vasopressin V2 receptor 8.61092437481 8.63827216398 P30518 Q00788 73070 473.926 Membrane receptor 4138,5160,5160,14475,30136,37042,37905,37905 3173,4138,14475 IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50 Vasopressin V1a receptor 6.82390874094 6.46852108296 P37288 P30560 73070 473.926 Membrane receptor 4138,5160,6363,14475,30136,37042,37905 3173,4138,14475 IC50,IC50,Ki,IC50,IC50,IC50,IC50 IC50,IC50,IC50 Sodium/hydrogen exchanger 1 5.92081875395 7.18708664336 P19634 P26431 97246 283.347 Transporter 21666,36727 36446,48215 IC50,IC50 IC50,IC50 Dopamine transporter 6.49079747767 6.70996538864 Q01959 P23977 359546 359.203 Transporter 36559 31656 Ki Ki Serotonin transporter 6.54211810327 6.77728352885 P31645 P31652 359546 359.203 Transporter 36559 31656 Ki Ki Metabotropic glutamate receptor 1 8.0 8.5 Q13255 P23385 359820 343.447 Membrane receptor 35368 31805,44256 IC50 IC50,IC50 Adenosine A2a receptor 9.39794000867 8.0268721464 P29274 P30543 424882 460.528 Membrane receptor 38360 38360 Ki Ki Vanilloid receptor 8.65757731918 8.49148333035 Q8NER1 O35433 622613 435.325 Ion channel 50778,52179 50778,52179 IC50,IC50 IC50,IC50 Dipeptidyl peptidase IV 9.0 9.0 P27487 P14740 360699 395.455 Enzyme 31905 31905 Ki Ki Dopamine transporter 8.76955107862 9.3767507096 Q01959 P23977 360905 338.24 Transporter 35284 31814 IC50 Ki Serotonin transporter 8.49621145085 8.38721614328 P31645 P31652 360905 338.24 Transporter 35284,35284 31814 IC50,Ki Ki Muscarinic acetylcholine receptor M2 6.31875876262 6.31875876262 P08172 P10980 98821 169.221 Membrane receptor 14434 14434 Ki Ki Muscarinic acetylcholine receptor M4 5.10237290871 5.10237290871 P08173 P08485 98821 169.221 Membrane receptor 14434 14434 Ki Ki Vasopressin V2 receptor 6.65937938131 6.82390874094 P30518 Q00788 453410 462.584 Membrane receptor 44817,44817 44817 IC50,Ki IC50 Muscarinic acetylcholine receptor M1 8.33724216832 8.25181197299 P11229 P08482 99028 169.221 Membrane receptor 15502 14434,14434 Ki Ki,Ki Muscarinic acetylcholine receptor M3 6.16749108729 6.16749108729 P20309 P08483 99028 169.221 Membrane receptor 15502 14434 Ki Ki Muscarinic acetylcholine receptor M2 8.15490195999 7.76955107862 P08172 P10980 99028 169.221 Membrane receptor 14434,14434,14434,15502,15502 14434,14434,14434 IC50,IC50,Ki,Ki,Ki IC50,IC50,Ki Muscarinic acetylcholine receptor M4 7.48148606012 7.48148606012 P08173 P08485 99028 169.221 Membrane receptor 14434,15502,15502 14434 Ki,Ki,Ki Ki Muscarinic acetylcholine receptor M1 5.63827216398 5.58502665203 P11229 P08482 99081 183.247 Membrane receptor 15502 14434,14434 Ki Ki,Ki Muscarinic acetylcholine receptor M3 4.82390874094 4.82390874094 P20309 P08483 99081 183.247 Membrane receptor 15502 14434 Ki Ki Muscarinic acetylcholine receptor M2 5.56863623584 5.56863623584 P08172 P10980 99081 183.247 Membrane receptor 14434,15502,15502 14434 Ki,Ki,Ki Ki Muscarinic acetylcholine receptor M4 5.08092190762 5.08092190762 P08173 P08485 99081 183.247 Membrane receptor 14434,15502,15502 14434 Ki,Ki,Ki Ki Anandamide amidohydrolase 7.43179827593 7.85387196432 O00519 P97612 453427 379.409 Enzyme 44028 44028,44028,44028 Ki IC50,Ki,Ki Muscarinic acetylcholine receptor M2 6.42021640338 6.42021640338 P08172 P10980 99320 160.234 Membrane receptor 14434,14434,14434 14434,14434,14434 IC50,IC50,Ki IC50,IC50,Ki Muscarinic acetylcholine receptor M4 5.79588001734 5.79588001734 P08173 P08485 99320 160.234 Membrane receptor 14434 14434 Ki Ki Adenosine A1 receptor 7.22184874962 8.0 P30542 P25099 361499 357.45 Membrane receptor 31858 31858 Ki Ki Adenosine A1 receptor 7.65757731918 8.22184874962 P30542 P25099 361643 371.477 Membrane receptor 31858 31858 Ki Ki Adenosine A2a receptor 5.35654732351 5.56863623584 P29274 P30543 361643 371.477 Membrane receptor 31858 31858 Ki Ki Gonadotropin-releasing hormone receptor 9.52287874528 9.30102999566 P30968 P30969 453493 1209.4 Membrane receptor 31350 14661,31350 IC50 IC50,IC50 Adenosine A1 receptor 7.48148606012 8.10790539731 P30542 P25099 361668 388.461 Membrane receptor 31861 31861 Ki Ki Adenosine A1 receptor 7.45593195565 8.39794000867 P30542 P25099 361728 385.503 Membrane receptor 31858 31858 Ki Ki Adenosine A2a receptor 5.79588001734 5.95860731484 P29274 P30543 361728 385.503 Membrane receptor 31858 31858 Ki Ki Adenosine A1 receptor 8.14283512013 8.94302832385 P30542 P25099 361763 416.514 Membrane receptor 31858,49741 31858,49741 Ki,Ki Ki,Ki Adenosine A2a receptor 5.19348099825 5.61261017366 P29274 P30543 361763 416.514 Membrane receptor 31858,49741 49741 Ki,Ki Ki Adenosine A1 receptor 8.13076828027 8.88605664769 P30542 P25099 361768 416.514 Membrane receptor 31861 31861 Ki Ki Adenosine A2a receptor 5.19314197048 5.61261017366 P29274 P30543 361768 416.514 Membrane receptor 31861 31861 Ki Ki Adenosine A1 receptor 8.69897000434 9.22184874962 P30542 P25099 361770 360.451 Membrane receptor 31858 31858 Ki Ki Adenosine A1 receptor 7.45593195565 8.07572071394 P30542 P25099 361777 427.54 Membrane receptor 31858 31858 Ki Ki Adenosine A1 receptor 7.5376020021 8.39794000867 P30542 P25099 361783 430.54 Membrane receptor 31861 31861 Ki Ki Adenosine A1 receptor 7.34678748622 7.97881070093 P30542 P25099 361785 441.566 Membrane receptor 31858 31858 Ki Ki Adenosine A1 receptor 7.92081875395 9.15490195999 P30542 P25099 361791 344.408 Membrane receptor 31861 31861 Ki Ki Adenosine A2a receptor 5.77989191196 5.90308998699 P29274 P30543 361791 344.408 Membrane receptor 31861 31861 Ki Ki Histamine H3 receptor 9.08092190762 8.58502665203 Q9Y5N1 Q9QYN8 631809 361.437 Membrane receptor 51341 51341 Ki Ki Metabotropic glutamate receptor 5 8.30102999566 7.83117055449 P41594 P31424 99686 200.26 Membrane receptor 20024,20796 46751,51157 IC50,IC50 IC50,Ki Pyrimidinergic receptor P2Y6 6.82102305271 6.88605664769 Q15077 Q63371 361881 483.057 Membrane receptor 31866 31866,49584 IC50 IC50,IC50 Metabotropic glutamate receptor 5 8.26143937264 7.92081875395 P41594 P31424 100257 193.244 Membrane receptor 35537,36099 31368,35537,36024,36835,36835,37490,38151,38151,46751,50238,50238 Ki,IC50 IC50,Ki,Ki,IC50,Ki,Ki,IC50,Ki,IC50,Ki,Ki Adenosine A1 receptor 5.87289520164 7.22184874962 P30542 P25099 100299 256.26 Membrane receptor 16115 9678,17675,148 IC50 IC50,Ki,Ki Adenosine A1 receptor 5.0 5.7447274949 P30542 P25099 101358 203.244 Membrane receptor 46210 11175 Ki Ki Adenosine A1 receptor 5.13076828027 4.33724216832 P30542 P25099 102004 163.18 Membrane receptor 46210 11175 Ki Ki Adenosine A3 receptor 8.02227639471 5.74714696902 P33765 P28647 364465 438.44 Membrane receptor 34747 34747 Ki Ki Adenosine A3 receptor 8.88605664769 6.50584540598 P33765 P28647 364592 430.461 Membrane receptor 34747 34747 Ki Ki Androgen Receptor 7.36957212497 6.7878123956 P10275 P15207 364605 427.797 Transcription Factor 34749 34749 IC50 IC50 Androgen Receptor 8.59522014268 6.53580207387 P10275 P15207 364795 327.292 Transcription Factor 34764,34764 34764,34764 Ki,Ki IC50,IC50 Androgen Receptor 8.45593195565 8.35654732351 P10275 P15207 364981 327.292 Transcription Factor 34764 34764 Ki IC50 Androgen Receptor 8.75084472311 7.68760121052 P10275 P15207 364982 327.292 Transcription Factor 34764,34764 34764,34764 Ki,Ki IC50,IC50 Cannabinoid CB1 receptor 9.52287874528 9.06550154876 P21554 P20272 364983 515.955 Membrane receptor 34762,36167,38671,43931,47927,48817,48817,50608,51391,52033 45882 IC50,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50,IC50 IC50 Androgen Receptor 9.0 6.41453927049 P10275 P15207 364988 337.329 Transcription Factor 34764 34764 Ki IC50 Androgen Receptor 8.25963731051 8.20065945055 P10275 P15207 364989 307.303 Transcription Factor 34764 34764 Ki IC50 Androgen Receptor 7.61978875829 6.58502665203 P10275 P15207 364996 317.341 Transcription Factor 34764 34764 Ki IC50 Histamine H3 receptor 8.57426054148 8.09 Q9Y5N1 Q9QYN8 627167 361.454 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Histamine H3 receptor 8.84794000867 7.93 Q9Y5N1 Q9QYN8 627168 361.454 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Histamine H3 receptor 8.85948500217 8.3 Q9Y5N1 Q9QYN8 627169 377.908 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Androgen Receptor 6.79048498546 6.92233198127 P10275 P15207 102911 430.373 Transcription Factor 35490,35490,35972,35972,36333,36333,36717,36717,37004,37004,38475,38475,38697,38697,38697,39522,39522,43799,43799,51143,51143,51964,51964,51964,54081,54081 34890,45812 IC50,IC50,IC50,Ki,IC50,Ki,IC50,Ki,IC50,IC50,Ki,IC50,IC50,Ki,IC50,IC50,Ki,Ki,IC50,IC50,IC50,Ki,IC50,IC50,IC50,IC50 IC50,Ki Histamine H3 receptor 8.94102999566 8.59 Q9Y5N1 Q9QYN8 627235 377.908 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Histamine H3 receptor 8.64989437914 7.9 Q9Y5N1 Q9QYN8 627236 368.473 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Histamine H3 receptor 8.59360807164 8.21 Q9Y5N1 Q9QYN8 627237 375.48 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Histamine H3 receptor 8.82242501084 8.51 Q9Y5N1 Q9QYN8 627238 382.499 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Histamine H3 receptor 9.34695437047 8.64 Q9Y5N1 Q9QYN8 627309 403.49 Membrane receptor 51148,51148 51148 Ki,IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.13076828027 7.21467016499 P36544 Q05941 632814 266.341 Ion channel 51372 51372 IC50 Ki P2X purinoceptor 7 7.03151705145 6.82102305271 Q99572 Q64663 467412 490.0 Ion channel 43867 43867 IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 7.49148333035 8.22184874962 P28845 P16232 365476 438.486 Enzyme 34818,34818 34818 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.98940535047 8.52287874528 P28845 P16232 365500 346.388 Enzyme 34818,34818 34818 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.72488582347 7.28399665637 P28845 P16232 365663 388.476 Enzyme 34818,34818 34818 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 8.03786035697 7.88605664769 P28845 P16232 365664 412.522 Enzyme 34818,34818 34818 Ki,IC50 Ki Renin 8.69897000434 6.39794000867 P00797 P08424 82009 730.012 Enzyme 9855,9855,9855,9855,9855 9855 IC50,IC50,IC50,IC50,IC50 IC50 Cannabinoid CB1 receptor 8.61828600322 9.15490195999 P21554 P20272 627910 541.856 Membrane receptor 50972,50972 50972 IC50,IC50 IC50 Cannabinoid CB2 receptor 5.82390874094 5.82390874094 P34972 Q9QZN9 627910 541.856 Membrane receptor 50972 50972 IC50 IC50 Glucagon receptor 7.7447274949 7.17866883428 P47871 P30082 366040 566.475 Membrane receptor 34824,45153 34824,45153 IC50,IC50 IC50,IC50 Gastric inhibitory polypeptide receptor 7.19382002602 6.66554624885 P48546 P43219 366040 566.475 Membrane receptor 45153 45153 IC50 IC50 Prolyl endopeptidase 8.82390874094 8.88605664769 P48147 O70196 630034 384.535 Enzyme 51017 51017 Ki Ki Adenosine A3 receptor 7.55284196866 8.02227639471 P33765 P28647 105982 483.26 Membrane receptor 3885 15464 Ki Ki Cathepsin K 8.31875876262 7.23657200644 P43235 O35186 630328 515.643 Enzyme 51289 51289 IC50 IC50 Serotonin 2a (5-HT2a) receptor 8.95860731484 8.63827216398 P28223 P14842 368556 319.392 Membrane receptor 34921 34921 IC50 IC50 Histamine H3 receptor 7.95860731484 7.45593195565 Q9Y5N1 Q9QYN8 438904 231.376 Membrane receptor 38490 38490 Ki Ki Glycine transporter 1 7.89962945488 7.99567862622 P48067 P28572 368844 489.988 Transporter 34944 34944 IC50 IC50 Glycine transporter 1 8.07572071394 7.70553377384 P48067 P28572 368987 507.979 Transporter 34944 34944 IC50 IC50 Glycine transporter 1 7.90308998699 7.65560772631 P48067 P28572 368988 489.988 Transporter 34944 34944 IC50 IC50 Glycine transporter 1 8.20065945055 8.13076828027 P48067 P28572 368995 524.434 Transporter 34944 34944 IC50 IC50 Glycine transporter 1 8.01322826573 7.73754891027 P48067 P28572 369003 471.998 Transporter 34944 34944 IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 7.47539098866 7.79588001734 P28845 P16232 369013 313.222 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 8.08374554365 8.09691001301 P28845 P16232 369021 341.275 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.89257807598 8.39794000867 P28845 P16232 369028 325.233 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.174360993 5.56863623584 P28845 P16232 369045 390.306 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 6.64672644868 6.67778070527 P28845 P16232 369046 392.322 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.36996430601 8.2757241304 P28845 P16232 369053 327.249 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 6.79929972961 8.39794000867 P28845 P16232 369059 399.311 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.09022803223 7.16749108729 P28845 P16232 369076 466.444 Enzyme 34972,34972 34972 Ki,IC50 Ki Adenosine A2a receptor 8.5376020021 7.60205999133 P29274 P30543 440013 451.565 Membrane receptor 38555 38555 Ki Ki 11-beta-hydroxysteroid dehydrogenase 1 6.15490195999 7.69897000434 P28845 P16232 369098 428.31 Enzyme 34972 34972 Ki Ki Transient receptor potential cation channel subfamily A member 1 7.67778070527 7.18045606446 O75762 Q6RI86 631244 395.131 NA 51267,51267,51267 51267 IC50,IC50,IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 6.03993833685 8.28399665637 P28845 P16232 369104 424.364 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.0 8.22184874962 P28845 P16232 369135 379.284 Enzyme 34972 34972 Ki Ki 11-beta-hydroxysteroid dehydrogenase 1 7.09793028383 7.85387196432 P28845 P16232 369136 388.289 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.36062319952 7.7447274949 P28845 P16232 369142 408.322 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.08247194914 7.63827216398 P28845 P16232 369143 451.346 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.12785350844 8.30102999566 P28845 P16232 369150 394.298 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.15313652554 6.85387196432 P28845 P16232 369151 420.289 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.53174312876 6.79588001734 P28845 P16232 369158 434.316 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 7.38838186345 7.40893539297 P28845 P16232 369159 385.288 Enzyme 34972,34972 34972 Ki,IC50 Ki Transient receptor potential cation channel subfamily A member 1 5.85387196432 8.42021640338 O75762 Q6RI86 631337 409.158 NA 51267 51267 IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 6.25181197299 8.04575749056 P28845 P16232 369236 453.405 Enzyme 34972 34972 Ki Ki 11-beta-hydroxysteroid dehydrogenase 1 5.95860731484 7.76955107862 P28845 P16232 369245 441.395 Enzyme 34972 34972 Ki Ki Transient receptor potential cation channel subfamily A member 1 5.95860731484 7.82390874094 O75762 Q6RI86 631466 361.072 NA 51267 51267 IC50 IC50 Histamine H3 receptor 9.25181197299 8.5376020021 Q9Y5N1 Q9QYN8 631496 422.586 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.46852108296 8.63827216398 Q9Y5N1 Q9QYN8 631497 414.566 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.45593195565 8.72124639905 Q9Y5N1 Q9QYN8 631498 414.566 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.5376020021 9.45593195565 Q9Y5N1 Q9QYN8 631499 433.496 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.10790539731 7.44369749923 Q9Y5N1 Q9QYN8 631568 431.957 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.79588001734 9.39794000867 Q9Y5N1 Q9QYN8 631569 431.957 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.38721614328 9.22914798836 Q9Y5N1 Q9QYN8 631570 430.972 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.5376020021 8.07058107429 Q9Y5N1 Q9QYN8 631649 373.514 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.44369749923 9.10790539731 Q9Y5N1 Q9QYN8 631650 426.576 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.07058107429 8.30980391997 Q9Y5N1 Q9QYN8 631652 364.507 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.92081875395 9.30102999566 Q9Y5N1 Q9QYN8 631653 370.49 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.43179827593 8.76955107862 Q9Y5N1 Q9QYN8 631732 368.474 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.39794000867 8.63827216398 Q9Y5N1 Q9QYN8 631733 374.475 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.49485002168 8.92081875395 Q9Y5N1 Q9QYN8 631734 347.477 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.18708664336 8.63827216398 Q9Y5N1 Q9QYN8 631735 393.545 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.49485002168 8.55284196866 Q9Y5N1 Q9QYN8 631806 414.566 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.76955107862 7.95860731484 Q9Y5N1 Q9QYN8 631807 420.593 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.05060999336 8.30980391997 Q9Y5N1 Q9QYN8 631808 404.528 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.16115090926 8.55284196866 Q9Y5N1 Q9QYN8 631885 358.44 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.72124639905 8.95860731484 Q9Y5N1 Q9QYN8 631953 441.571 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.13076828027 8.67778070527 Q9Y5N1 Q9QYN8 631954 465.417 Membrane receptor 51341 51341 Ki Ki Anandamide amidohydrolase 7.36653154442 5.60205999133 O00519 P97612 369814 257.328 Enzyme 38447 38493,38493,44028,44843,44843 IC50 Ki,IC50,IC50,Ki,IC50 Anandamide amidohydrolase 7.49485002168 7.52287874528 O00519 P97612 369820 301.337 Enzyme 35154 38493,38493,44843,44843 Ki Ki,IC50,Ki,IC50 Anandamide amidohydrolase 9.0 9.39794000867 O00519 P97612 369858 282.337 Enzyme 35154 38493,38493,38830,44843,44843 Ki Ki,IC50,Ki,Ki,IC50 Histamine H3 receptor 8.95860731484 8.22914798836 Q9Y5N1 Q9QYN8 632017 479.54 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.16749108729 7.50863830617 Q9Y5N1 Q9QYN8 632018 399.551 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 7.60205999133 7.23657200644 Q9Y5N1 Q9QYN8 632019 498.563 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 7.67778070527 7.14874165128 Q9Y5N1 Q9QYN8 632020 418.617 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.95860731484 8.16749108729 Q9Y5N1 Q9QYN8 632089 399.551 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.92081875395 9.52287874528 Q9Y5N1 Q9QYN8 632090 409.523 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.0 8.63827216398 Q9Y5N1 Q9QYN8 632091 399.571 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 10.3010299957 10.096910013 Q9Y5N1 Q9QYN8 632092 337.502 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.76955107862 8.85387196432 Q9Y5N1 Q9QYN8 632195 408.538 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.72124639905 9.18045606446 Q9Y5N1 Q9QYN8 632197 318.415 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.0 8.44369749923 Q9Y5N1 Q9QYN8 632198 322.467 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.44369749923 8.65757731918 Q9Y5N1 Q9QYN8 632262 345.481 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.00877392431 8.25963731051 Q9Y5N1 Q9QYN8 632264 388.505 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 6.63827216398 6.0 Q9Y5N1 Q9QYN8 632265 401.425 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 7.55284196866 7.25963731051 Q9Y5N1 Q9QYN8 632335 469.429 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.72124639905 8.85387196432 Q9Y5N1 Q9QYN8 632336 351.508 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.95860731484 9.30102999566 Q9Y5N1 Q9QYN8 632337 317.427 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.65757731918 8.72124639905 Q9Y5N1 Q9QYN8 632338 317.427 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.13076828027 7.38721614328 Q9Y5N1 Q9QYN8 632403 240.343 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 7.92081875395 7.18708664336 Q9Y5N1 Q9QYN8 632404 254.37 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.13076828027 7.32790214206 Q9Y5N1 Q9QYN8 632405 280.407 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 7.95860731484 7.2924298239 Q9Y5N1 Q9QYN8 632468 296.45 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.60205999133 8.16115090926 Q9Y5N1 Q9QYN8 632470 322.467 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.03151705145 8.26760624018 Q9Y5N1 Q9QYN8 632471 334.458 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.79588001734 9.16749108729 Q9Y5N1 Q9QYN8 632472 334.458 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.69897000434 8.82390874094 Q9Y5N1 Q9QYN8 632525 320.431 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.49485002168 7.85387196432 Q9Y5N1 Q9QYN8 632526 306.405 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.45593195565 7.79588001734 Q9Y5N1 Q9QYN8 632528 379.452 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.14874165128 8.26760624018 Q9Y5N1 Q9QYN8 632529 393.479 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.25181197299 8.82390874094 Q9Y5N1 Q9QYN8 632618 335.443 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.7447274949 8.25963731051 Q9Y5N1 Q9QYN8 632619 386.286 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.42021640338 7.76955107862 Q9Y5N1 Q9QYN8 632621 325.471 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.45593195565 8.85387196432 Q9Y5N1 Q9QYN8 632622 415.554 Membrane receptor 51341 51341 Ki Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.92081875395 7.45593195565 P36544 Q05941 632726 322.427 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.56863623584 7.02227639471 P36544 Q05941 632815 306.362 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.48148606012 7.48148606012 P36544 Q05941 632816 322.427 Ion channel 51372 51372 IC50 Ki Sodium channel protein type X alpha subunit 7.0 6.67778070527 Q9Y5Y9 Q62968 710667 320.36 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 7.65757731918 7.07058107429 Q9Y5Y9 Q62968 710669 322.788 Ion channel 53444 53444 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 6.09691001301 8.11918640772 P36544 Q05941 632918 306.365 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.15490195999 8.95860731484 P36544 Q05941 632919 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.7447274949 7.82390874094 P36544 Q05941 632920 373.375 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.33724216832 7.13667713988 P36544 Q05941 632921 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.32790214206 8.35654732351 P36544 Q05941 632999 305.374 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.2757241304 8.5376020021 P36544 Q05941 633000 321.439 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.52287874528 9.52287874528 P36544 Q05941 633001 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.0 9.69897000434 P36544 Q05941 633002 304.389 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.55284196866 8.52287874528 P36544 Q05941 633003 372.387 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.40893539297 8.0 P36544 Q05941 633071 304.389 Ion channel 51372 51372 IC50 Ki Gonadotropin-releasing hormone receptor 9.69897000434 7.22184874962 P30968 P30969 109406 657.769 Membrane receptor 31350,42049 31350,42049 IC50,IC50 IC50,IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.82390874094 8.50863830617 P36544 Q05941 633823 322.427 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.95860731484 9.04575749056 P36544 Q05941 633824 306.365 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.04575749056 9.39794000867 P36544 Q05941 633825 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.92081875395 8.67778070527 P36544 Q05941 633897 373.375 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.56863623584 7.88605664769 P36544 Q05941 633898 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.25181197299 7.7447274949 P36544 Q05941 633901 266.341 Ion channel 51372 51372 IC50 Ki Cathepsin S 8.96040937698 8.76955107862 P25774 Q02765 372597 527.675 Enzyme 37689,42511 37689 IC50,IC50 IC50 Cathepsin L 8.19951355216 8.38721614328 P07711 P07154 372597 527.675 Enzyme 37689,42511 37689 IC50,IC50 IC50 Cathepsin B 5.60643135489 6.13371266092 P07858 P00787 372597 527.675 Enzyme 37689,42511 37689 IC50,IC50 IC50 Adenosine A3 receptor 6.55206782438 6.58502665203 P33765 P28647 110480 335.358 Membrane receptor 3885,30314,38198,39088,44049,49741 16866,15464,30314 Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki,Ki Adenosine A2a receptor 5.94108472729 6.23657200644 P29274 P30543 110480 335.358 Membrane receptor 30314,38198,39088,44049 14372,14372,3885,15396,15464,16866,49741 Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki,Ki,Ki,Ki Adenosine A1 receptor 8.32390874094 7.99700886368 P30542 P25099 110480 335.358 Membrane receptor 30314,38198,39088,44049 14372,14372,9678,9678,9748,9679,9679,127,11687,14372,14372,14372,14372,11295,11295,11295,13861,13861,10854,9748,3885,4712,9901,10663,41516,49741,49741,49741 Ki,Ki,Ki,Ki IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,IC50,IC50 Vasopressin V2 receptor 8.49485002168 8.50863830617 P30518 Q00788 110739 476.354 Membrane receptor 4138,14475 4138,14475 IC50,IC50 IC50,IC50 Vasopressin V1a receptor 7.82390874094 7.63827216398 P37288 P30560 110739 476.354 Membrane receptor 4138,14475 4138,14475 IC50,IC50 IC50,IC50 Adenosine A2a receptor 9.69897000434 9.69897000434 P29274 P30543 373013 464.495 Membrane receptor 44049 35271 Ki Ki Bradykinin B1 receptor 9.30102999566 6.92445303861 P46663 P97583 373122 490.92 Membrane receptor 35288 35288 Ki Ki Bradykinin B1 receptor 8.22184874962 7.92081875395 P46663 P97583 373127 490.92 Membrane receptor 35288 35288 Ki Ki Bradykinin B1 receptor 9.15490195999 7.44733178389 P46663 P97583 373156 483.347 Membrane receptor 35288 35288 Ki Ki Bradykinin B1 receptor 9.39794000867 7.45222529461 P46663 P97583 373197 466.892 Membrane receptor 35288 35288 Ki Ki Bradykinin B1 receptor 9.30102999566 7.09151498112 P46663 P97583 373211 490.917 Membrane receptor 35288 35288 Ki Ki Neurokinin 3 receptor 8.05551732785 7.18045606446 P29371 P16177 368221 427.452 Membrane receptor 34911 34911 IC50 IC50 Cannabinoid CB1 receptor 7.67778070527 8.0 P21554 P20272 374473 426.507 Membrane receptor 21631,30511,30590,35365,35375,35863,37625,37625,37843,37904,39110,42403,42742,44405,46289,46425,49092,49092,49843,52442 41874,46425,49092 Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,IC50,Ki,Ki IC50,Ki,IC50 Cannabinoid CB2 receptor 8.67778070527 7.24074303006 P34972 Q9QZN9 374473 426.507 Membrane receptor 20667,30511,30560,35365,35863,37625,37625,37843,37843,37904,39110,39110,44405,44405,46289,46425,49092,49092,49092,49843,52442 41874,49092 Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,IC50,Ki,Ki,IC50,Ki,IC50,Ki,Ki,Ki,IC50,IC50,Ki,Ki IC50,IC50 Metabotropic glutamate receptor 1 7.34678748622 7.65269740053 Q13255 P23385 374837 391.274 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.40893539297 6.99614744282 Q13255 P23385 374838 353.398 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 6.91364016933 7.2076083105 Q13255 P23385 374846 362.408 Membrane receptor 35368 35368 IC50 Ki Metabotropic glutamate receptor 1 6.60032627852 6.72401896707 Q13255 P23385 374847 350.437 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 8.04575749056 8.13380312009 Q13255 P23385 374856 350.437 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 6.55129368009 6.80588721374 Q13255 P23385 374866 336.411 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.69897000434 7.69897000434 Q13255 P23385 374867 322.384 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.7447274949 6.7447274949 Q13255 P23385 374878 364.464 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 5.07058107429 5.07058107429 Q13255 P23385 374888 378.491 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.19928292172 6.19928292172 Q13255 P23385 374900 286.352 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.77728352885 6.77728352885 Q13255 P23385 374901 300.379 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 8.30102999566 8.30102999566 Q13255 P23385 374909 314.405 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.30102999566 7.30102999566 Q13255 P23385 374910 328.432 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.88605664769 6.88605664769 Q13255 P23385 374911 342.458 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.31695296176 6.31695296176 Q13255 P23385 374917 342.458 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.85387196432 6.85387196432 Q13255 P23385 374918 342.458 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 9.0 9.0 Q13255 P23385 374923 342.458 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.88605664769 7.88605664769 Q13255 P23385 374928 356.485 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.11918640772 7.11918640772 Q13255 P23385 374929 380.506 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.47495519296 6.47495519296 Q13255 P23385 374934 316.421 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.58502665203 7.58502665203 Q13255 P23385 374935 328.432 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.85698519975 6.85698519975 Q13255 P23385 374936 342.458 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 5 6.05060999336 6.30102999566 P41594 P31424 374941 336.411 Membrane receptor 35368 35368 IC50 Ki Metabotropic glutamate receptor 1 8.30102999566 8.5 Q13255 P23385 374941 336.411 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.35654732351 7.35654732351 Q13255 P23385 374943 364.464 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.30102999566 7.15269740053 Q13255 P23385 374960 338.384 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.63827216398 7.8675910885 Q13255 P23385 374961 340.375 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 5 5.74232142513 5.98716277529 P41594 P31424 374970 356.829 Membrane receptor 35368 35368 IC50 Ki Metabotropic glutamate receptor 1 7.79588001734 8.09691001301 Q13255 P23385 374970 356.829 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 8.39794000867 8.69897000434 Q13255 P23385 374971 401.28 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.49485002168 7.79588001734 Q13255 P23385 374978 390.382 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.76955107862 8.08374554365 Q13255 P23385 374979 350.437 Membrane receptor 35368 35368,44256 IC50 Ki,IC50 Metabotropic glutamate receptor 1 7.43179827593 7.43179827593 Q13255 P23385 374995 364.464 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.14874165128 7.14874165128 Q13255 P23385 375006 394.49 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.94692155652 6.94692155652 Q13255 P23385 375016 362.448 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.38721614328 7.38721614328 Q13255 P23385 375022 362.448 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.30980391997 7.30980391997 Q13255 P23385 375023 361.42 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.0043648054 7.0043648054 Q13255 P23385 375028 404.409 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.00877392431 7.00877392431 Q13255 P23385 375029 336.411 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.51427857352 6.51427857352 Q13255 P23385 375036 366.437 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.07572071394 7.07572071394 Q13255 P23385 375094 378.491 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 6.99567862622 6.99567862622 Q13255 P23385 375095 406.544 Membrane receptor 35368 44256 IC50 IC50 Histamine H3 receptor 9.55284196866 8.69897000434 Q9Y5N1 Q9QYN8 632263 370.49 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.0 7.14266750357 Q9Y5N1 Q9QYN8 438953 231.376 Membrane receptor 38490 38490 Ki Ki Neprilysin 8.26760624018 9.22184874962 P08473 P07861 376146 395.92 Enzyme 35497,35497,35497 35497 IC50,IC50,IC50 IC50 Dipeptidyl peptidase IV 6.95078197733 7.00086945871 P27487 P14740 376387 317.449 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.95860731484 7.70996538864 P27487 P14740 376388 303.422 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.10237290871 7.98716277529 P27487 P14740 376389 348.42 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.7166987713 7.67778070527 P27487 P14740 376410 322.383 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.31875876262 8.21467016499 P27487 P14740 376411 333.448 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.28819277096 7.26042765555 P27487 P14740 376412 307.411 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.23657200644 7.99567862622 P27487 P14740 376419 321.413 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.15490195999 7.87289520164 P27487 P14740 376420 337.867 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.34294414714 7.25884840115 P27487 P14740 376421 311.83 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.18708664336 7.97061622231 P27487 P14740 376428 382.319 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.59516628338 7.51712641639 P27487 P14740 376429 303.383 Enzyme 35539,45969 45969 IC50,IC50 IC50 Dipeptidyl peptidase IV 6.2612917627 6.21681130892 P27487 P14740 376430 186.275 Enzyme 35539,37469 37469 IC50,IC50 IC50 Dipeptidyl peptidase IV 6.83268266525 6.72124639905 P27487 P14740 376469 277.385 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.59859945922 7.47366072261 P27487 P14740 376470 302.395 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 6.74232142513 6.76700388961 P27487 P14740 376471 291.412 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.42945706012 7.46724562101 P27487 P14740 376479 330.405 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 6.81247927916 6.82102305271 P27487 P14740 376488 320.41 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.06600683617 7.11804502866 P27487 P14740 376495 345.419 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.01772876696 7.86646109163 P27487 P14740 376501 330.448 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.14874165128 7.90308998699 P27487 P14740 376502 358.501 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.04095860768 8.30102999566 P27487 P14740 376509 372.527 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 8.19382002602 8.03151705145 P27487 P14740 376510 431.553 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.86646109163 7.81530856918 P27487 P14740 376518 402.51 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.85698519975 7.78251605579 P27487 P14740 376519 373.473 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.77469071827 7.7878123956 P27487 P14740 376526 374.457 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.76955107862 7.63827216398 P27487 P14740 376527 360.474 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 6.642065153 6.77469071827 P27487 P14740 376534 445.537 Enzyme 35539 35539 IC50 IC50 Dipeptidyl peptidase IV 7.57839607313 7.40893539297 P27487 P14740 376535 303.422 Enzyme 35539 35539 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.65757731918 7.31875876262 Q92633 P61794 412317 460.931 Membrane receptor 37582 37582 IC50 IC50 Metabotropic glutamate receptor 5 8.61978875829 8.55063740921 P41594 P31424 376818 240.3 Membrane receptor 35537,35537,35537,35537,35537 35537,51237 Ki,IC50,Ki,IC50,IC50 Ki,Ki Butyrylcholinesterase 8.24718356881 6.82681373159 P06276 Q9JKC1 47469 492.697 Enzyme 37270 3267,31775,42156 IC50 IC50,IC50,IC50 Acetylcholinesterase 9.16033148474 8.82390874094 P22303 P37136 47469 492.697 Enzyme 21244,37270 3267,31775,42156 IC50,IC50 IC50,IC50,IC50 Nitric-oxide synthase, brain 5.35654732351 5.28191867648 P29475 P29476 377219 219.199 Enzyme 46991 46991,53925 IC50 IC50,Ki Glutamate receptor ionotropic, AMPA 4 6.06148027482 4.73426054148 P48058 P19493 116265 147.129 Ion channel 14175 38673,45271,47617,50876 Ki IC50,Ki,IC50,IC50 Metabotropic glutamate receptor 8 8.24412514433 5.46852108296 O00222 P70579 116265 147.129 Membrane receptor 20685 30522,36453 IC50 Ki,Ki Glutamate receptor ionotropic, AMPA 1 5.86646109163 4.45593195565 P42261 P19490 116265 147.129 Ion channel 14175 38673,45271,47617,50876,50876 Ki IC50,Ki,IC50,IC50,IC50 Glutamate receptor ionotropic, AMPA 2 6.0268721464 3.85387196432 P42262 P19491 116265 147.129 Ion channel 14175 38673,45271,47617,50876,51222 Ki IC50,Ki,IC50,IC50,Ki Metabotropic glutamate receptor 1 6.42309256783 5.13667713988 Q13255 P23385 116265 147.129 Membrane receptor 36681,45031 36453 Ki,Ki IC50 Metabotropic glutamate receptor 5 6.17223870187 5.92081875395 P41594 P31424 116265 147.129 Membrane receptor 36681,45031 36453 Ki,Ki IC50 Glutamate receptor ionotropic kainate 2 5.95624487303 6.4788619163 Q13002 P42260 116265 147.129 Ion channel 15441 38673,43825,45271,47617,51222 Ki IC50,Ki,Ki,IC50,Ki Metabotropic glutamate receptor 4 5.73683036131 5.46852108296 Q14833 P31423 116265 147.129 Membrane receptor 36681,45031 30522,36453,36453 Ki,Ki Ki,IC50,Ki Cannabinoid CB2 receptor 7.20065945055 7.04095860768 P34972 Q9QZN9 378616 449.254 Membrane receptor 35787,38328,45100,46158,48965 35787 IC50,IC50,IC50,IC50,IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 7.5 8.22184874962 P28845 P16232 369026 353.286 Enzyme 34972,34972 34972 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 6.23298694697 7.85387196432 P28845 P16232 369087 456.363 Enzyme 34972,34972 34972 Ki,IC50 Ki Histamine H3 receptor 9.82390874094 9.34678748622 Q9Y5N1 Q9QYN8 632401 331.454 Membrane receptor 51341 51341 Ki Ki Transient receptor potential cation channel subfamily A member 1 7.04095860768 6.93930215965 O75762 Q6RI86 631245 425.157 NA 51267,51267,51267 51267 IC50,IC50,IC50 IC50 Transient receptor potential cation channel subfamily A member 1 5.92006607645 8.39794000867 O75762 Q6RI86 631248 419.71 NA 51267,51267,51267,51267,51267,51267 51267 IC50,IC50,IC50,IC50,IC50,IC50 IC50 Adenosine A1 receptor 5.63827216398 6.24872089602 P30542 P25099 500259 562.564 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 7.15864052955 6.19722627471 P29274 P30543 500259 562.564 Membrane receptor 46829 46829 Ki Ki Vanilloid receptor 7.68225812659 7.43179827593 Q8NER1 O35433 380474 423.568 Ion channel 30167,30167 35885,35885,46701,49387,49776 IC50,IC50 Ki,Ki,IC50,IC50,IC50 Monoamine oxidase A 6.87614835903 6.61083391564 P21397 P21396 380636 181.298 Enzyme 35838 35838 Ki Ki Monoamine oxidase A 7.12493873661 7.26760624018 P21397 P21396 380637 195.324 Enzyme 35838 35838 Ki Ki Monoamine oxidase B 4.85294232897 1.82390874094 P27338 P19643 380638 209.351 Enzyme 35838 35838 Ki Ki Monoamine oxidase A 7.52287874528 6.93930215965 P21397 P21396 380638 209.351 Enzyme 35838 35838 Ki Ki Monoamine oxidase B 5.339134522 5.04939177522 P27338 P19643 380639 223.378 Enzyme 35838 35838 Ki Ki Monoamine oxidase A 7.65757731918 6.40671393298 P21397 P21396 380639 223.378 Enzyme 35838 35838 Ki Ki Dipeptidyl peptidase IV 8.69897000434 7.46040937698 P27487 P14740 643458 364.401 Enzyme 34705,34705 34705,34705 Ki,Ki Ki,Ki Adenosine A3 receptor 4.06550154876 4.03529053714 P33765 P28647 381693 180.164 Membrane receptor 15855,15563,20724,30321,31281,31341,36623,46829,42133,46235,49741,49760 46829,49741 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A2b receptor 5.04239271294 4.82102305271 P29275 P29276 381693 180.164 Membrane receptor 20724,30250,31281,46829,49741,49760,51928 16424,46829,49741 Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki,Ki Adenosine A1 receptor 5.2076083105 5.04190467001 P30542 P25099 381693 180.164 Membrane receptor 17602,20724,30321,31281,31341,36623,46829,42133,46235,49741,49760 11377,12700,11687,11377,9562,9562,11292,11292,10574,46829,43227,49741 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Adenosine A2a receptor 5.10237290871 4.65757731918 P29274 P30543 381693 180.164 Membrane receptor 20724,30321,31281,31341,36623,46829,42133,46235,49741,49760 46829,43227,49741 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki,Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.52287874528 6.61978875829 P36544 Q05941 643934 294.348 Ion channel 45299 51501 IC50 Ki Androgen Receptor 8.76582633479 8.10790539731 P10275 P15207 381838 305.716 Transcription Factor 35979,35979,36077,36077,36821,47060 47060 IC50,Ki,Ki,IC50,Ki,Ki IC50 Androgen Receptor 8.22184874962 8.19382002602 P10275 P15207 381840 291.733 Transcription Factor 36077,36077,47060 47060 Ki,IC50,Ki IC50 Androgen Receptor 8.79588001734 8.26760624018 P10275 P15207 381842 305.759 Transcription Factor 36077,36077,47060 47060 Ki,IC50,Ki IC50 Androgen Receptor 9.04575749056 8.7447274949 P10275 P15207 381843 319.786 Transcription Factor 36077,36077,47060 47060 Ki,IC50,Ki IC50 Butyrylcholinesterase 5.80687540165 6.98422124361 P06276 Q9JKC1 119802 337.416 Enzyme 10673,10673,21519 50487 IC50,IC50,IC50 IC50 Acetylcholinesterase 7.65659252275 7.92445303861 P22303 P37136 119802 337.416 Enzyme 10673,10673,21519,52762 50487 IC50,IC50,IC50,IC50 IC50 Dihydrofolate reductase 5.5376020021 1.39685562738 P00374 Q920D2 382012 335.426 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.22184874962 2.06449273418 P00374 Q920D2 382013 335.426 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.23657200644 2.49485002168 P00374 Q920D2 382014 330.365 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.56863623584 1.99567862622 P00374 Q920D2 382015 364.263 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.55284196866 1.08830984125 P00374 Q920D2 382018 353.269 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.85387196432 2.93181413825 P00374 Q920D2 382019 354.258 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.5376020021 1.49757288002 P00374 Q920D2 382021 315.393 Enzyme 36076 36076 IC50 IC50 Dihydrofolate reductase 5.23657200644 3.89254497679 P00374 Q920D2 382022 345.419 Enzyme 36076 36076,43976 IC50 IC50,IC50 Dihydrofolate reductase 4.7447274949 3.75181197299 P00374 Q920D2 382024 285.367 Enzyme 36076 36076,43976 IC50 IC50,IC50 Dihydrofolate reductase 5.85387196432 2.44977164694 P00374 Q920D2 382025 336.414 Enzyme 36076 36076 IC50 IC50 Butyrylcholinesterase 6.89350690763 8.23657200644 P06276 Q9JKC1 119989 367.441 Enzyme 10673,10673 50487 IC50,IC50 IC50 Acetylcholinesterase 6.54710205982 7.52432881168 P22303 P37136 119989 367.441 Enzyme 10673,10673 50487 IC50,IC50 IC50 Anandamide amidohydrolase 8.92081875395 9.04575749056 O00519 P97612 382554 403.302 Enzyme 36082 36082 Ki Ki Anandamide amidohydrolase 9.34678748622 8.88605664769 O00519 P97612 382560 384.427 Enzyme 36082 36082,38493 Ki Ki,Ki Anandamide amidohydrolase 8.30102999566 9.0 O00519 P97612 382564 384.427 Enzyme 36082,38493 36082,38493,38493,38493 Ki,Ki Ki,Ki,Ki,IC50 Anandamide amidohydrolase 8.5376020021 9.12493873661 O00519 P97612 382570 354.401 Enzyme 36082,38493 36082,38493,38493,38493 Ki,Ki Ki,Ki,Ki,IC50 Vanilloid receptor 6.76143937264 6.14367514919 Q8NER1 O35433 382654 373.329 Ion channel 36134,36134 36134,36134 IC50,IC50 IC50,IC50 Vanilloid receptor 8.44119865415 8.17827366176 Q8NER1 O35433 382655 354.448 Ion channel 36134,36134 36134,36134 IC50,IC50 IC50,IC50 Vanilloid receptor 9.37236374745 8.26362177534 Q8NER1 O35433 382656 366.339 Ion channel 36134,36134 36134,36134 IC50,IC50 IC50,IC50 Vanilloid receptor 8.40427449277 8.11383914664 Q8NER1 O35433 382657 367.324 Ion channel 36134,36134 36134,36134,36135,36135 IC50,IC50 IC50,IC50,IC50,IC50 Serotonin 2a (5-HT2a) receptor 9.50863830617 9.04899855432 P28223 P14842 120674 373.461 Membrane receptor 51416 38805,46285,46285,46285 Ki Ki,Ki,Ki,Ki Vanilloid receptor 9.11918640772 9.04575749056 Q8NER1 O35433 382857 430.403 Ion channel 36135,36135,36135,38526,41998,41998,50778 36135,36135,36136,36136,37901,37901,38526,45756,45756,41998,41998 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 Histamine H3 receptor 9.11918640772 8.14266750357 Q9Y5N1 Q9QYN8 631805 317.427 Membrane receptor 51341 51341 Ki Ki Dopamine transporter 7.7447274949 8.24412514433 Q01959 P23977 382978 394.96 Transporter 36158 36158 Ki IC50 Dopamine transporter 7.92081875395 8.22184874962 Q01959 P23977 382979 412.951 Transporter 36158 36158 Ki IC50 Serotonin transporter 6.18508681872 6.43062609038 P31645 P31652 382979 412.951 Transporter 36158 36158 Ki Ki Dopamine transporter 7.55284196866 7.69897000434 Q01959 P23977 382980 429.405 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.62160209905 6.04431224969 P31645 P31652 382980 429.405 Transporter 36158 36158 Ki Ki Dopamine transporter 7.45593195565 6.97061622231 Q01959 P23977 382981 473.856 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.24412514433 6.07572071394 P31645 P31652 382981 473.856 Transporter 36158 36158 Ki Ki Dopamine transporter 7.40893539297 7.7447274949 Q01959 P23977 382982 473.856 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.82390874094 6.55284196866 P31645 P31652 382982 473.856 Transporter 36158 36158 Ki Ki Dopamine transporter 8.21467016499 7.69897000434 Q01959 P23977 382983 439.958 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.73992861201 6.00877392431 P31645 P31652 382983 439.958 Transporter 36158 36158 Ki Ki Dopamine transporter 8.11350927483 8.30102999566 Q01959 P23977 382984 439.958 Transporter 36158 36158 Ki IC50 Serotonin transporter 6.13076828027 6.52143350441 P31645 P31652 382984 439.958 Transporter 36158 36158 Ki Ki Dopamine transporter 8.06550154876 7.85387196432 Q01959 P23977 382985 424.986 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.28399665637 6.09691001301 P31645 P31652 382985 424.986 Transporter 36158 36158 Ki Ki Dopamine transporter 7.18045606446 6.35654732351 Q01959 P23977 382988 463.85 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.56703070913 6.42021640338 P31645 P31652 382988 463.85 Transporter 36158 36158 Ki Ki Dopamine transporter 6.63078414259 7.18708664336 Q01959 P23977 382989 455.012 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.44490555142 5.82102305271 P31645 P31652 382989 455.012 Transporter 36158 36158 Ki Ki Dopamine transporter 7.21467016499 7.92081875395 Q01959 P23977 382990 392.532 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.76447155309 5.64975198167 P31645 P31652 382990 392.532 Transporter 36158 36158 Ki Ki Dopamine transporter 6.67366413907 7.65757731918 Q01959 P23977 382991 408.987 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.87942606879 5.95467702121 P31645 P31652 382991 408.987 Transporter 36158 36158 Ki Ki Dopamine transporter 7.92081875395 8.0 Q01959 P23977 382993 453.438 Transporter 36158 36158 Ki IC50 Serotonin transporter 6.06048074738 6.50584540598 P31645 P31652 382993 453.438 Transporter 36158 36158 Ki Ki Dopamine transporter 6.85387196432 7.38721614328 Q01959 P23977 382995 419.539 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.78515615195 5.77211329539 P31645 P31652 382995 419.539 Transporter 36158 36158 Ki Ki Dopamine transporter 7.85387196432 8.39794000867 Q01959 P23977 382996 419.539 Transporter 36158 36158 Ki IC50 Serotonin transporter 6.23657200644 5.0 P31645 P31652 382996 419.539 Transporter 36158 36158 Ki Ki Dopamine transporter 7.2757241304 7.82390874094 Q01959 P23977 383010 404.568 Transporter 36158 36158 Ki IC50 Dopamine transporter 6.97881070093 6.99139982824 Q01959 P23977 383011 443.432 Transporter 36158 36158 Ki IC50 Serotonin transporter 5.53165266959 6.72124639905 P31645 P31652 383011 443.432 Transporter 36158 36158 Ki Ki Dopamine transporter 6.27654432796 7.08092190762 Q01959 P23977 383012 434.594 Transporter 36158 36158 Ki IC50 Vanilloid receptor 9.09691001301 9.21897258517 Q8NER1 O35433 383030 399.326 Ion channel 36135,36135,36135 36135,36135,41998,41998 IC50,IC50,IC50 IC50,IC50,IC50,IC50 Histamine H3 receptor 9.61092437481 8.00877392431 Q9Y5N1 Q9QYN8 383717 419.562 Membrane receptor 36041,36041 36041 IC50,Ki Ki Urotensin II receptor 8.37236374745 7.76955107862 Q9UKP6 P49684 646331 418.531 Membrane receptor 51448,51448 51448 IC50,Ki IC50 Urotensin II receptor 7.92081875395 6.22184874962 Q9UKP6 P49684 646392 536.729 Membrane receptor 51448 51448 Ki Ki Anandamide amidohydrolase 7.58502665203 7.76880100105 O00519 P97612 369880 378.421 Enzyme 35154,44028 38493,44028,44028,44028 Ki,Ki IC50,Ki,Ki,Ki Cannabinoid CB1 receptor 8.55284196866 8.63827216398 P21554 P20272 384382 501.039 Membrane receptor 35980 35980 IC50 IC50 Adenosine A1 receptor 5.52287874528 6.63827216398 P30542 P25099 122252 384.429 Membrane receptor 52381 2252,2252,37033,37600 Ki Ki,Ki,Ki,Ki Adenosine A2a receptor 7.83277312442 8.47865319091 P29274 P30543 122252 384.429 Membrane receptor 30254,38162,47546,52381 2252,37033,37600,38162 Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki Histamine H3 receptor 7.27518367476 7.55284196866 Q9Y5N1 Q9QYN8 501017 370.488 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.5 8.15490195999 Q9Y5N1 Q9QYN8 501019 233.22 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.22457399418 8.01913608199 Q9Y5N1 Q9QYN8 647352 385.887 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 8.69380100105 7.59989437914 Q9Y5N1 Q9QYN8 647410 369.433 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 9.63827216398 9.0 Q9Y5N1 Q9QYN8 632196 348.441 Membrane receptor 51341 51341 Ki Ki Monoglyceride lipase 5.0 3.69897000434 Q99685 Q8R431 123166 295.376 Enzyme 48666 52343 IC50 IC50 Histamine H3 receptor 8.33724216832 7.43179827593 Q9Y5N1 Q9QYN8 647456 385.498 Membrane receptor 51662 51662 Ki Ki Anandamide amidohydrolase 7.20065945055 7.20065945055 O00519 P97612 123224 295.376 Enzyme 45322 42205 IC50 IC50 Histamine H3 receptor 9.95860731484 9.2924298239 Q9Y5N1 Q9QYN8 632266 318.415 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.89360807164 8.02889035263 Q9Y5N1 Q9QYN8 648039 369.433 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 9.13693598216 8.04413608199 Q9Y5N1 Q9QYN8 648105 369.433 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 9.06736374745 7.98930365742 Q9Y5N1 Q9QYN8 648107 376.452 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 8.96327366176 8.12695437047 Q9Y5N1 Q9QYN8 648109 351.442 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 8.68959320386 8.08 Q9Y5N1 Q9QYN8 648180 420.332 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Histamine H3 receptor 7.76955107862 7.5324693683 Q9Y5N1 Q9QYN8 648181 371.861 Membrane receptor 51662 51662,51662 Ki IC50,Ki Histamine H3 receptor 9.03 8.06195437047 Q9Y5N1 Q9QYN8 648182 385.887 Membrane receptor 51662,51662 51662,51662 Ki,IC50 IC50,Ki Serotonin 2a (5-HT2a) receptor 6.97881070093 8.68193666504 P28223 P14842 335829 191.23 Membrane receptor 30538 30538 Ki IC50 Histamine H3 receptor 9.60205999133 9.31875876262 Q9Y5N1 Q9QYN8 632339 351.872 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.16115090926 8.40893539297 Q9Y5N1 Q9QYN8 632402 341.449 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 8.2924298239 7.69897000434 Q9Y5N1 Q9QYN8 632469 306.401 Membrane receptor 51341 51341 Ki Ki Cannabinoid CB1 receptor 7.82390874094 7.65757731918 P21554 P20272 387205 368.468 Membrane receptor 36602 36602 IC50 IC50 Histamine H3 receptor 9.05060999336 8.22914798836 Q9Y5N1 Q9QYN8 632527 306.405 Membrane receptor 51341 51341 Ki Ki Histamine H3 receptor 9.43179827593 8.54060751224 Q9Y5N1 Q9QYN8 451252 455.719 Membrane receptor 44314 44314 Ki Ki Neurotensin receptor 1 7.97469413474 7.55439579673 P30989 P20789 649986 817.05 Membrane receptor 51829 51829 IC50 IC50 Histamine H3 receptor 9.35654732351 8.79588001734 Q9Y5N1 Q9QYN8 632620 323.455 Membrane receptor 51341 51341 Ki Ki Peroxisome proliferator-activated receptor gamma 6.30050946667 6.53487707393 P37231 O88275 650045 414.564 Transcription Factor 51854,51854 51854,51854 IC50,IC50 IC50,IC50 Oxytocin receptor 8.30980391997 7.85387196432 P30559 P70536 108428 586.678 Membrane receptor 52842 52842 Ki Ki Vasopressin V2 receptor 4.55284196866 5.01322826573 P30518 Q00788 108428 586.678 Membrane receptor 52842 52842 Ki Ki Vasopressin V1a receptor 5.49485002168 9.11918640772 P37288 P30560 108428 586.678 Membrane receptor 52842 52842 Ki Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.95860731484 7.21467016499 P36544 Q05941 632725 306.362 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.82390874094 8.20065945055 P36544 Q05941 632727 306.365 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.26760624018 9.0 P36544 Q05941 632728 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 4.92081875395 7.76955107862 P36544 Q05941 632729 373.375 Ion channel 51372 51372 IC50 Ki Monoamine oxidase B 6.34678748622 7.00877392431 P27338 P19643 388574 302.343 Enzyme 37112 36690 Ki IC50 Monoamine oxidase A 3.43770713554 3.23657200644 P21397 P21396 388574 302.343 Enzyme 37112 36690 Ki IC50 Serotonin transporter 6.53461714855 6.49485002168 P31645 P31652 161345 281.821 Transporter 43754 43754 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.49485002168 7.30102999566 P36544 Q05941 632813 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.7447274949 8.50863830617 P36544 Q05941 632922 265.353 Ion channel 51372 51372 IC50 Ki Histamine H3 receptor 7.69897000434 6.58502665203 Q9Y5N1 Q9QYN8 438997 234.294 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.77212089845 7.92081875395 Q9Y5N1 Q9QYN8 453013 363.453 Membrane receptor 44908,47713 47713 IC50,Ki Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.79588001734 8.26760624018 P36544 Q05941 633072 304.389 Ion channel 51372 51372 IC50 Ki Serotonin 2a (5-HT2a) receptor 6.69897000434 6.76955107862 P28223 P14842 358744 312.202 Membrane receptor 31732 31732 Ki Ki Vasopressin V2 receptor 8.69897000434 8.08092190762 P30518 Q00788 128716 510.799 Membrane receptor 14475 14475 IC50 IC50 Vasopressin V1a receptor 6.19382002602 7.34678748622 P37288 P30560 128716 510.799 Membrane receptor 14475 14475 IC50 IC50 Vasopressin V2 receptor 6.30102999566 6.52287874528 P30518 Q00788 129399 427.538 Membrane receptor 17861 17861 IC50 IC50 Mu opioid receptor 6.64608376908 5.41907502432 P35372 P33535 391631 495.571 Membrane receptor 41961 36495 Ki IC50 Acetylcholinesterase 7.32790214206 6.94309514866 P22303 P37136 391755 242.316 Enzyme 21557,21519,30919,31257,31842,49254 3267,21462,36243,42156,42156 IC50,IC50,IC50,Ki,IC50,IC50 IC50,IC50,IC50,IC50,IC50 Vasopressin V2 receptor 9.0 8.34678748622 P30518 Q00788 129637 455.935 Membrane receptor 14475 14475 IC50 IC50 Vasopressin V1a receptor 7.22914798836 7.26760624018 P37288 P30560 129637 455.935 Membrane receptor 14475 14475 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.67778070527 7.58502665203 P36544 Q05941 632812 305.377 Ion channel 51372 51372 IC50 Ki Aldose reductase 6.82390874094 6.79588001734 P15121 P07943 130164 448.377 Enzyme 38948 41934 IC50 IC50 Mu opioid receptor 9.79783976639 10.2207657187 P35372 P33535 393379 638.756 Membrane receptor 42132,42132 36256,42132 Ki,IC50 Ki,Ki Dopamine D2 receptor 8.32790214206 7.3767507096 P14416 P61169 131346 419.491 Membrane receptor 30228 36547 Ki Ki Serotonin transporter 8.2924298239 8.69897000434 P31645 P31652 393960 394.55 Transporter 36227,36991,36991,37349 36227,37349 Ki,Ki,Ki,Ki Ki,Ki Serotonin transporter 8.18708664336 8.31875876262 P31645 P31652 393961 396.522 Transporter 36227,37349 36227,37349 Ki,Ki Ki,Ki Serotonin transporter 8.5376020021 8.78271554798 P31645 P31652 393962 412.54 Transporter 36227,37349,37349,37349 36227,37349,37349,37349 Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki Serotonin transporter 8.18708664336 8.24412514433 P31645 P31652 393963 430.531 Transporter 36227 36227 Ki Ki Serotonin transporter 8.08618614762 8.0 P31645 P31652 393964 430.531 Transporter 36227 36227 Ki Ki Serotonin transporter 8.42021640338 8.85387196432 P31645 P31652 393965 410.549 Transporter 36227 36227 Ki Ki Serotonin transporter 8.49485002168 8.69897000434 P31645 P31652 393966 424.576 Transporter 36227 36227 Ki Ki Serotonin transporter 8.2757241304 8.2757241304 P31645 P31652 393967 419.559 Transporter 36227 36227 Ki Ki Serotonin transporter 7.85387196432 7.72124639905 P31645 P31652 393968 462.548 Transporter 36227 36227 Ki Ki Serotonin transporter 7.92081875395 8.20065945055 P31645 P31652 393971 444.587 Transporter 36227 36227 Ki Ki Serotonin transporter 8.5376020021 8.69897000434 P31645 P31652 393974 402.477 Transporter 36227 36227 Ki Ki Serotonin transporter 8.13667713988 8.09691001301 P31645 P31652 393976 416.504 Transporter 36227 36227 Ki Ki Serotonin transporter 8.46852108296 9.13667713988 P31645 P31652 393977 354.486 Transporter 36227 36227 Ki Ki Serotonin transporter 8.39794000867 8.65757731918 P31645 P31652 393979 382.539 Transporter 36227 36227 Ki Ki Serotonin transporter 7.71444269099 8.52287874528 P31645 P31652 393982 366.496 Transporter 36227 36227 Ki Ki Serotonin transporter 8.01322826573 8.11918640772 P31645 P31652 393984 406.56 Transporter 36227 36227 Ki Ki Serotonin transporter 8.69897000434 8.82390874094 P31645 P31652 393986 423.591 Transporter 36227 36227 Ki Ki Serotonin transporter 8.7447274949 8.88605664769 P31645 P31652 393987 437.617 Transporter 36227 36227 Ki Ki Serotonin transporter 7.7447274949 8.0 P31645 P31652 393990 435.602 Transporter 36227 36227 Ki Ki Serotonin transporter 8.14266750357 8.24412514433 P31645 P31652 393992 487.633 Transporter 36227 36227 Ki Ki Serotonin transporter 8.09691001301 8.48148606012 P31645 P31652 393994 496.643 Transporter 36227 36227 Ki Ki Serotonin transporter 8.2757241304 8.56863623584 P31645 P31652 393998 478.649 Transporter 36227 36227 Ki Ki Serotonin transporter 8.39794000867 8.2757241304 P31645 P31652 394000 472.622 Transporter 36227 36227 Ki Ki Serotonin transporter 7.48148606012 7.60205999133 P31645 P31652 394002 539.632 Transporter 36227 36227 Ki Ki Serotonin transporter 7.3767507096 7.82390874094 P31645 P31652 394004 437.574 Transporter 36227 36227 Ki Ki Serotonin transporter 7.82390874094 7.82390874094 P31645 P31652 394006 465.628 Transporter 36227 36227 Ki Ki Serotonin transporter 8.05551732785 8.07572071394 P31645 P31652 394008 502.648 Transporter 36227 36227 Ki Ki Serotonin transporter 7.72124639905 7.67778070527 P31645 P31652 394010 500.632 Transporter 36227 36227 Ki Ki Nociceptin receptor 9.24074303006 8.51136689379 P41146 P35370 394466 1809.04 Membrane receptor 16753,16753,38383,38487,38487,43854,45320,45320,45630,45630 44658,44658 IC50,Ki,Ki,IC50,IC50,IC50,Ki,IC50,Ki,IC50 IC50,IC50 Nitric-oxide synthase, brain 5.88605664769 7.30102999566 P29475 P29476 394492 379.502 Enzyme 36390 36390 IC50 IC50 Nitric oxide synthase, inducible 4.88605664769 4.60205999133 P35228 Q06518 394492 379.502 Enzyme 36390 36390 IC50 IC50 Nitric-oxide synthase, brain 6.69897000434 6.09691001301 P29475 P29476 394493 387.522 Enzyme 36390 36390 IC50 IC50 Nitric oxide synthase, inducible 4.43179827593 4.35654732351 P35228 Q06518 394493 387.522 Enzyme 36390 36390 IC50 IC50 Nitric-oxide synthase, brain 6.30102999566 7.04575749056 P29475 P29476 394494 447.619 Enzyme 36390 36390 IC50 IC50 Nitric oxide synthase, inducible 4.85387196432 4.44369749923 P35228 Q06518 394494 447.619 Enzyme 36390 36390 IC50 IC50 Nitric-oxide synthase, brain 6.52287874528 5.31875876262 P29475 P29476 394496 451.611 Enzyme 36390 36390 IC50 IC50 Nitric oxide synthase, inducible 5.22184874962 4.58502665203 P35228 Q06518 394496 451.611 Enzyme 36390 36390 IC50 IC50 Nitric-oxide synthase, brain 5.35654732351 5.32790214206 P29475 P29476 394497 540.541 Enzyme 36390 36390 IC50 IC50 Nitric-oxide synthase, brain 7.0 5.1739251973 P29475 P29476 394499 477.645 Enzyme 36390 36390 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.02227639471 8.03151705145 P36544 Q05941 633821 266.341 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.56863623584 7.85387196432 P36544 Q05941 633822 306.362 Ion channel 51372 51372 IC50 Ki Cannabinoid CB2 receptor 7.0268721464 7.00877392431 P34972 Q9QZN9 590148 366.518 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 8.56863623584 7.88605664769 P34972 Q9QZN9 590180 366.518 Membrane receptor 49415 49415 Ki IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.76955107862 8.15490195999 P36544 Q05941 633899 305.377 Ion channel 51372 51372 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.39794000867 9.52287874528 P36544 Q05941 633900 319.404 Ion channel 51372 51372 IC50 Ki Anandamide amidohydrolase 8.73426054148 8.69897000434 O00519 P97612 396149 471.566 Enzyme 36571,49892 45059 IC50,IC50 Ki Bradykinin B1 receptor 9.35654732351 5.78972509323 P46663 P97583 396930 486.844 Membrane receptor 34832,36763,44560 34832,44560 Ki,Ki,Ki Ki,Ki Gonadotropin-releasing hormone receptor 8.82390874094 9.69897000434 P30968 P30969 397688 659.719 Membrane receptor 42049 36790,42049 IC50 Ki,IC50 Melanocortin receptor 3 6.12493873661 6.61978875829 P41968 P32244 398483 592.575 Membrane receptor 37011,37248 37011 Ki,Ki Ki Melanocortin receptor 4 8.35232642583 9.0 P32245 P70596 398483 592.575 Membrane receptor 37011,37011,37248,37248 37011 Ki,IC50,Ki,IC50 Ki Histamine H3 receptor 8.38299965888 7.189767482 Q9Y5N1 Q9QYN8 563225 353.46 Membrane receptor 47387 47387 Ki Ki Serotonin transporter 7.19382002602 8.65757731918 P31645 P31652 353736 382.471 Transporter 31450 31450 IC50 Ki Serotonin transporter 6.41341269533 8.04575749056 P31645 P31652 353737 396.498 Transporter 31450,44692 31450,36510,44692 IC50,IC50 Ki,Ki,Ki Serotonin transporter 9.15490195999 9.15490195999 P31645 P31652 399911 394.573 Transporter 36915 36915 Ki Ki Serotonin transporter 9.09691001301 9.04575749056 P31645 P31652 399913 396.546 Transporter 36915,38371 36915 Ki,Ki Ki Serotonin transporter 8.7447274949 8.61978875829 P31645 P31652 399916 419.344 Transporter 36915 36915 Ki Ki Serotonin transporter 8.72124639905 8.7447274949 P31645 P31652 399923 410.572 Transporter 36915 36915 Ki Ki Serotonin transporter 8.92081875395 8.95860731484 P31645 P31652 399924 384.899 Transporter 36915 36915 Ki Ki Serotonin transporter 7.52287874528 7.95860731484 P31645 P31652 399925 350.454 Transporter 36915 36915 Ki Ki Serotonin transporter 8.56863623584 8.69897000434 P31645 P31652 399926 418.452 Transporter 36915 36915 Ki Ki Serotonin transporter 7.76955107862 8.13667713988 P31645 P31652 399927 452.897 Transporter 36915 36915 Ki Ki Serotonin transporter 7.61978875829 8.0 P31645 P31652 399929 368.444 Transporter 36915 36915 Ki Ki Serotonin transporter 8.13667713988 8.52287874528 P31645 P31652 399932 384.899 Transporter 36915 36915 Ki Ki Serotonin transporter 8.44369749923 8.46852108296 P31645 P31652 399934 402.89 Transporter 36915 36915 Ki Ki Serotonin transporter 8.60205999133 9.04575749056 P31645 P31652 399936 412.611 Transporter 36915 36915 Ki Ki Serotonin transporter 8.1739251973 8.24412514433 P31645 P31652 399939 435.41 Transporter 36915 36915 Ki Ki Serotonin transporter 7.88605664769 9.30102999566 P31645 P31652 399940 437.641 Transporter 36915 36915 Ki Ki Serotonin transporter 9.04575749056 9.22184874962 P31645 P31652 399942 412.563 Transporter 36915 36915 Ki Ki Serotonin transporter 7.56863623584 8.67778070527 P31645 P31652 399944 435.362 Transporter 36915 36915 Ki Ki Serotonin transporter 8.45593195565 8.69897000434 P31645 P31652 399956 435.625 Transporter 36915 36915 Ki Ki Serotonin transporter 7.92081875395 9.52287874528 P31645 P31652 399959 366.52 Transporter 36915 36915 Ki Ki Serotonin transporter 8.85387196432 8.7447274949 P31645 P31652 399961 389.318 Transporter 36915 36915 Ki Ki Serotonin transporter 8.95860731484 8.88605664769 P31645 P31652 399962 380.546 Transporter 36915 36915 Ki Ki Serotonin transporter 8.22914798836 8.19382002602 P31645 P31652 399963 403.345 Transporter 36915 36915 Ki Ki Serotonin transporter 8.88605664769 9.39794000867 P31645 P31652 399964 409.544 Transporter 36915 36915 Ki Ki Serotonin transporter 8.92081875395 9.0 P31645 P31652 399965 451.624 Transporter 36915 36915 Ki Ki Serotonin transporter 8.44369749923 9.15490195999 P31645 P31652 399967 451.667 Transporter 36915 36915 Ki Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.02872415126 8.44369749923 P36544 Q05941 590953 357.452 Ion channel 49457 49457 IC50 Ki Histamine H3 receptor 9.09691001301 8.33 Q9Y5N1 Q9QYN8 400105 312.449 Membrane receptor 36915,48407,53407 48407 Ki,IC50,Ki IC50 Serotonin transporter 8.76955107862 9.30102999566 P31645 P31652 400115 338.263 Transporter 36915 36915 Ki Ki Serotonin transporter 8.46852108296 8.7447274949 P31645 P31652 400116 396.546 Transporter 36915 36915 Ki Ki Serotonin transporter 8.72124639905 9.04575749056 P31645 P31652 400117 416.643 Transporter 36915 36915 Ki Ki Serotonin transporter 8.85387196432 9.39794000867 P31645 P31652 400118 441.672 Transporter 36915 36915 Ki Ki Serotonin transporter 8.69897000434 9.22184874962 P31645 P31652 400119 439.656 Transporter 36915 36915 Ki Ki Cannabinoid CB1 receptor 6.39794000867 6.39794000867 P21554 P20272 400418 354.439 Membrane receptor 45100 37263 Ki Ki Neurokinin 1 receptor 8.82390874094 9.4397130344 P25103 P14600 400492 1347.63 Membrane receptor 44512 9460,11728 IC50 Ki,IC50 Melanocortin receptor 4 6.2924298239 8.04095860768 P32245 P70596 400646 565.07 Membrane receptor 36866 36866 IC50 Ki Vanilloid receptor 5.39794000867 8.56415516716 Q8NER1 O35433 591068 754.605 Ion channel 49452 38123,38123 IC50 Ki,Ki HMG-CoA reductase 7.95469464609 8.05562951966 P04035 P51639 138562 418.566 Enzyme 20826,20826,20826,20770 36875,42035 Ki,Ki,IC50,IC50 IC50,IC50 P2X purinoceptor 7 8.3 7.52287874528 Q99572 Q64663 400849 401.973 Ion channel 37197 37197 IC50 IC50 P2X purinoceptor 7 8.2 7.52287874528 Q99572 Q64663 400851 400.985 Ion channel 37197 37197 IC50 IC50 Monoamine oxidase A 3.44203588645 5.40893539297 P21397 P21396 139099 268.739 Enzyme 47084,44148,44874,46413,49935,50304,51147,52183,52782,52818,52882 45377,45377,44921,49220,49220,49443,49630 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,Ki,IC50,IC50,Ki,Ki,IC50 Urotensin II receptor 6.36653154442 5.60205999133 Q9UKP6 P49684 401314 576.726 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 6.85387196432 6.22184874962 Q9UKP6 P49684 401317 611.171 Membrane receptor 37148 37148 Ki IC50 Cannabinoid CB2 receptor 7.63827216398 7.95860731484 P34972 Q9QZN9 519648 380.502 Membrane receptor 46648,46648,49415 49415 Ki,IC50,Ki IC50 Urotensin II receptor 7.26760624018 6.39794000867 Q9UKP6 P49684 401349 645.188 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 6.79588001734 6.28399665637 Q9UKP6 P49684 401354 615.162 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 7.56863623584 6.48148606012 Q9UKP6 P49684 401358 609.198 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 7.52287874528 6.67778070527 Q9UKP6 P49684 401366 644.203 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 7.52287874528 7.2757241304 Q9UKP6 P49684 401368 665.242 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 7.11350927483 7.0 Q9UKP6 P49684 401383 625.198 Membrane receptor 37148 37148 Ki IC50 Urotensin II receptor 7.18708664336 8.0 Q9UKP6 P49684 401384 626.186 Membrane receptor 37148 37148 Ki IC50 Mu opioid receptor 8.59031030055 8.75701159064 P35372 P33535 139449 610.703 Membrane receptor 41961,42132,42132,48894 17669,17669,36256,36495,43813,43813,43813,46977,42132,47725 Ki,Ki,IC50,Ki Ki,Ki,Ki,IC50,Ki,Ki,IC50,IC50,Ki,Ki Serotonin transporter 7.59006687667 9.0 P31645 P31652 401982 396.566 Transporter 36991,36991,37541 37541 Ki,Ki,Ki Ki Serotonin transporter 6.97061622231 7.46852108296 P31645 P31652 401984 395.538 Transporter 36991,36991,37465 37465 Ki,Ki,Ki Ki Serotonin transporter 7.47500357154 7.93181413825 P31645 P31652 401985 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.74837711427 7.93181413825 P31645 P31652 401986 458.658 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 6.40364938333 6.39469495386 P31645 P31652 401987 458.658 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.23688206919 7.59006687667 P31645 P31652 401988 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 6.69042723683 6.73992861201 P31645 P31652 401989 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.52174770484 8.01322826573 P31645 P31652 401990 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 6.43663890427 6.75945075172 P31645 P31652 401991 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 8.04224731912 8.06048074738 P31645 P31652 401992 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 8.0320952731 8.36653154442 P31645 P31652 401993 458.658 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.8556518697 8.12493873661 P31645 P31652 401994 459.646 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.34369978037 7.95860731484 P31645 P31652 401996 461.619 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.5728469791 7.84466396253 P31645 P31652 401997 477.637 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 8.02528059948 8.28399665637 P31645 P31652 401998 465.674 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 7.2532361222 7.85387196432 P31645 P31652 401999 467.647 Transporter 36991,36991 36991 Ki,Ki Ki Serotonin transporter 8.08943983811 8.39794000867 P31645 P31652 402000 465.674 Transporter 36991,36991 36991 Ki,Ki Ki Metabotropic glutamate receptor 1 8.02227639471 8.10237290871 Q13255 P23385 402038 352.41 Membrane receptor 37138,50821 37138 IC50,IC50 Ki Metabotropic glutamate receptor 1 9.15490195999 7.77211329539 Q13255 P23385 402039 332.379 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 9.39794000867 8.61978875829 Q13255 P23385 402040 352.798 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.30980391997 7.54363396687 Q13255 P23385 402041 348.378 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.22184874962 7.96657624451 Q13255 P23385 402042 353.786 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.00877392431 6.98505965021 Q13255 P23385 402043 367.812 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 7.77469071827 7.74957999769 Q13255 P23385 402044 333.367 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 7.42481215507 7.70774392864 Q13255 P23385 402045 353.786 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 6.26680273489 6.0 Q13255 P23385 402047 382.482 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 6.19654288435 6.10347378251 Q13255 P23385 402049 396.509 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 6.35066514129 6.0 Q13255 P23385 402051 366.417 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.65757731918 9.30102999566 Q13255 P23385 402052 350.394 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.2757241304 9.22184874962 Q13255 P23385 402055 364.421 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.60205999133 9.0 Q13255 P23385 402057 366.394 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.61978875829 9.52287874528 Q13255 P23385 402058 380.42 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.5376020021 9.39794000867 Q13255 P23385 402059 370.813 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 7.61261017366 8.04095860768 Q13255 P23385 402061 384.839 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 7.92081875395 9.30102999566 Q13255 P23385 402064 384.839 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.65757731918 8.82390874094 Q13255 P23385 402065 384.839 Membrane receptor 37138 37138 IC50 Ki Metabotropic glutamate receptor 1 8.85387196432 9.69897000434 Q13255 P23385 402067 384.839 Membrane receptor 37138 37138 IC50 Ki Histamine H3 receptor 9.72124639905 9.22028610012 Q9Y5N1 Q9QYN8 403068 442.556 Membrane receptor 37121,37121,51341 37121,37121,37121,51341 Ki,IC50,Ki Ki,Ki,IC50,Ki Histamine H3 receptor 9.58502665203 8.74052599132 Q9Y5N1 Q9QYN8 403091 397.515 Membrane receptor 37121,37121,51341 37121,37121,37121,51341 Ki,IC50,Ki Ki,Ki,IC50,Ki Histamine H3 receptor 9.5376020021 8.9263164461 Q9Y5N1 Q9QYN8 403093 401.547 Membrane receptor 37121,37121,51341 37121,37121,37121,51341 Ki,IC50,Ki Ki,Ki,IC50,Ki Histamine H3 receptor 9.61978875829 9.03151705145 Q9Y5N1 Q9QYN8 403095 385.505 Membrane receptor 37121,37121,51341 37121,37121,37121,51341 Ki,IC50,Ki Ki,Ki,IC50,Ki Histamine H3 receptor 9.34678748622 8.65026325302 Q9Y5N1 Q9QYN8 403097 334.458 Membrane receptor 37121,37121,51341 37121,37121,37121,51341 Ki,IC50,Ki Ki,Ki,IC50,Ki Histamine H3 receptor 9.46852108296 8.57437082564 Q9Y5N1 Q9QYN8 403099 382.501 Membrane receptor 37121,37121,51341 37121,37121,37121,51341 Ki,IC50,Ki Ki,Ki,IC50,Ki Angiotensin II type 2 (AT-2) receptor 9.15490195999 9.15490195999 P50052 P35351 110876 611.735 Membrane receptor 30228 12035 IC50 IC50 HMG-CoA reductase 8.0 8.55284196866 P04035 P51639 403465 459.55 Enzyme 20770 36875,38124,42035 IC50 IC50,IC50,IC50 Adenosine A3 receptor 7.57835868874 5.84771165562 P33765 P28647 141567 477.55 Membrane receptor 13700,15057 15333 Ki,Ki Ki Adenosine A3 receptor 6.96259177968 5.38090666937 P33765 P28647 142047 417.497 Membrane receptor 13700,15057 13484 Ki,Ki Ki Acetylcholinesterase 7.08354605145 7.11069829749 P22303 P37136 404962 423.344 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 6.86838133565 6.87419354186 P22303 P37136 404963 329.394 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 6.63676419552 6.63115549317 P22303 P37136 404965 367.441 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 6.63544900465 6.66514431038 P22303 P37136 404966 342.432 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 6.54302698636 6.55222199071 P22303 P37136 404969 346.851 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 6.41623463172 6.44794046581 P22303 P37136 404970 670.844 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 7.15490195999 7.15490195999 P22303 P37136 404971 363.292 Enzyme 37075 37075 IC50 IC50 Plasminogen 4.88605664769 4.82390874094 P00747 Q01177 405410 468.442 Enzyme 37274 37274 IC50 IC50 Urokinase-type plasminogen activator 8.50863830617 7.70996538864 P00749 P29598 405410 468.442 Enzyme 37274 37274 IC50 IC50 Thrombin 5.94692155652 4.34678748622 P00734 P18292 405430 582.545 Enzyme 37274 37274 IC50 IC50 Plasminogen 5.55284196866 5.65757731918 P00747 Q01177 405430 582.545 Enzyme 37274 37274 IC50 IC50 Urokinase-type plasminogen activator 8.46852108296 7.61083391564 P00749 P29598 405430 582.545 Enzyme 37274 37274 IC50 IC50 Dopamine D2 receptor 8.55284196866 8.78919803657 P14416 P61169 155006 448.385 Membrane receptor 49693,49693,53091 45067,51830 Ki,Ki,Ki Ki,Ki Serotonin 2a (5-HT2a) receptor 8.39794000867 8.06048074738 P28223 P14842 155006 448.385 Membrane receptor 53091 45067,49687,51830 Ki Ki,Ki,Ki Serotonin 1a (5-HT1a) receptor 8.15490195999 8.25181197299 P08908 P19327 155006 448.385 Membrane receptor 53091 45067,49687,51830 Ki Ki,Ki,Ki Dopamine D2 receptor 6.02227639471 7.0 P14416 P61169 405786 219.326 Membrane receptor 21630,21630,21630,21630,30162,30162,30162,48491,48491 10581 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki IC50 Adenosine A2a receptor 5.53910215724 6.49485002168 P29274 P30543 406416 339.392 Membrane receptor 37033 37033 Ki Ki Adenosine A2a receptor 6.20065945055 6.63827216398 P29274 P30543 406418 355.391 Membrane receptor 37033 37033 Ki Ki Adenosine A2a receptor 5.34103515734 6.48148606012 P29274 P30543 406426 378.428 Membrane receptor 37033 37033 Ki Ki Adenosine A2a receptor 4.94692155652 6.15552282425 P29274 P30543 406704 355.391 Membrane receptor 37600 37600 Ki Ki Urotensin II receptor 6.86062319952 7.09691001301 Q9UKP6 P49684 580960 688.856 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Dopamine D2 receptor 6.58922276662 8.01322826573 P14416 P61169 146092 292.378 Membrane receptor 2789 2789 Ki Ki Dopamine D2 receptor 8.38721614328 9.2924298239 P14416 P61169 146093 360.376 Membrane receptor 2789 2789 Ki Ki Dopamine D2 receptor 6.26760624018 7.07160414774 P14416 P61169 146128 341.835 Membrane receptor 2789 2789 Ki Ki Serotonin transporter 7.49485002168 7.69897000434 P31645 P31652 408450 420.375 Transporter 37465 37465 Ki Ki Serotonin transporter 6.92081875395 7.82390874094 P31645 P31652 408451 434.402 Transporter 37465 37465 Ki Ki Serotonin transporter 6.85078088734 7.52287874528 P31645 P31652 408453 385.93 Transporter 37465 37465 Ki Ki Serotonin transporter 6.97469413474 7.65757731918 P31645 P31652 408455 399.957 Transporter 37465 37465 Ki Ki Serotonin transporter 5.87516985059 6.71219827007 P31645 P31652 408456 385.93 Transporter 37465 37465 Ki Ki Serotonin transporter 6.08301995268 6.8416375079 P31645 P31652 408457 399.957 Transporter 37465 37465 Ki Ki Urotensin II receptor 6.94336265377 7.79588001734 Q9UKP6 P49684 580989 598.733 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Serotonin transporter 6.83268266525 7.58502665203 P31645 P31652 408478 417.947 Transporter 37465 37465 Ki Ki Serotonin transporter 6.51999305704 7.22914798836 P31645 P31652 408481 395.538 Transporter 37465 37465 Ki Ki Serotonin transporter 6.83268266525 7.33724216832 P31645 P31652 408482 381.511 Transporter 37465 37465 Ki Ki Serotonin transporter 6.44129142947 6.73048705578 P31645 P31652 408491 383.502 Transporter 37465 37465 Ki Ki Serotonin transporter 5.94423953531 6.2448877336 P31645 P31652 408529 365.512 Transporter 37465 37465 Ki Ki Serotonin transporter 5.63208526121 5.77806440017 P31645 P31652 408530 351.485 Transporter 37465 37465 Ki Ki Serotonin transporter 6.11463877997 6.71896663275 P31645 P31652 408531 383.502 Transporter 37465 37465 Ki Ki Serotonin transporter 7.58502665203 7.82390874094 P31645 P31652 408532 408.365 Transporter 37465 37465 Ki Ki Serotonin transporter 6.64589156085 6.8894102897 P31645 P31652 408534 369.5 Transporter 37465 37465 Ki Ki Serotonin transporter 7.18045606446 7.72124639905 P31645 P31652 408535 383.527 Transporter 37465 37465 Ki Ki Serotonin transporter 5.69897000434 6.23433144524 P31645 P31652 408536 353.501 Transporter 37465 37465 Ki Ki Serotonin transporter 6.72353819583 7.2757241304 P31645 P31652 408537 383.484 Transporter 37465 37465 Ki Ki Serotonin transporter 7.15490195999 7.5376020021 P31645 P31652 408539 397.511 Transporter 37465 37465 Ki Ki Serotonin transporter 5.32175484807 5.69897000434 P31645 P31652 408540 353.458 Transporter 37465 37465 Ki Ki Serotonin transporter 7.43179827593 7.7447274949 P31645 P31652 408541 434.402 Transporter 37465 37465 Ki Ki Serotonin transporter 7.50863830617 7.63827216398 P31645 P31652 408542 448.428 Transporter 37465 37465 Ki Ki Serotonin transporter 7.03151705145 7.82390874094 P31645 P31652 408543 395.538 Transporter 37465 37465 Ki Ki Serotonin transporter 7.2076083105 7.34678748622 P31645 P31652 408544 409.564 Transporter 37465 37465 Ki Ki Vanilloid receptor 7.21843751983 6.28399665637 Q8NER1 O35433 408740 376.9 Ion channel 38185,38185,38185,38185 17091,37301,37301,38123,38123,38185,38185 IC50,IC50,IC50,IC50 Ki,Ki,Ki,Ki,Ki,IC50,IC50 Dopamine D2 receptor 8.09691001301 9.25181197299 P14416 P61169 146597 307.39 Membrane receptor 2789 2789 Ki Ki Dopamine D2 receptor 7.2757241304 8.49485002168 P14416 P61169 146649 291.39 Membrane receptor 2789 2789 Ki Ki Dopamine D2 receptor 7.08990945441 8.04095860768 P14416 P61169 146684 325.835 Membrane receptor 2789 2789 Ki Ki Dipeptidyl peptidase IV 6.89619627904 6.91721462968 P27487 P14740 409524 255.38 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.32239304728 7.12842706445 P27487 P14740 409525 269.406 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.85698519975 7.72353819583 P27487 P14740 409526 271.379 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.24033215531 7.09097914579 P27487 P14740 409527 284.421 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.96257350206 7.75448733219 P27487 P14740 409528 346.49 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.51570016065 7.41680122603 P27487 P14740 409529 360.517 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.67778070527 7.50307035193 P27487 P14740 409530 436.613 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.8696662315 7.77211329539 P27487 P14740 409531 376.516 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.91364016933 7.75696195131 P27487 P14740 409532 364.481 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.06048074738 7.98716277529 P27487 P14740 409533 380.935 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.38721614328 8.14266750357 P27487 P14740 409534 380.935 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 7.96657624451 7.96257350206 P27487 P14740 409535 380.935 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.08618614762 8.04575749056 P27487 P14740 409536 425.386 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.79588001734 8.65757731918 P27487 P14740 409537 391.488 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.36653154442 8.32790214206 P27487 P14740 409539 371.5 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.16749108729 8.14266750357 P27487 P14740 409540 414.488 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.52287874528 8.3767507096 P27487 P14740 409541 415.38 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.88605664769 8.7447274949 P27487 P14740 409542 396.509 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.25181197299 8.01772876696 P27487 P14740 409543 345.502 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.63827216398 8.48148606012 P27487 P14740 409544 390.5 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.61978875829 8.5376020021 P27487 P14740 409545 405.514 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.56863623584 8.45593195565 P27487 P14740 409546 347.478 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.50863830617 8.40893539297 P27487 P14740 409547 347.478 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.60205999133 8.50863830617 P27487 P14740 409548 381.923 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.79588001734 8.72124639905 P27487 P14740 409550 372.488 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 9.03621217265 8.95860731484 P27487 P14740 409551 392.476 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.82390874094 8.7447274949 P27487 P14740 409553 415.476 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 9.0 8.85387196432 P27487 P14740 409557 372.488 Enzyme 37469 37469 IC50 IC50 Dipeptidyl peptidase IV 8.92081875395 8.92081875395 P27487 P14740 409558 372.488 Enzyme 37469 37469 IC50 IC50 Vasopressin V1b receptor 6.68193666504 6.05848856737 P47901 P48974 678354 619.836 Membrane receptor 48483 48483 Ki Ki Vasopressin V1a receptor 5.94730605808 5.42969061456 P37288 P30560 678354 619.836 Membrane receptor 48483 48483 Ki Ki Adenosine A2a receptor 8.62981865525 8.60205999133 P29274 P30543 410123 503.556 Membrane receptor 37410,52381 37410 Ki,Ki Ki Serotonin transporter 7.85387196432 8.0 P31645 P31652 410264 464.564 Transporter 37541 37541 Ki Ki Serotonin transporter 6.70114692359 7.79588001734 P31645 P31652 410265 396.566 Transporter 37541 37541 Ki Ki Serotonin transporter 6.55129368009 7.7447274949 P31645 P31652 410266 396.566 Transporter 37541 37541 Ki Ki Serotonin transporter 5.82973828461 7.18708664336 P31645 P31652 410267 396.566 Transporter 37541 37541 Ki Ki Serotonin transporter 6.77211329539 7.40893539297 P31645 P31652 410268 396.566 Transporter 37541 37541 Ki Ki Serotonin transporter 7.3767507096 7.35654732351 P31645 P31652 410269 477.562 Transporter 37541 37541 Ki Ki Serotonin transporter 6.61083391564 7.20065945055 P31645 P31652 410270 409.564 Transporter 37541 37541 Ki Ki Serotonin transporter 7.21467016499 7.48148606012 P31645 P31652 410271 458.559 Transporter 37541 37541 Ki Ki Serotonin transporter 7.5376020021 8.22184874962 P31645 P31652 410272 390.561 Transporter 37541 37541 Ki Ki Serotonin transporter 8.0 8.88605664769 P31645 P31652 410273 442.657 Transporter 37541 37541 Ki Ki Serotonin transporter 7.79588001734 8.82390874094 P31645 P31652 410274 410.592 Transporter 37541 37541 Ki Ki Serotonin transporter 7.22184874962 8.69897000434 P31645 P31652 410275 426.592 Transporter 37541 37541 Ki Ki Serotonin transporter 7.95860731484 8.69897000434 P31645 P31652 410276 426.592 Transporter 37541 37541 Ki Ki Serotonin transporter 7.33724216832 8.88605664769 P31645 P31652 410277 414.556 Transporter 37541 37541 Ki Ki Serotonin transporter 7.79588001734 8.63827216398 P31645 P31652 410278 431.011 Transporter 37541 37541 Ki Ki Serotonin transporter 8.12320847055 8.40053406503 P31645 P31652 410279 431.011 Transporter 37541,37541 37541,37541 Ki,Ki Ki,Ki Serotonin transporter 8.20620063514 8.06336877028 P31645 P31652 410280 465.456 Transporter 37541,37541,37541,37541 37541,37541,37541,37541 Ki,Ki,Ki,Ki Ki,Ki,Ki,Ki Serotonin transporter 8.04575749056 8.30102999566 P31645 P31652 410281 475.462 Transporter 37541 37541 Ki Ki Serotonin transporter 8.39794000867 8.63827216398 P31645 P31652 410282 475.462 Transporter 37541 37541 Ki Ki Serotonin transporter 8.06048074738 8.43179827593 P31645 P31652 410283 441.563 Transporter 37541 37541 Ki Ki Serotonin transporter 6.79860287568 8.11350927483 P31645 P31652 410284 421.575 Transporter 37541 37541 Ki Ki Serotonin transporter 8.36653154442 8.36653154442 P31645 P31652 410285 412.54 Transporter 37349 37349 Ki Ki Serotonin transporter 8.32790214206 8.56863623584 P31645 P31652 410286 426.567 Transporter 37349 37349 Ki Ki Serotonin transporter 8.24412514433 8.2757241304 P31645 P31652 410287 446.985 Transporter 37349 37349 Ki Ki Serotonin transporter 7.95860731484 7.79588001734 P31645 P31652 410288 416.959 Transporter 37349 37349 Ki Ki Serotonin transporter 7.61978875829 7.85387196432 P31645 P31652 410289 416.959 Transporter 37349 37349 Ki Ki Serotonin transporter 7.7447274949 7.76955107862 P31645 P31652 410290 416.959 Transporter 37349 37349 Ki Ki Serotonin transporter 7.67778070527 8.08092190762 P31645 P31652 410291 451.404 Transporter 37349 37349 Ki Ki Serotonin transporter 6.97061622231 6.92081875395 P31645 P31652 410292 451.404 Transporter 37349 37349 Ki Ki Serotonin transporter 7.33724216832 7.88605664769 P31645 P31652 410293 382.514 Transporter 37349 37349 Ki Ki Serotonin transporter 8.06550154876 7.85387196432 P31645 P31652 410294 450.512 Transporter 37349 37349 Ki Ki Serotonin transporter 7.82390874094 7.52287874528 P31645 P31652 410295 450.512 Transporter 37349 37349 Ki Ki Serotonin transporter 8.3767507096 8.63827216398 P31645 P31652 410296 428.606 Transporter 37349,37349,37349 37349,37349,37349 Ki,Ki,Ki Ki,Ki,Ki Serotonin transporter 7.79588001734 8.10790539731 P31645 P31652 410297 407.524 Transporter 37349 37349 Ki Ki Serotonin transporter 7.88605664769 8.35654732351 P31645 P31652 410298 396.541 Transporter 37349 37349 Ki Ki Serotonin transporter 7.46852108296 7.44369749923 P31645 P31652 410299 482.577 Transporter 37349 37349 Ki Ki Serotonin transporter 6.8696662315 7.65757731918 P31645 P31652 410300 460.605 Transporter 37349 37349 Ki Ki Serotonin transporter 8.36653154442 8.52287874528 P31645 P31652 410301 448.521 Transporter 37349 37349 Ki Ki Serotonin transporter 8.28399665637 8.52287874528 P31645 P31652 410302 412.588 Transporter 37349,37349,37349 37349,37349,37349 Ki,Ki,Ki Ki,Ki,Ki Serotonin transporter 7.88605664769 8.22184874962 P31645 P31652 410303 410.549 Transporter 37349 37349 Ki Ki Serotonin transporter 7.88605664769 8.30102999566 P31645 P31652 410304 410.549 Transporter 37349 37349 Ki Ki Norepinephrine transporter 5.90483064857 6.28567024025 P23975 Q9WTR4 411284 274.333 Transporter 49772 37723 Ki Ki Dopamine transporter 6.29843201494 5.55439579673 Q01959 P23977 411284 274.333 Transporter 49772 37723 Ki Ki Serotonin transporter 8.09691001301 8.15428198203 P31645 P31652 411284 274.333 Transporter 49772 37723 Ki Ki Cannabinoid CB1 receptor 7.7447274949 7.09691001301 P21554 P20272 411703 421.533 Membrane receptor 37620 37620 Ki Ki Cannabinoid CB1 receptor 7.34678748622 7.45593195565 P21554 P20272 411711 403.517 Membrane receptor 37620 37620 Ki Ki Cannabinoid CB1 receptor 7.85387196432 7.52287874528 P21554 P20272 411772 444.354 Membrane receptor 37620 37620 Ki Ki Histamine H3 receptor 9.65757731918 8.70774392864 Q9Y5N1 Q9QYN8 411856 320.428 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.61978875829 8.60554831917 Q9Y5N1 Q9QYN8 411859 340.461 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.92081875395 8.45967052521 Q9Y5N1 Q9QYN8 411861 340.461 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.7447274949 8.90657831484 Q9Y5N1 Q9QYN8 411862 340.461 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.30980391997 8.19246497193 Q9Y5N1 Q9QYN8 411864 326.434 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.48017200622 7.17979854051 Q9Y5N1 Q9QYN8 411865 326.434 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.06499684855 7.47237009913 Q9Y5N1 Q9QYN8 411866 354.487 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 7.56383735296 6.63264407897 Q9Y5N1 Q9QYN8 411929 368.514 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 6.56383735296 6.33254704711 Q9Y5N1 Q9QYN8 411930 382.54 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.53910215724 7.36855623099 Q9Y5N1 Q9QYN8 411931 356.46 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.35654732351 7.95860731484 Q9Y5N1 Q9QYN8 411932 356.46 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.09151498112 8.01010543628 Q9Y5N1 Q9QYN8 411933 358.451 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 7.69680394258 7.0 Q9Y5N1 Q9QYN8 411935 369.502 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.80687540165 7.51004152058 Q9Y5N1 Q9QYN8 411937 342.434 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.05998184499 6.85078088734 Q9Y5N1 Q9QYN8 411938 354.487 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.57675412606 7.34390179799 Q9Y5N1 Q9QYN8 411960 300.397 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 9.07572071394 7.90308998699 Q9Y5N1 Q9QYN8 411961 328.45 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.67985371389 7.59006687667 Q9Y5N1 Q9QYN8 411962 328.45 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.96257350206 7.55439579673 Q9Y5N1 Q9QYN8 411965 342.477 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 8.33535802444 7.5185573715 Q9Y5N1 Q9QYN8 411972 342.477 Membrane receptor 37369 37369 Ki Ki Histamine H3 receptor 7.97881070093 6.34008379993 Q9Y5N1 Q9QYN8 411974 302.37 Membrane receptor 37369 37369 Ki Ki Serotonin transporter 7.91009488856 8.22184874962 P31645 P31652 412281 458.595 Transporter 37677 37677 Ki Ki Serotonin transporter 7.77728352885 8.1739251973 P31645 P31652 412283 458.595 Transporter 37677 37677 Ki Ki Serotonin transporter 7.18045606446 7.69897000434 P31645 P31652 412284 391.549 Transporter 37677 37677 Ki Ki Serotonin transporter 8.08092190762 8.69897000434 P31645 P31652 412300 391.549 Transporter 37677 37677 Ki Ki Serotonin transporter 7.91009488856 8.36653154442 P31645 P31652 412303 393.522 Transporter 37677 37677 Ki Ki Serotonin transporter 7.72815839346 8.48148606012 P31645 P31652 412304 391.549 Transporter 37677 37677 Ki Ki Serotonin transporter 7.50445566245 8.08092190762 P31645 P31652 412306 393.522 Transporter 37677 37677 Ki Ki Serotonin transporter 7.05551732785 7.64397414281 P31645 P31652 412308 394.51 Transporter 37677 37677 Ki Ki Serotonin transporter 8.56863623584 8.92081875395 P31645 P31652 412311 396.589 Transporter 37677 37677 Ki Ki Serotonin transporter 8.22184874962 8.52287874528 P31645 P31652 412313 398.561 Transporter 37677 37677 Ki Ki Lysophosphatidic acid receptor Edg-2 6.58502665203 7.09151498112 Q92633 P61794 412314 460.931 Membrane receptor 37582 37582 IC50 IC50 Serotonin transporter 8.88605664769 9.15490195999 P31645 P31652 412316 396.589 Transporter 37677 37677 Ki Ki Serotonin transporter 8.30102999566 8.69897000434 P31645 P31652 412319 398.561 Transporter 37677 37677 Ki Ki Serotonin transporter 7.70553377384 8.22184874962 P31645 P31652 412320 399.55 Transporter 37677 37677 Ki Ki Serotonin transporter 6.53610701101 7.27327279097 P31645 P31652 412321 399.55 Transporter 37677 37677 Ki Ki Serotonin transporter 6.91721462968 7.6143937264 P31645 P31652 412324 382.499 Transporter 37677 37677 Ki Ki Serotonin transporter 6.92445303861 7.40893539297 P31645 P31652 412325 432.558 Transporter 37677 37677 Ki Ki Lysophosphatidic acid receptor Edg-2 6.36653154442 7.13076828027 Q92633 P61794 412326 496.984 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.55284196866 6.95860731484 Q92633 P61794 412328 492.929 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.69897000434 7.14266750357 Q92633 P61794 412331 442.892 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.43179827593 6.92081875395 Q92633 P61794 412334 470.945 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.85387196432 7.13667713988 Q92633 P61794 412336 457.864 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.88605664769 7.0 Q92633 P61794 412339 460.931 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.76955107862 7.25181197299 Q92633 P61794 412340 464.962 Membrane receptor 37582 37582 IC50 IC50 Lysophosphatidic acid receptor Edg-2 6.88605664769 7.5376020021 Q92633 P61794 412363 450.936 Membrane receptor 37582 37582 IC50 IC50 Monoamine oxidase B 5.12262865413 5.12493873661 P27338 P19643 150743 179.219 Enzyme 47084,44148,44874,46413,48800,49935,50304,51147,52183,52379,52782,52818,52882 49630 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Monoamine oxidase A 5.18309616062 5.30102999566 P21397 P21396 150743 179.219 Enzyme 47084,44148,44874,46413,48800,49935,50304,51147,52183,52379,52782,52818,52882 49630 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Histamine H3 receptor 7.38721614328 6.43179827593 Q9Y5N1 Q9QYN8 438654 205.296 Membrane receptor 38490 38490 Ki Ki Cathepsin S 7.97930365742 5.97839728397 P25774 Q02765 413415 468.289 Enzyme 37689,42511 37689 IC50,IC50 IC50 Cathepsin L 6.3680518347 5.89346914618 P07711 P07154 413415 468.289 Enzyme 37689,42511 37689 IC50,IC50 IC50 Cathepsin B 6.55129643017 7.18045606446 P07858 P00787 413415 468.289 Enzyme 37689,42511 37689 IC50,IC50 IC50 Cathepsin S 8.7447274949 6.3705904009 P25774 Q02765 413426 407.383 Enzyme 37689 37689 IC50 IC50 Cathepsin L 5.99439055464 5.50045037409 P07711 P07154 413426 407.383 Enzyme 37689 37689 IC50 IC50 Cathepsin B 5.95703092661 6.49620931694 P07858 P00787 413426 407.383 Enzyme 37689 37689 IC50 IC50 Cathepsin S 9.30102999566 6.1197582241 P25774 Q02765 413441 447.447 Enzyme 37689 37689 IC50 IC50 Cathepsin L 6.72584215074 6.13194363818 P07711 P07154 413441 447.447 Enzyme 37689 37689 IC50 IC50 Cathepsin B 6.0 6.56543109597 P07858 P00787 413441 447.447 Enzyme 37689 37689 IC50 IC50 Cathepsin S 9.52287874528 7.67778070527 P25774 Q02765 413449 519.46 Enzyme 37689 37689 IC50 IC50 Cathepsin L 6.91721462968 6.39902710431 P07711 P07154 413449 519.46 Enzyme 37689 37689 IC50 IC50 Cathepsin B 5.87975520445 6.41566877563 P07858 P00787 413449 519.46 Enzyme 37689 37689 IC50 IC50 Cathepsin S 9.52287874528 7.18045606446 P25774 Q02765 413472 530.358 Enzyme 37689 37689 IC50 IC50 Cathepsin L 7.82390874094 7.14266750357 P07711 P07154 413472 530.358 Enzyme 37689 37689 IC50 IC50 Cathepsin B 5.46180342165 5.74256143314 P07858 P00787 413472 530.358 Enzyme 37689 37689 IC50 IC50 Cathepsin S 9.69897000434 7.82390874094 P25774 Q02765 413480 520.352 Enzyme 37689 37689 IC50 IC50 Cathepsin L 7.61978875829 7.31875876262 P07711 P07154 413480 520.352 Enzyme 37689 37689 IC50 IC50 Cathepsin B 5.0702235672 5.24458253719 P07858 P00787 413480 520.352 Enzyme 37689 37689 IC50 IC50 Cathepsin S 9.69897000434 7.35654732351 P25774 Q02765 413650 530.358 Enzyme 37689 37689 IC50 IC50 Cathepsin L 7.63827216398 6.87942606879 P07711 P07154 413650 530.358 Enzyme 37689 37689 IC50 IC50 Cathepsin B 5.17855198098 5.32771737521 P07858 P00787 413650 530.358 Enzyme 37689 37689 IC50 IC50 Neuropeptide Y receptor type 5 8.88605664769 8.67778070527 Q15761 Q63634 593301 406.41 Membrane receptor 49253 49253 IC50 IC50 Metabotropic glutamate receptor 1 6.39040559077 6.39040559077 Q13255 P23385 374879 364.464 Membrane receptor 35368 44256 IC50 IC50 Metabotropic glutamate receptor 1 7.06048074738 7.06048074738 Q13255 P23385 374889 362.448 Membrane receptor 35368 44256 IC50 IC50 Neuropeptide Y receptor type 5 8.88605664769 8.32790214206 Q15761 Q63634 593389 388.419 Membrane receptor 49253 49253 IC50 IC50 Mu opioid receptor 6.32422165833 6.32422165833 P35372 P33535 415408 390.475 Membrane receptor 48048 37724 Ki Ki Delta opioid receptor 8.34678748622 8.34678748622 P41143 P33533 415408 390.475 Membrane receptor 48048 37724 Ki Ki Vasopressin V1b receptor 7.35654732351 7.67778070527 P47901 P48974 678077 619.836 Membrane receptor 48483 48483 Ki Ki Vasopressin V1a receptor 6.50307035193 5.71851211206 P37288 P30560 678077 619.836 Membrane receptor 48483 48483 Ki Ki Renin 9.41457589818 5.59345981957 P00797 P08424 154467 701.898 Enzyme 11967,11967 11967 IC50,IC50 IC50 Beta-3 adrenergic receptor 8.28399665637 8.18708664336 P13945 P26255 417069 518.604 Membrane receptor 37880 37880 IC50 IC50 HMG-CoA reductase 8.22184874962 8.2076083105 P04035 P51639 417180 558.64 Enzyme 20770 38124,38261,42035 IC50 IC50,IC50,IC50 Beta-3 adrenergic receptor 7.56863623584 7.58502665203 P13945 P26255 417415 341.427 Membrane receptor 37716 37716 IC50 IC50 Beta-3 adrenergic receptor 6.76955107862 7.88605664769 P13945 P26255 417417 355.454 Membrane receptor 37716 37716 IC50 IC50 Gonadotropin-releasing hormone receptor 6.61261017366 7.0 P30968 P30969 417851 656.88 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.25963731051 7.82390874094 P30968 P30969 417853 708.955 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.45593195565 8.09691001301 P30968 P30969 417862 680.902 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.10237290871 7.56863623584 P30968 P30969 417864 722.982 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.01772876696 7.19382002602 P30968 P30969 417866 596.825 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.25181197299 7.79588001734 P30968 P30969 417871 637.877 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.79048498546 6.95860731484 P30968 P30969 417874 631.871 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.75202673364 6.76447155309 P30968 P30969 417876 589.834 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.70996538864 7.13076828027 P30968 P30969 417877 615.872 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.30539480107 6.93554201077 P30968 P30969 417879 601.845 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.76955107862 6.99567862622 P30968 P30969 417881 629.855 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.15739076039 6.27654432796 P30968 P30969 417883 601.845 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.46218090493 6.9829666607 P30968 P30969 417884 672.923 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.48017200622 6.80966830183 P30968 P30969 417886 688.965 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.13076828027 7.25963731051 P30968 P30969 417888 646.929 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.74957999769 7.2924298239 P30968 P30969 417891 588.846 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.56066730617 7.0268721464 P30968 P30969 417903 645.898 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.87942606879 7.2924298239 P30968 P30969 417906 630.883 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.43062609038 6.96657624451 P30968 P30969 417909 630.84 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.63264407897 7.19382002602 P30968 P30969 417910 616.856 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.77211329539 7.52287874528 P30968 P30969 417912 630.883 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.76195389687 7.2076083105 P30968 P30969 417914 630.883 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.73518217699 7.11918640772 P30968 P30969 417916 644.909 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.05551732785 7.36653154442 P30968 P30969 417918 630.883 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 6.47108329972 6.93554201077 P30968 P30969 417920 646.882 Membrane receptor 37902 37902 IC50 IC50 Gonadotropin-releasing hormone receptor 7.48148606012 7.52287874528 P30968 P30969 417922 618.915 Membrane receptor 37902 37902 IC50 IC50 Vasopressin V2 receptor 7.37625886966 7.52287874528 P30518 Q00788 418049 548.989 Membrane receptor 37905,37905 37905 IC50,IC50 IC50 Vasopressin V1a receptor 7.86062319952 6.19382002602 P37288 P30560 418049 548.989 Membrane receptor 37905,37905 37905 IC50,IC50 IC50 HMG-CoA reductase 8.28431811792 8.50863830617 P04035 P51639 418845 481.538 Enzyme 20826,20826,20826,20770 36875,37752,38124,38261,42035 Ki,Ki,IC50,IC50 IC50,IC50,IC50,IC50,IC50 Adenosine A2a receptor 8.56863623584 7.58502665203 P29274 P30543 418969 367.405 Membrane receptor 38162,38554,45839 38162 Ki,Ki,Ki Ki Adenosine A2a receptor 9.04575749056 7.95860731484 P29274 P30543 418973 384.455 Membrane receptor 38162,38554,38554 38162 Ki,Ki,IC50 Ki Adenosine A2a receptor 8.69897000434 7.85387196432 P29274 P30543 418975 395.458 Membrane receptor 38162,38554 38162 Ki,Ki Ki Peripheral-type benzodiazepine receptor 8.34678748622 9.13667713988 B1AH88 P16257 419371 351.847 Membrane receptor 38121 38121 Ki Ki Peripheral-type benzodiazepine receptor 9.61618463402 10.1390633793 B1AH88 P16257 419372 394.413 Membrane receptor 38121 38121 Ki Ki Peripheral-type benzodiazepine receptor 8.85387196432 10.0096611452 B1AH88 P16257 419376 374.406 Membrane receptor 38121 38121 Ki Ki Peripheral-type benzodiazepine receptor 8.60730304674 9.16749108729 B1AH88 P16257 419377 347.384 Membrane receptor 38121 38121 Ki Ki Metabotropic glutamate receptor 5 6.76447155309 6.78271554798 P41594 P31424 419523 247.291 Membrane receptor 38151 38151,38151 IC50 Ki,IC50 Metabotropic glutamate receptor 5 5.94692155652 5.71449516385 P41594 P31424 419526 249.307 Membrane receptor 38151 38151,38151 IC50 Ki,IC50 Metabotropic glutamate receptor 5 5.96657624451 5.81725600755 P41594 P31424 419529 249.307 Membrane receptor 38151 38151,38151 IC50 Ki,IC50 Metabotropic glutamate receptor 5 6.00877392431 6.03585329388 P41594 P31424 419530 249.307 Membrane receptor 38151 38151,38151 IC50 Ki,IC50 Sodium channel protein type X alpha subunit 8.09691001301 6.85387196432 Q9Y5Y9 Q62968 420803 357.788 Ion channel 38154,38190,38620,38620,38620,53932 38620,38620,38620,53444,53932 IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50,IC50 Serotonin transporter 9.0 9.05060999336 P31645 P31652 421007 324.392 Transporter 48944,51064 52243 Ki,Ki Ki Metabotropic glutamate receptor 4 6.0 6.0 Q14833 P31423 683234 197.236 Membrane receptor 52028 52028 IC50 IC50 Dopamine transporter 5.21467016499 4.43179827593 Q01959 P23977 421102 246.348 Transporter 45878 45878 IC50 IC50 Serotonin transporter 5.91634133263 7.01020305208 P31645 P31652 421102 246.348 Transporter 30228,38698,38710,45878 45878,45878 IC50,IC50,IC50,IC50 IC50,IC50 Neurokinin 1 receptor 8.43179827593 6.25181197299 P25103 P14600 594525 1211.3 Membrane receptor 49287 49287 Ki Ki Neurokinin 1 receptor 10.0 7.52287874528 P25103 P14600 594527 1211.3 Membrane receptor 49287 49287 Ki Ki Neurokinin 1 receptor 9.60205999133 8.14874165128 P25103 P14600 594528 1211.3 Membrane receptor 49287 49287 Ki Ki Dihydrofolate reductase 5.43872823797 5.47204338804 P00374 Q920D2 594576 322.361 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Dihydrofolate reductase 5.51104678618 5.50796148305 P00374 Q920D2 594590 338.404 Enzyme 49279,49279 49279,49279 IC50,Ki IC50,Ki Oxytocin receptor 8.30989437914 8.56863623584 P30559 P70536 332497 598.07 Membrane receptor 30371,30371 30371 Ki,IC50 Ki Cytochrome P450 17A1 7.14266750357 6.65757731918 P05093 P11715 422175 349.509 Enzyme 38222,38400,44174,44186,47824,51866,52270 38400 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Cannabinoid CB1 receptor 8.33889035263 9.0 P21554 P20272 684598 731.08 Membrane receptor 51963,51963 51963 IC50,IC50 IC50 Serotonin transporter 6.75202673364 7.88605664769 P31645 P31652 160746 281.821 Transporter 43754 43754 IC50 IC50 Muscarinic acetylcholine receptor M1 7.93554201077 7.93554201077 P11229 P08482 161229 343.41 Membrane receptor 30380 6436,5453,31903 Ki Ki,Ki,Ki Norepinephrine transporter 6.07365755337 6.14416385918 P23975 Q9WTR4 161229 343.41 Transporter 30380 17584,6436,5453,31903 Ki Ki,Ki,Ki,Ki Serotonin transporter 5.48678239993 5.48678239993 P31645 P31652 161229 343.41 Transporter 30380 6436,5453,31903 Ki Ki,Ki,Ki Serotonin transporter 7.05551732785 6.72124639905 P31645 P31652 161346 277.402 Transporter 43754 43754 IC50 IC50 Serotonin transporter 6.27245874297 5.8416375079 P31645 P31652 161503 315.374 Transporter 43754 43754 IC50 IC50 Vanilloid receptor 8.25963731051 8.20065945055 Q8NER1 O35433 685996 436.313 Ion channel 52179 52179 IC50 IC50 Dipeptidyl peptidase IV 7.46852108296 7.46470587996 P27487 P14740 376477 316.421 Enzyme 35539 35539 IC50 IC50 Vanilloid receptor 8.07572071394 8.14874165128 Q8NER1 O35433 686118 436.313 Ion channel 52179 52179 IC50 IC50 Vanilloid receptor 7.34948500217 8.69045333469 Q8NER1 O35433 686255 479.338 Ion channel 52179,52179 52179,52179 IC50,IC50 IC50,IC50 Vanilloid receptor 7.15490195999 6.58502665203 Q8NER1 O35433 424232 369.353 Ion channel 38263 38263 IC50 IC50 Vanilloid receptor 7.63827216398 6.38721614328 Q8NER1 O35433 424234 418.409 Ion channel 38263 38263 IC50 IC50 Vanilloid receptor 7.85387196432 7.35654732351 Q8NER1 O35433 424235 405.367 Ion channel 38263 38263 IC50 IC50 Vanilloid receptor 6.61897000434 5.28399665637 Q8NER1 O35433 424344 392.372 Ion channel 38263,38263 38263 IC50,IC50 IC50 Vanilloid receptor 7.30102999566 6.97881070093 Q8NER1 O35433 424786 382.883 Ion channel 38185 38185 IC50 IC50 Vanilloid receptor 7.18708664336 7.39363992279 Q8NER1 O35433 424787 419.324 Ion channel 38185,38185,53995 38185,38185 IC50,IC50,IC50 IC50,IC50 Histamine H3 receptor 7.08092190762 7.12493873661 Q9Y5N1 Q9QYN8 424791 430.588 Membrane receptor 38362 38362 Ki Ki Histamine H3 receptor 7.44369749923 6.16115090926 Q9Y5N1 Q9QYN8 424792 399.531 Membrane receptor 38362 38362 Ki Ki Histamine H3 receptor 7.61978875829 7.25963731051 Q9Y5N1 Q9QYN8 424793 356.508 Membrane receptor 38362 38362 Ki Ki Histamine H3 receptor 8.18045606446 8.20065945055 Q9Y5N1 Q9QYN8 424794 370.535 Membrane receptor 38362 38362 Ki Ki Histamine H3 receptor 8.61978875829 8.06893431034 Q9Y5N1 Q9QYN8 424796 384.561 Membrane receptor 38362 38362,38362 Ki Ki,IC50 Histamine H3 receptor 9.42021640338 9.16115090926 Q9Y5N1 Q9QYN8 424802 356.508 Membrane receptor 38362 38362 Ki Ki Histamine H3 receptor 9.48148606012 8.73864750363 Q9Y5N1 Q9QYN8 424803 356.508 Membrane receptor 38362 38362,38362 Ki Ki,IC50 Histamine H3 receptor 8.88605664769 8.95860731484 Q9Y5N1 Q9QYN8 424804 356.508 Membrane receptor 38362 38362 Ki Ki Histamine H3 receptor 9.32790214206 9.11350927483 Q9Y5N1 Q9QYN8 424805 356.508 Membrane receptor 38362 38362 Ki Ki Cannabinoid CB2 receptor 7.39794000867 7.04575749056 P34972 Q9QZN9 595131 354.464 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 7.76955107862 7.42021640338 P34972 Q9QZN9 595138 368.491 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 8.95860731484 7.08618614762 P34972 Q9QZN9 595147 396.544 Membrane receptor 49415 49415 Ki IC50 Cannabinoid CB2 receptor 7.79588001734 7.18045606446 P34972 Q9QZN9 595157 394.528 Membrane receptor 49415 49415 Ki IC50 Acyl coenzyme A:cholesterol acyltransferase 1 6.31966448659 6.31966448659 P35610 O70536 163574 501.721 Enzyme 45920 48377 IC50 IC50 Serotonin transporter 6.85387196432 7.56863623584 P31645 P31652 425797 264.386 Transporter 38710 45878 IC50 IC50 Melanocortin receptor 4 8.10790539731 9.0 P32245 P70596 425857 592.135 Membrane receptor 38716 38716 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 8.04575749056 8.5376020021 P36544 Q05941 425914 271.314 Ion channel 39478 39478 Ki Ki Melanocortin receptor 4 8.53786035697 9.03529053714 P32245 P70596 425998 621.024 Membrane receptor 38716,38716 38716,38716 IC50,IC50 IC50,IC50 Melanocortin receptor 4 8.38022513958 9.04575749056 P32245 P70596 426040 576.573 Membrane receptor 38716,38716 38716 IC50,IC50 IC50 Melanocortin receptor 4 8.48148606012 9.30102999566 P32245 P70596 426127 593.027 Membrane receptor 38716 38716 IC50 IC50 Serotonin transporter 6.49485002168 8.07058107429 P31645 P31652 164035 246.348 Transporter 38698,38710 13719,14579 IC50,IC50 Ki,Ki Cholecystokinin A receptor 9.4923201223 9.51436207563 P32238 P30551 164064 1143.27 Membrane receptor 45320,45320 14240,16223 IC50,Ki Ki,IC50 Cholecystokinin B receptor 9.43179827593 9.38721614328 P32239 P30553 164064 1143.27 Membrane receptor 45320,45320,42742 16223,14240,15481 IC50,Ki,IC50 IC50,Ki,Ki Cannabinoid CB1 receptor 6.6143937264 6.50723961097 P21554 P20272 337184 486.156 Membrane receptor 30590 30590 Ki Ki Neurokinin 1 receptor 9.65757731918 9.7447274949 P25103 P14600 164637 484.437 Membrane receptor 13477 2360 IC50 IC50 Histamine H3 receptor 8.52287874528 7.92081875395 Q9Y5N1 Q9QYN8 689600 459.587 Membrane receptor 52388 52388 IC50 IC50 Histamine H3 receptor 8.79588001734 7.76955107862 Q9Y5N1 Q9QYN8 689601 480.626 Membrane receptor 52388 52388 IC50 IC50 Histamine H3 receptor 9.39794000867 9.39794000867 Q9Y5N1 Q9QYN8 689602 514.708 Membrane receptor 52388 52388 IC50 IC50 Histamine H3 receptor 8.79588001734 8.03621217265 Q9Y5N1 Q9QYN8 689679 469.585 Membrane receptor 52388 52388 IC50 IC50 Histamine H3 receptor 8.33724216832 7.76955107862 Q9Y5N1 Q9QYN8 689680 483.611 Membrane receptor 52388 52388 IC50 IC50 Norepinephrine transporter 8.09691001301 8.22184874962 P23975 Q9WTR4 427891 333.809 Transporter 39371 39371 Ki Ki Serotonin transporter 6.95860731484 7.22914798836 P31645 P31652 427891 333.809 Transporter 39371 39371 Ki Ki Vasopressin V1b receptor 6.92081875395 6.67778070527 P47901 P48974 690264 476.567 Membrane receptor 52500 52500 IC50 IC50 HM74 nicotinic acid GPCR 4.48148606012 6.28755918168 P49019 Q80Z39 690523 331.754 Membrane receptor 52507 52507,52507 IC50 IC50,IC50 Histamine H3 receptor 7.25671392474 8.48734706737 Q9Y5N1 Q9QYN8 429662 292.443 Membrane receptor 21227,31675,50228,51191 16985,3951 Ki,Ki,Ki,Ki Ki,Ki Fructose-1,6-bisphosphatase 5.22184874962 4.69897000434 P09467 P19112 581701 293.215 Enzyme 49142 49142 IC50 IC50 Neurokinin 2 receptor 9.30102999566 9.30102999566 P21452 P16610 115369 552.534 Membrane receptor 3941 610 Ki Ki Nitric-oxide synthase, brain 6.5376020021 7.30102999566 P29475 P29476 692730 358.453 Enzyme 53397 53397 Ki Ki Nitric-oxide synthase, brain 5.7447274949 6.65757731918 P29475 P29476 692731 358.453 Enzyme 53397 53397 Ki Ki Casein kinase I delta 6.52287874528 6.52287874528 P48730 Q06486 430613 398.414 Enzyme 48310 48784 IC50 IC50 Serotonin 2a (5-HT2a) receptor 5.82390874094 7.82390874094 P28223 P14842 596209 345.386 Membrane receptor 49402 49402 IC50 Ki Melanocortin receptor 4 8.63380312009 8.95860731484 P32245 P70596 683594 598.123 Membrane receptor 52008,52008 52008 IC50,IC50 IC50 Vitamin D receptor 7.82390874094 8.30102999566 P11473 P13053 431616 426.588 Transcription Factor 39177,39177,39177 39177 IC50,IC50,IC50 IC50 Vitamin D receptor 7.69897000434 8.30102999566 P11473 P13053 431674 426.588 Transcription Factor 39177,39177,39177 39177 IC50,IC50,IC50 IC50 Vitamin D receptor 7.60205999133 8.69897000434 P11473 P13053 431677 426.588 Transcription Factor 39177,39177,39177 39177,44545,44545 IC50,IC50,IC50 IC50,Ki,IC50 Vitamin D receptor 6.61092437481 7.69897000434 P11473 P13053 431797 426.588 Transcription Factor 39177,39177,39177,39177 39177,44545,44545 IC50,IC50,IC50,IC50 IC50,Ki,IC50 Vanilloid receptor 8.39794000867 8.04575749056 Q8NER1 O35433 169747 345.318 Ion channel 36045,36128,38159,38185,38185 38185 IC50,IC50,IC50,IC50,IC50 IC50 Cannabinoid CB1 receptor 6.08206121842 6.60554831917 P21554 P20272 433316 354.486 Membrane receptor 39110,45100,49092,49092 49092 Ki,IC50,Ki,IC50 IC50 Cannabinoid CB2 receptor 8.34689474592 8.79588001734 P34972 Q9QZN9 433316 354.486 Membrane receptor 39110,39110,45100,49092,49092,49092 49092 Ki,IC50,IC50,Ki,IC50,IC50 IC50 Cannabinoid CB2 receptor 8.6411647485 8.85387196432 P34972 Q9QZN9 433551 397.41 Membrane receptor 39045,39045 39045 IC50,IC50 IC50 Anandamide amidohydrolase 9.58502665203 9.69897000434 O00519 P97612 433849 302.327 Enzyme 38493,38830 38493,38493,38830 Ki,Ki Ki,IC50,Ki Serotonin transporter 8.82390874094 8.83564714422 P31645 P31652 172234 358.436 Transporter 30228 5272 Ki Ki Calcitonin gene-related peptide type 1 receptor 10.8114393726 8.19382002602 Q16602 Q63118 328730 869.645 Membrane receptor 30176,30176 30176 IC50,IC50 IC50 Vanilloid receptor 8.0 6.72124639905 Q8NER1 O35433 435919 387.355 Ion channel 38526 38526 IC50 IC50 Vanilloid receptor 8.5376020021 7.55284196866 Q8NER1 O35433 435922 421.8 Ion channel 38526 38526 IC50 IC50 Vanilloid receptor 8.95860731484 7.36653154442 Q8NER1 O35433 435971 403.373 Ion channel 38526 38526 IC50 IC50 Vanilloid receptor 8.85387196432 8.25181197299 Q8NER1 O35433 435973 419.827 Ion channel 38526 38526 IC50 IC50 Vanilloid receptor 8.95860731484 7.95860731484 Q8NER1 O35433 435974 419.827 Ion channel 38526 38526 IC50 IC50 Vanilloid receptor 8.67778070527 8.01772876696 Q8NER1 O35433 435976 464.278 Ion channel 38526 38526 IC50 IC50 Vanilloid receptor 9.2076083105 8.25963731051 Q8NER1 O35433 436021 385.382 Ion channel 38526,38526,38526 38526,38526,38526 IC50,IC50,IC50 IC50,IC50,IC50 Histamine H3 receptor 9.46852108296 9.02000258084 Q9Y5N1 Q9QYN8 424806 356.508 Membrane receptor 38362 38362,38362 Ki Ki,IC50 P2X purinoceptor 7 6.85387196432 6.95860731484 Q99572 Q64663 436956 471.981 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.2924298239 6.65757731918 Q99572 Q64663 436958 497.588 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.05551732785 6.42021640338 Q99572 Q64663 436959 437.536 Ion channel 38841 38841 IC50 IC50 Bradykinin B1 receptor 9.18045606446 8.6615435064 P46663 P97583 436999 490.811 Membrane receptor 38375,38375,45754 38375 Ki,IC50,Ki Ki P2X purinoceptor 7 7.23657200644 6.85387196432 Q99572 Q64663 437000 497.588 Ion channel 38841,38841,43867 38841,38841,43867 IC50,IC50,IC50 IC50,IC50,IC50 P2X purinoceptor 7 6.72124639905 6.3767507096 Q99572 Q64663 437045 477.598 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 6.65757731918 6.60205999133 Q99572 Q64663 437141 427.498 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 6.36653154442 5.34678748622 Q99572 Q64663 437147 477.598 Ion channel 38841 38841 IC50 IC50 Muscarinic acetylcholine receptor M1 5.49485002168 5.30102999566 P11229 P08482 437264 343.85 Membrane receptor 50646 38774,50646 IC50 IC50,IC50 P2X purinoceptor 7 7.22914798836 7.52287874528 Q99572 Q64663 437346 520.582 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.15490195999 7.02227639471 Q99572 Q64663 437349 525.641 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.24412514433 7.11918640772 Q99572 Q64663 437390 511.615 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.0268721464 6.5376020021 Q99572 Q64663 437394 483.562 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.0 6.67778070527 Q99572 Q64663 437443 476.572 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 5.82390874094 6.20065945055 Q99572 Q64663 437444 495.658 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 6.92081875395 7.85387196432 Q99572 Q64663 437448 437.535 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 6.0 4.85387196432 Q99572 Q64663 437492 427.502 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.39794000867 6.49485002168 Q99572 Q64663 437538 441.528 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.22184874962 6.25181197299 Q99572 Q64663 437540 441.528 Ion channel 38841 38841 IC50 IC50 Glycogen synthase kinase-3 beta 7.52287874528 5.49485002168 P49841 P18266 437567 443.478 Enzyme 38602 38602 IC50 IC50 P2X purinoceptor 7 6.95860731484 6.28399665637 Q99572 Q64663 437582 427.498 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.14874165128 6.56863623584 Q99572 Q64663 437584 443.564 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.33724216832 6.82390874094 Q99572 Q64663 437619 443.564 Ion channel 38841 38841 IC50 IC50 Muscarinic acetylcholine receptor M1 9.60205999133 9.10237290871 P11229 P08482 437621 289.369 Membrane receptor 16845 10799,38774,52040 Ki Ki,Ki,Ki Muscarinic acetylcholine receptor M3 9.17339374311 9.05731938998 P20309 P08483 437621 289.369 Membrane receptor 16845,52761 38774,52040 Ki,Ki Ki,Ki Muscarinic acetylcholine receptor M2 8.77257757 8.83863199777 P08172 P10980 437621 289.369 Membrane receptor 16845,52761 9794,9794,10799,38774,52040 Ki,Ki Ki,Ki,Ki,Ki,Ki Muscarinic acetylcholine receptor M5 9.26760624018 8.90511452183 P08912 P08911 437621 289.369 Membrane receptor 16845,46746,52761 38774,52040 Ki,Ki,Ki Ki,Ki Muscarinic acetylcholine receptor M4 8.99569991412 9.28399665637 P08173 P08485 437621 289.369 Membrane receptor 16845,52761 38774,52040,52040 Ki,Ki Ki,Ki,Ki P2X purinoceptor 7 6.38721614328 6.21467016499 Q99572 Q64663 437661 442.513 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.33724216832 6.76955107862 Q99572 Q64663 437665 442.513 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.44369749923 6.82390874094 Q99572 Q64663 437666 438.524 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.39794000867 6.40893539297 Q99572 Q64663 437667 438.524 Ion channel 38841 38841 IC50 IC50 P2X purinoceptor 7 7.19637974808 7.7447274949 Q99572 Q64663 437668 474.555 Ion channel 38841,48423,48423,48423 38841,48423 IC50,IC50,IC50,IC50 IC50,IC50 Serotonin transporter 8.04575749056 8.04095860768 P31645 P31652 437760 448.385 Transporter 38371 38371 Ki Ki Serotonin transporter 8.0 8.42021640338 P31645 P31652 437761 413.94 Transporter 38371 38371 Ki Ki Serotonin transporter 7.92081875395 8.02227639471 P31645 P31652 437804 439.613 Transporter 38371 38371 Ki Ki Serotonin transporter 8.5376020021 8.65757731918 P31645 P31652 437806 425.587 Transporter 38371 38371 Ki Ki Serotonin transporter 6.15366288787 6.52432881168 P31645 P31652 438077 463.493 Transporter 38371 38371 Ki Ki Serotonin transporter 7.02227639471 7.95860731484 P31645 P31652 438078 479.558 Transporter 38371 38371 Ki Ki Mu opioid receptor 6.93930215965 6.93930215965 P35372 P33535 509926 871.931 Membrane receptor 42132 42132 Ki Ki Serotonin transporter 7.0268721464 7.61978875829 P31645 P31652 438126 404.505 Transporter 38371 38371 Ki Ki Serotonin transporter 6.91364016933 7.88605664769 P31645 P31652 438129 404.505 Transporter 38371 38371 Ki Ki Serotonin transporter 7.38721614328 8.10237290871 P31645 P31652 438178 431.931 Transporter 38371 38371 Ki Ki Serotonin transporter 7.76955107862 7.95860731484 P31645 P31652 438179 447.493 Transporter 38371 38371 Ki Ki Serotonin transporter 7.44369749923 8.07058107429 P31645 P31652 438180 431.931 Transporter 38371 38371 Ki Ki Serotonin transporter 5.85387196432 6.04575749056 P31645 P31652 438184 447.493 Transporter 38371 38371 Ki Ki Serotonin transporter 7.16749108729 8.1739251973 P31645 P31652 438227 397.486 Transporter 38371 38371 Ki Ki Serotonin transporter 6.25026368443 6.93181413825 P31645 P31652 438232 397.486 Transporter 38371 38371 Ki Ki Serotonin transporter 7.32790214206 8.01322826573 P31645 P31652 438272 413.94 Transporter 38371 38371 Ki Ki Serotonin transporter 6.64016451766 7.43179827593 P31645 P31652 438273 379.495 Transporter 38371 38371 Ki Ki Serotonin transporter 7.88605664769 8.34678748622 P31645 P31652 438278 409.521 Transporter 38371 38371 Ki Ki Serotonin transporter 8.19382002602 8.85387196432 P31645 P31652 438320 415.956 Transporter 38371 38371 Ki Ki Serotonin transporter 6.93554201077 7.85387196432 P31645 P31652 438321 415.956 Transporter 38371 38371 Ki Ki Serotonin transporter 7.85387196432 8.72124639905 P31645 P31652 438358 450.401 Transporter 38371 38371 Ki Ki Serotonin transporter 8.30102999566 9.0 P31645 P31652 438363 427.603 Transporter 38371 38371 Ki Ki Serotonin transporter 8.09151498112 8.23657200644 P31645 P31652 438399 427.603 Transporter 38371 38371 Ki Ki Histamine H3 receptor 8.79588001734 8.22914798836 Q9Y5N1 Q9QYN8 438422 295.419 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.30102999566 7.39794000867 Q9Y5N1 Q9QYN8 438425 281.392 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.88605664769 8.14874165128 Q9Y5N1 Q9QYN8 438427 239.355 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.52287874528 6.49485002168 Q9Y5N1 Q9QYN8 438431 190.285 Membrane receptor 38490 38490 Ki Ki Dipeptidyl peptidase IV 7.6205440538 7.22184874962 P27487 P14740 438444 410.557 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 7.49676697888 7.16115090926 P27487 P14740 438445 392.519 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 7.3758907194 6.85387196432 P27487 P14740 438446 432.464 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 7.55063740921 7.11918640772 P27487 P14740 438448 396.531 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 8.30102999566 8.39794000867 P31645 P31652 438451 411.56 Transporter 38371 38371 Ki Ki Histamine H3 receptor 7.85387196432 7.05060999336 Q9Y5N1 Q9QYN8 438471 239.355 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.45593195565 7.2076083105 Q9Y5N1 Q9QYN8 438474 270.369 Membrane receptor 38490 38490 Ki Ki Dipeptidyl peptidase IV 7.05395269865 6.72124639905 P27487 P14740 438492 406.546 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 7.37164112701 6.95860731484 P27487 P14740 438495 406.546 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 6.44009337496 6.99139982824 P31645 P31652 438498 383.459 Transporter 38371 38371 Ki Ki Serotonin transporter 8.22914798836 8.7447274949 P31645 P31652 438503 413.576 Transporter 38371 38371 Ki Ki Histamine H3 receptor 7.55284196866 6.35654732351 Q9Y5N1 Q9QYN8 438523 270.369 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.58502665203 6.67778070527 Q9Y5N1 Q9QYN8 438525 256.343 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.82390874094 7.38721614328 Q9Y5N1 Q9QYN8 438527 258.359 Membrane receptor 38490 38490 Ki Ki Dipeptidyl peptidase IV 7.23400522429 6.92081875395 P27487 P14740 438530 392.519 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 6.05250985454 6.01772876696 P27487 P14740 438541 362.427 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 7.47890920274 7.34678748622 P27487 P14740 438542 364.466 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 6.27164621798 6.73048705578 P31645 P31652 438543 365.469 Transporter 38371 38371 Ki Ki Serotonin 5a (5-HT5a) receptor 8.16749108729 8.5376020021 P47898 P35364 438544 259.683 Membrane receptor 38456 38456 Ki Ki Dipeptidyl peptidase IV 6.5468324791 6.46852108296 P27487 P14740 438545 377.504 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 6.80966830183 6.94692155652 P31645 P31652 438546 399.914 Transporter 38371 38371 Ki Ki Dipeptidyl peptidase IV 6.05423127116 6.2924298239 P27487 P14740 438582 391.531 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 6.91946580726 6.61978875829 P27487 P14740 438584 377.504 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 6.2135641989 6.49485002168 P27487 P14740 438585 377.504 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin 5a (5-HT5a) receptor 8.79588001734 8.88605664769 P47898 P35364 438586 195.649 Membrane receptor 38456 38456 Ki Ki Histamine H3 receptor 8.05060999336 7.20065945055 Q9Y5N1 Q9QYN8 438611 219.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.63827216398 7.92081875395 Q9Y5N1 Q9QYN8 438612 219.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.7447274949 6.46852108296 Q9Y5N1 Q9QYN8 438614 228.333 Membrane receptor 38490 38490 Ki Ki Adenosine A1 receptor 7.2410881076 7.65560772631 P30542 P25099 597391 398.477 Membrane receptor 49741 49741,49741,49741 Ki Ki,IC50,IC50 Histamine H3 receptor 7.18708664336 6.76955107862 Q9Y5N1 Q9QYN8 438652 219.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.50863830617 6.61978875829 Q9Y5N1 Q9QYN8 438656 219.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.45593195565 6.95860731484 Q9Y5N1 Q9QYN8 438657 219.323 Membrane receptor 38490 38490 Ki Ki Dipeptidyl peptidase IV 7.05395269865 7.21467016499 P27487 P14740 438670 377.504 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 7.61978875829 8.09151498112 P31645 P31652 438674 427.967 Transporter 38371 38371 Ki Ki Histamine H3 receptor 7.56863623584 6.48148606012 Q9Y5N1 Q9QYN8 438698 203.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.30102999566 7.43179827593 Q9Y5N1 Q9QYN8 438699 203.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.46852108296 6.58502665203 Q9Y5N1 Q9QYN8 438701 205.296 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.49485002168 6.61978875829 Q9Y5N1 Q9QYN8 438703 203.323 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.30102999566 7.52287874528 Q9Y5N1 Q9QYN8 438704 203.323 Membrane receptor 38490 38490 Ki Ki Dipeptidyl peptidase IV 6.26093328595 6.11918640772 P27487 P14740 438720 392.519 Enzyme 38801,38801 38801 IC50,IC50 IC50 Dipeptidyl peptidase IV 6.23458011069 6.34678748622 P27487 P14740 438721 377.504 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 7.40893539297 8.0 P31645 P31652 438723 413.94 Transporter 38371 38371 Ki Ki Serotonin transporter 7.63827216398 8.01322826573 P31645 P31652 438777 399.914 Transporter 38371 38371 Ki Ki Serotonin transporter 7.61978875829 8.08618614762 P31645 P31652 438783 401.93 Transporter 38371 38371 Ki Ki Dipeptidyl peptidase IV 7.03786035697 6.82390874094 P27487 P14740 438826 440.562 Enzyme 38801,38801 38801 IC50,IC50 IC50 Serotonin transporter 7.82390874094 7.95860731484 P31645 P31652 438830 462.412 Transporter 38371 38371 Ki Ki Cytochrome P450 17A1 6.42829116819 6.25026368443 P05093 P11715 438863 268.377 Enzyme 38400 38400 IC50 IC50 Cytochrome P450 17A1 6.02090709936 6.17005330406 P05093 P11715 438864 254.35 Enzyme 38400 38400 IC50 IC50 Serotonin transporter 7.79588001734 7.92081875395 P31645 P31652 438877 448.385 Transporter 38371 38371 Ki Ki Serotonin transporter 8.16749108729 8.03151705145 P31645 P31652 438879 434.359 Transporter 38371 38371 Ki Ki Serotonin transporter 8.20065945055 8.30980391997 P31645 P31652 438924 436.375 Transporter 38371 38371 Ki Ki Histamine H3 receptor 7.67778070527 6.61978875829 Q9Y5N1 Q9QYN8 438950 205.296 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.39794000867 6.63827216398 Q9Y5N1 Q9QYN8 438951 217.35 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.01772876696 6.65757731918 Q9Y5N1 Q9QYN8 438952 205.296 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.01772876696 6.55284196866 Q9Y5N1 Q9QYN8 438990 234.294 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.56863623584 6.46852108296 Q9Y5N1 Q9QYN8 438991 191.269 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.36653154442 6.63827216398 Q9Y5N1 Q9QYN8 439043 232.364 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 8.22184874962 7.36653154442 Q9Y5N1 Q9QYN8 439044 232.364 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.95860731484 6.46852108296 Q9Y5N1 Q9QYN8 439048 195.324 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.46852108296 6.85387196432 Q9Y5N1 Q9QYN8 439049 195.324 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.76955107862 7.09151498112 Q9Y5N1 Q9QYN8 439084 196.312 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.48148606012 6.79588001734 Q9Y5N1 Q9QYN8 439086 196.312 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.46852108296 6.82390874094 Q9Y5N1 Q9QYN8 439088 218.338 Membrane receptor 38490 38490 Ki Ki Serotonin transporter 7.95860731484 8.3767507096 P31645 P31652 439103 425.587 Transporter 38371 38371 Ki Ki Histamine H3 receptor 9.40893539297 8.40893539297 Q9Y5N1 Q9QYN8 439134 295.419 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.63827216398 6.79588001734 Q9Y5N1 Q9QYN8 439135 204.311 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 7.15490195999 6.49485002168 Q9Y5N1 Q9QYN8 439139 190.285 Membrane receptor 38490 38490 Ki Ki Histamine H3 receptor 6.45593195565 6.49485002168 Q9Y5N1 Q9QYN8 439140 176.258 Membrane receptor 38490 38490 Ki Ki C-X-C chemokine receptor type 4 8.61798295743 8.36653154442 P61073 O08565 701437 420.55 Membrane receptor 52638,52638,52638,52638,52638,52638,52638 52638 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Niemann-Pick C1-like protein 1 6.52287874528 6.49064975067 Q9UHC9 Q6T3U3 177304 585.549 Membrane other 46716,46716 38403,46716 IC50,IC50 Ki,IC50 Adenosine A2a receptor 7.82390874094 5.79588001734 P29274 P30543 439973 424.496 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.26760624018 6.98716277529 P29274 P30543 439974 408.497 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.22184874962 6.63827216398 P29274 P30543 439975 410.47 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.24412514433 6.36653154442 P29274 P30543 440012 396.443 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.44369749923 6.76955107862 P29274 P30543 440014 437.495 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.0 7.33068311943 P29274 P30543 440058 423.511 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.0 7.06048074738 P29274 P30543 440059 451.565 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 7.95860731484 6.56863623584 P29274 P30543 440061 423.511 Membrane receptor 38555 38555 Ki Ki Neurokinin 1 receptor 10.3372421683 8.79588001734 P25103 P14600 440088 1079.09 Membrane receptor 38754 38754 Ki Ki Neurokinin 1 receptor 7.0 6.56863623584 P25103 P14600 440089 943.097 Membrane receptor 38754 38754 Ki Ki Adenosine A2a receptor 7.92081875395 6.88173527391 P29274 P30543 440098 409.485 Membrane receptor 38554,38555,45867 38555 Ki,Ki,Ki Ki Adenosine A2a receptor 8.67778070527 7.36653154442 P29274 P30543 440430 368.433 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.67778070527 7.55595520408 P29274 P30543 440434 437.538 Membrane receptor 38555 38555 Ki Ki Adenosine A2a receptor 8.35654732351 6.80966830183 P29274 P30543 440436 451.565 Membrane receptor 38555 38555 Ki Ki Neurokinin 1 receptor 8.85387196432 8.21467016499 P25103 P14600 440468 1092.13 Membrane receptor 38754 38754 Ki Ki Adenosine A2a receptor 8.60205999133 7.43179827593 P29274 P30543 440472 423.511 Membrane receptor 38555 38555 Ki Ki Neurokinin 1 receptor 9.21467016499 7.48148606012 P25103 P14600 440507 1078.11 Membrane receptor 38754 38754 Ki Ki Adenosine A3 receptor 5.61798295743 5.72124639905 P33765 P28647 178365 453.529 Membrane receptor 14546 14546 Ki Ki Adenosine A2a receptor 8.43179827593 6.79588001734 P29274 P30543 440547 423.511 Membrane receptor 38555 38555 Ki Ki Cannabinoid CB1 receptor 7.92081875395 7.92081875395 P21554 P20272 440704 339.471 Membrane receptor 39110,49092,49092 49092 Ki,Ki,IC50 IC50 Cannabinoid CB2 receptor 8.56863623584 9.76955107862 P34972 Q9QZN9 440704 339.471 Membrane receptor 39110,39110,49092,49092,49092 49092 Ki,IC50,Ki,IC50,IC50 IC50 Bradykinin B1 receptor 8.9751971937 8.79452707066 P46663 P97583 702951 601.741 Membrane receptor 52840,52840 52840,52840 Ki,IC50 IC50,Ki Oxytocin receptor 9.30102999566 8.63294000867 P30559 P70536 702953 604.523 Membrane receptor 52842 52842,52842 Ki Ki,IC50 Vasopressin V1a receptor 6.84466396253 7.0043648054 P37288 P30560 702953 604.523 Membrane receptor 52842 52842 Ki Ki Dopamine D2 receptor 6.96657624451 7.21485698846 P14416 P61169 703227 469.661 Membrane receptor 52843 52843,52843 IC50 Ki,Ki Dopamine D3 receptor 8.98716277529 8.41836264686 P35462 P19020 703227 469.661 Membrane receptor 52843 52843,52843 IC50 Ki,Ki Adenosine A1 receptor 9.53017798402 9.72124639905 P30542 P25099 597804 328.409 Membrane receptor 49741 49741 Ki Ki Oxytocin receptor 7.88605664769 8.44369749923 P30559 P70536 703311 554.766 Membrane receptor 52842 52842 Ki Ki Vasopressin V2 receptor 6.22914798836 6.69897000434 P30518 Q00788 703311 554.766 Membrane receptor 52842 52842 Ki Ki Vasopressin V1a receptor 6.7447274949 6.95860731484 P37288 P30560 703311 554.766 Membrane receptor 52842 52842 Ki Ki Oxytocin receptor 7.02227639471 6.67778070527 P30559 P70536 703484 338.4 Membrane receptor 52842 52842 Ki Ki Oxytocin receptor 7.85387196432 9.1739251973 P30559 P70536 703577 492.547 Membrane receptor 52842 52842 Ki Ki Sodium/glucose cotransporter 2 8.95860731484 8.52287874528 P31639 P53792 441579 408.873 Transporter 38587,46153,48692,49070,49735,50501,51306,51619,52206,54007 38587,46153 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50 Corticotropin releasing factor receptor 1 8.07058107429 8.16749108729 P34998 P35353 441706 327.46 Membrane receptor 38734 38419,38734,38734 Ki IC50,IC50,Ki Anandamide amidohydrolase 9.1739251973 9.09691001301 O00519 P97612 441958 375.341 Enzyme 38493 38493 Ki Ki Anandamide amidohydrolase 8.92081875395 8.92081875395 O00519 P97612 441959 412.437 Enzyme 38493 38493 Ki Ki Anandamide amidohydrolase 9.07058107429 8.69897000434 O00519 P97612 442081 318.326 Enzyme 38493 38493,38493 Ki Ki,IC50 Anandamide amidohydrolase 9.0 8.69897000434 O00519 P97612 442110 361.315 Enzyme 38493 38493 Ki Ki Dopamine D2 receptor 7.27901425585 7.27083521031 P14416 P61169 704416 469.661 Membrane receptor 52843 52843 IC50 Ki Dopamine D3 receptor 9.60205999133 8.62708799703 P35462 P19020 704416 469.661 Membrane receptor 52843 52843 IC50 Ki Adenosine A1 receptor 8.04575749056 8.92081875395 P30542 P25099 442361 428.485 Membrane receptor 38739,42591,47890 11627,8687,16896,11292 Ki,Ki,Ki Ki,Ki,Ki,Ki Adenosine A2a receptor 7.80687540165 7.20065945055 P29274 P30543 442361 428.485 Membrane receptor 14051,14051,14051 16896,16318 Ki,Ki,Ki Ki,Ki Anandamide amidohydrolase 9.2924298239 9.0 O00519 P97612 442377 332.353 Enzyme 38493 38493,38493 Ki Ki,IC50 Alpha-1a adrenergic receptor 8.04575749056 5.4 P35348 P43140 180673 265.331 Membrane receptor 39519 42637 IC50 IC50 Serotonin transporter 6.91009488856 6.7447274949 P31645 P31652 161309 281.821 Transporter 43754 43754 IC50 IC50 Metabotropic glutamate receptor 5 7.55284196866 7.76955107862 P41594 P31424 706271 320.32 Membrane receptor 53102 53102 IC50 Ki Metabotropic glutamate receptor 5 7.79588001734 7.76955107862 P41594 P31424 706506 334.347 Membrane receptor 53102 53102 IC50 Ki Angiotensin-converting enzyme 9.20065945055 7.48940535047 P12821 P47820 444750 217.285 Enzyme 30228,43854,48262 8407,8407 IC50,IC50,IC50 IC50,IC50 Histamine H3 receptor 8.02287874528 7.83277312442 Q9Y5N1 Q9QYN8 706970 395.538 Membrane receptor 53081,53081 53081,53081 Ki,IC50 Ki,IC50 Vanilloid receptor 8.35654732351 8.33724216832 Q8NER1 O35433 685997 436.313 Ion channel 52179 52179 IC50 IC50 Endothelin receptor ET-A 4.39794000867 3.23657200644 P25101 P26684 446140 430.491 Membrane receptor 41260 41260 IC50 IC50 Histamine H3 receptor 7.64089913797 6.82876011547 Q9Y5N1 Q9QYN8 494955 346.464 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Cholecystokinin A receptor 7.000315092 7.13225005259 P32238 P30551 708488 594.705 Membrane receptor 53436,53436 53436,53436 IC50,IC50 IC50,IC50 Cholecystokinin A receptor 7.32696147443 7.61531133696 P32238 P30551 708491 556.657 Membrane receptor 53436,53436 53436,53436 IC50,IC50 IC50,IC50 Cholecystokinin A receptor 6.7982938792 6.9977275433 P32238 P30551 708493 581.666 Membrane receptor 53436,53436 53436,53436 IC50,IC50 IC50,IC50 Phospholipase A2 group IIA 4.71425622347 4.43297363384 P14555 P14423 446373 400.551 Enzyme 40039,40039 40039 IC50,IC50 IC50 Cannabinoid CB1 receptor 7.22623694277 6.14387555576 P21554 P20272 709000 858.47 Membrane receptor 53408,53408,53408,53408 53408 Ki,Ki,IC50,IC50 IC50 Cannabinoid CB1 receptor 7.99504744428 5.92335955633 P21554 P20272 709002 970.682 Membrane receptor 53408,53408,53408,53408 53408 Ki,Ki,IC50,IC50 IC50 Cannabinoid CB1 receptor 7.41059926581 8.87289520164 P21554 P20272 709003 1026.79 Membrane receptor 53408,53408,53408,53408 53408 Ki,Ki,IC50,IC50 IC50 Cannabinoid CB1 receptor 7.68614451749 8.74957999769 P21554 P20272 709005 928.602 Membrane receptor 53408,53408,53408,53408 53408 Ki,Ki,IC50,IC50 IC50 Cannabinoid CB1 receptor 7.66131060152 5.83564714422 P21554 P20272 709006 984.709 Membrane receptor 53408,53408,53408,53408 53408 Ki,Ki,IC50,IC50 IC50 Cannabinoid CB1 receptor 5.88873748634 7.53313237965 P21554 P20272 709008 1096.92 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Cannabinoid CB1 receptor 8.25 5.62105730139 P21554 P20272 709009 663.163 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Cannabinoid CB1 receptor 8.5 5.4417715782 P21554 P20272 709010 719.27 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Cannabinoid CB1 receptor 8.21324857785 5.46801044859 P21554 P20272 709011 677.19 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Cannabinoid CB1 receptor 7.83268266525 5.05709945886 P21554 P20272 709012 733.296 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Cannabinoid CB1 receptor 6.37263414341 6.80134291305 P21554 P20272 446956 494.884 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.50031291738 6.10623823794 P21554 P20272 446958 454.82 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.89279003035 7.13786862069 P21554 P20272 446974 446.413 Membrane receptor 42580 42580 IC50 IC50 Sodium channel protein type X alpha subunit 8.69897000434 8.04575749056 Q9Y5Y9 Q62968 709119 336.815 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 8.39794000867 7.18045606446 Q9Y5Y9 Q62968 709120 357.233 Ion channel 53444 53444 IC50 IC50 Cannabinoid CB1 receptor 5.9829666607 6.58169870868 P21554 P20272 446990 494.884 Membrane receptor 42580 42580 IC50 IC50 Adenosine A2a receptor 8.50863830617 7.79588001734 P29274 P30543 709138 433.503 Membrane receptor 53459 53459 Ki Ki Cannabinoid CB1 receptor 6.56383735296 6.72353819583 P21554 P20272 447000 460.439 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.35359627378 6.91364016933 P21554 P20272 447001 420.375 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.70996538864 6.60554831917 P21554 P20272 447002 425.994 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.7878123956 6.82102305271 P21554 P20272 447003 440.021 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.46852108296 6.53610701101 P21554 P20272 447033 440.021 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.47625353319 6.16749108729 P21554 P20272 447034 399.957 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.73048705578 6.7878123956 P21554 P20272 447035 479.965 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.69036983257 6.85078088734 P21554 P20272 447036 493.992 Membrane receptor 42580 42580 IC50 IC50 Sodium channel protein type X alpha subunit 8.09691001301 7.34678748622 Q9Y5Y9 Q62968 709228 405.92 Ion channel 53444 53444 IC50 IC50 Adenosine A2a receptor 7.76955107862 7.07058107429 P29274 P30543 709245 445.514 Membrane receptor 53459 53459 Ki Ki Sodium channel protein type X alpha subunit 6.85387196432 6.25181197299 Q9Y5Y9 Q62968 709339 358.221 Ion channel 53444 53444 IC50 IC50 Adenosine A2a receptor 8.60205999133 8.36653154442 P29274 P30543 709354 434.491 Membrane receptor 53459 53459 Ki Ki Sodium channel protein type X alpha subunit 8.15490195999 7.49485002168 Q9Y5Y9 Q62968 709447 367.829 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 8.52287874528 7.55284196866 Q9Y5Y9 Q62968 709448 421.8 Ion channel 53444 53444 IC50 IC50 Cannabinoid CB1 receptor 6.10385669723 5.1400815148 P21554 P20272 709511 466.791 Membrane receptor 53408,53408 53408 Ki,Ki IC50 Sodium channel protein type X alpha subunit 7.85387196432 8.09691001301 Q9Y5Y9 Q62968 709542 406.908 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 7.06048074738 7.00877392431 Q9Y5Y9 Q62968 709543 408.881 Ion channel 53444 53444 IC50 IC50 Cannabinoid CB1 receptor 6.45717457304 5.6532559454 P21554 P20272 709611 550.951 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Nitric-oxide synthase, brain 6.30980391997 6.95860731484 P29475 P29476 709703 362.485 Enzyme 53397 53397 Ki Ki Cannabinoid CB1 receptor 7.69 5.48425858333 P21554 P20272 709706 607.057 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Cannabinoid CB1 receptor 6.79048498546 5.51755520808 P21554 P20272 709807 564.977 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Adenosine A2a receptor 7.60205999133 7.61978875829 P29274 P30543 709854 420.464 Membrane receptor 53459 53459 Ki Ki Cannabinoid CB1 receptor 7.66 5.35981680808 P21554 P20272 709907 621.084 Membrane receptor 53408,53408,53408 53408 Ki,Ki,IC50 IC50 Adenosine A2a receptor 7.88605664769 7.92081875395 P29274 P30543 709954 434.491 Membrane receptor 53459 53459 Ki Ki Sodium channel protein type X alpha subunit 8.69897000434 6.88605664769 Q9Y5Y9 Q62968 710043 375.341 Ion channel 53444 53444 IC50 IC50 Adenosine A2a receptor 8.11350927483 8.19382002602 P29274 P30543 710059 460.528 Membrane receptor 53459 53459 Ki Ki Adenosine A2a receptor 7.95860731484 7.85387196432 P29274 P30543 710060 460.528 Membrane receptor 53459 53459 Ki Ki Sodium channel protein type X alpha subunit 6.55284196866 6.02227639471 Q9Y5Y9 Q62968 710145 376.329 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 6.7447274949 5.69897000434 Q9Y5Y9 Q62968 710146 376.329 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 6.32790214206 6.08618614762 Q9Y5Y9 Q62968 710246 377.317 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 7.2924298239 6.42021640338 Q9Y5Y9 Q62968 710247 392.395 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 8.09691001301 6.28399665637 Q9Y5Y9 Q62968 710354 393.383 Ion channel 53444 53444 IC50 IC50 Sodium channel protein type X alpha subunit 7.67778070527 7.46852108296 Q9Y5Y9 Q62968 710355 387.355 Ion channel 53444,53932 53444,53932 IC50,IC50 IC50,IC50 Sodium channel protein type X alpha subunit 7.63827216398 7.04095860768 Q9Y5Y9 Q62968 710560 327.379 Ion channel 53444 53444 IC50 IC50 Acetylcholinesterase 7.08354605145 7.04575749056 P22303 P37136 186513 385.501 Enzyme 37075 37075 IC50 IC50 Acetylcholinesterase 6.57057073562 6.56767220774 P22303 P37136 186514 460.608 Enzyme 37075 37075 IC50 IC50 Histamine H3 receptor 8.5484550065 9.15490195999 Q9Y5N1 Q9QYN8 448805 408.576 Membrane receptor 44506,44506 44506 Ki,Ki Ki Gonadotropin-releasing hormone receptor 5.4300604568 4.45241532428 P30968 P30969 448838 498.424 Membrane receptor 44386,44386 44386,44386 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 6.09691001301 4.39848355649 P30968 P30969 448839 462.491 Membrane receptor 44386,44386,42049 44386,44386 IC50,IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 4.85002854999 4.19382002602 P30968 P30969 449089 468.398 Membrane receptor 44386,44386 44386 IC50,IC50 IC50 Dopamine transporter 7.06785127947 6.42021640338 Q01959 P23977 449148 228.118 Transporter 44451,52510 44451 IC50,IC50 IC50 Serotonin transporter 7.26384122684 7.56863623584 P31645 P31652 449148 228.118 Transporter 44451,52510 44451 IC50,IC50 IC50 Dopamine transporter 6.8894102897 6.48148606012 Q01959 P23977 449149 228.118 Transporter 44451 44451 IC50 IC50 Serotonin transporter 6.87614835903 7.18045606446 P31645 P31652 449149 228.118 Transporter 44451 44451 IC50 IC50 Gonadotropin-releasing hormone receptor 5.8525465447 4.2924298239 P30968 P30969 449160 432.465 Membrane receptor 44386,44386 44386 IC50,IC50 IC50 Dopamine transporter 7.01772876696 6.58502665203 Q01959 P23977 449213 228.118 Transporter 44451 44451 IC50 IC50 Serotonin transporter 7.91009488856 8.06550154876 P31645 P31652 449213 228.118 Transporter 44451 44451 IC50 IC50 Acetylcholinesterase 6.618704377 6.6140364294 P22303 P37136 187207 418.528 Enzyme 37075 37075 IC50 IC50 Gonadotropin-releasing hormone receptor 5.20065945055 4.82390874094 P30968 P30969 449374 512.499 Membrane receptor 44386 44386 IC50 IC50 Adenosine A1 receptor 7.92081875395 7.55030864723 P30542 P25099 93525 374.393 Membrane receptor 49741 3214,49741 Ki IC50,Ki Dipeptidyl peptidase IV 8.69897000434 8.33889035263 P27487 P14740 643455 393.442 Enzyme 34705,34705 34705,34705 Ki,Ki Ki,Ki Fatty acid desaturase 1 5.87778412173 5.28659346783 O60427 Q920R3 711565 366.409 Enzyme 53539 53539 IC50 IC50 Gonadotropin-releasing hormone receptor 6.14792474158 5.28399665637 P30968 P30969 449440 534.575 Membrane receptor 44386,44386 44386 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 6.55731938998 5.40893539297 P30968 P30969 449441 498.642 Membrane receptor 44386,44386 44386 IC50,IC50 IC50 Endothelin receptor ET-A 11.3767507096 10.408935393 P25101 P26684 187303 598.511 Membrane receptor 16144 16144 Ki IC50 Gonadotropin-releasing hormone receptor 6.63380312009 6.0043648054 P30968 P30969 449514 548.602 Membrane receptor 44386,44386 44386 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 6.61092437481 6.14874165128 P30968 P30969 449515 562.629 Membrane receptor 44386,44386 44386 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 8.03074013741 6.78919803657 P30968 P30969 449517 496.67 Membrane receptor 44386,44386 44386,44386 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.63057009896 5.99569991412 P30968 P30969 449582 480.604 Membrane receptor 44386,44386 44386,44386 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.93195695131 6.7307131331 P30968 P30969 449583 508.614 Membrane receptor 44386,44386 44386,44386 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 8.16833803319 7.5 P30968 P30969 449644 508.614 Membrane receptor 44386,44386,46195,46195 44386,44386,46195,46195 IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Gonadotropin-releasing hormone receptor 8.10912231267 7.44103308248 P30968 P30969 449645 458.555 Membrane receptor 44386,44386 44386,44386 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 8.76955107862 7.7447274949 P30968 P30969 449646 486.609 Membrane receptor 44386,44386,42049,46170,46170 44386,44386,42049,46170 IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Glucagon receptor 8.40893539297 7.36653154442 P47871 P30082 450136 582.474 Membrane receptor 45153 45153 IC50 IC50 Gastric inhibitory polypeptide receptor 6.44490555142 6.30016227413 P48546 P43219 450136 582.474 Membrane receptor 45153 45153 IC50 IC50 Anandamide amidohydrolase 7.65269740053 7.46852108296 O00519 P97612 450555 365.452 Enzyme 45114,45114,45114,45114 45114 IC50,IC50,IC50,IC50 IC50 Anandamide amidohydrolase 6.81815641206 7.07572071394 O00519 P97612 450625 395.478 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 5.73048705578 6.55284196866 O00519 P97612 450626 395.478 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 6.76195389687 7.32790214206 O00519 P97612 450627 395.478 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 5.88605664769 5.89619627904 O00519 P97612 450628 379.479 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 6.71444269099 6.82973828461 O00519 P97612 450629 379.479 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 5.69897000434 5.77832500293 O00519 P97612 450701 379.479 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 6.45967052521 6.45593195565 O00519 P97612 450702 399.897 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.49894073778 7.73754891027 O00519 P97612 450704 399.897 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.01772876696 7.04095860768 O00519 P97612 450705 383.443 Enzyme 45114 45114 IC50 IC50 Sodium channel protein type X alpha subunit 7.0043648054 7.04575749056 Q9Y5Y9 Q62968 712852 408.762 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 7.72124639905 7.07058107429 Q9Y5Y9 Q62968 712853 459.421 Ion channel 53932 53932 IC50 IC50 Anandamide amidohydrolase 6.84466396253 6.81815641206 O00519 P97612 450780 383.443 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.72124639905 8.2076083105 O00519 P97612 450781 383.443 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 5.30102999566 5.07935499859 O00519 P97612 450782 449.449 Enzyme 45114 45114 IC50 IC50 Serotonin 2a (5-HT2a) receptor 8.43179827593 8.61978875829 P28223 P14842 686805 364.802 Membrane receptor 52268 52268 Ki Ki Anandamide amidohydrolase 5.97224279531 6.45593195565 O00519 P97612 450858 411.544 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 6.07935499859 6.93181413825 O00519 P97612 450859 383.443 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.16115090926 6.91364016933 O00519 P97612 450921 379.479 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.57348873864 7.58502665203 O00519 P97612 450923 366.44 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 8.00877392431 8.06048074738 O00519 P97612 450924 366.44 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 6.57511836337 7.24412514433 O00519 P97612 450988 367.428 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.98716277529 8.20065945055 O00519 P97612 450989 367.428 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.88605664769 7.54060751224 O00519 P97612 450990 397.454 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.30102999566 7.26760624018 O00519 P97612 450992 401.873 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 5.57397698431 5.88041422504 O00519 P97612 451057 368.416 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.63827216398 7.96657624451 O00519 P97612 451058 367.428 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 8.69464863055 8.8696662315 O00519 P97612 451059 423.515 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 5.98422124361 6.19517932128 O00519 P97612 451061 431.513 Enzyme 45114 45114 IC50 IC50 Steroid 5-alpha-reductase 2 6.67778070527 5.45593195565 P31213 P31214 188947 397.482 Enzyme 16544 16544 IC50 IC50 Steroid 5-alpha-reductase 2 6.08092190762 6.16115090926 P31213 P31214 188952 412.48 Enzyme 16544 16544 IC50 IC50 Anandamide amidohydrolase 6.49485002168 6.94692155652 O00519 P97612 451130 448.564 Enzyme 45114 45114 IC50 IC50 Anandamide amidohydrolase 7.15490195999 7.59006687667 O00519 P97612 451132 356.402 Enzyme 45114 45114 IC50 IC50 Histamine H3 receptor 8.13076828027 7.43179827593 Q9Y5N1 Q9QYN8 713387 404.544 Membrane receptor 53911 53911 Ki Ki Histamine H3 receptor 7.72124639905 6.8601209136 Q9Y5N1 Q9QYN8 451250 507.73 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 8.93930215965 8.64016451766 Q9Y5N1 Q9QYN8 451263 531.772 Membrane receptor 44314 44314 Ki Ki Steroid 5-alpha-reductase 2 6.2757241304 6.43179827593 P31213 P31214 189164 411.492 Enzyme 16544 16544 IC50 IC50 Histamine H3 receptor 8.79588001734 8.26760624018 Q9Y5N1 Q9QYN8 713477 339.474 Membrane receptor 53911 53911 Ki Ki Histamine H3 receptor 9.67778070527 8.59006687667 Q9Y5N1 Q9QYN8 451337 455.719 Membrane receptor 44314,47387 44314,44314,47387 Ki,Ki Ki,Ki,Ki Sodium channel protein type X alpha subunit 8.22184874962 6.72124639905 Q9Y5Y9 Q62968 713489 369.802 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 8.22184874962 6.55284196866 Q9Y5Y9 Q62968 713490 323.776 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 8.52287874528 7.28399665637 Q9Y5Y9 Q62968 713491 337.803 Ion channel 53932 53932 IC50 IC50 Steroid 5-alpha-reductase 2 6.38721614328 5.95860731484 P31213 P31214 189223 429.483 Enzyme 16544 16544 IC50 IC50 Steroid 5-alpha-reductase 2 5.45593195565 6.0268721464 P31213 P31214 189224 441.518 Enzyme 16544 16544 IC50 IC50 Steroid 5-alpha-reductase 2 8.15490195999 7.42021640338 P31213 P31214 189259 455.605 Enzyme 16544 16544 IC50 IC50 Histamine H3 receptor 8.85387196432 8.28399665637 Q9Y5N1 Q9QYN8 713572 338.486 Membrane receptor 53911 53911 Ki Ki Histamine H3 receptor 9.05060999336 8.5376020021 Q9Y5N1 Q9QYN8 713573 352.513 Membrane receptor 53911 53911 Ki Ki Sodium channel protein type X alpha subunit 7.56863623584 6.95860731484 Q9Y5Y9 Q62968 713584 337.803 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 7.72124639905 6.44369749923 Q9Y5Y9 Q62968 713585 372.248 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 7.43179827593 6.55284196866 Q9Y5Y9 Q62968 713679 409.869 Ion channel 53932 53932 IC50 IC50 Histamine H3 receptor 7.79588001734 8.06550154876 Q9Y5N1 Q9QYN8 424795 384.561 Membrane receptor 38362 38362 Ki Ki Sodium channel protein type X alpha subunit 7.52287874528 6.25963731051 Q9Y5Y9 Q62968 713857 393.869 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 8.69897000434 7.92081875395 Q9Y5Y9 Q62968 713858 347.41 Ion channel 53932 53932 IC50 IC50 Steroid 5-alpha-reductase 2 5.95860731484 6.05551732785 P31213 P31214 189634 425.519 Enzyme 16544 16544 IC50 IC50 Sodium channel protein type X alpha subunit 9.0 7.16749108729 Q9Y5Y9 Q62968 713940 333.384 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 8.69897000434 7.72124639905 Q9Y5Y9 Q62968 713941 347.41 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 8.09691001301 7.07572071394 Q9Y5Y9 Q62968 714027 328.367 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 7.30980391997 6.88605664769 Q9Y5Y9 Q62968 714028 358.393 Ion channel 53932 53932 IC50 IC50 Steroid 5-alpha-reductase 2 7.22184874962 7.09691001301 P31213 P31214 189828 423.588 Enzyme 16544 16544 IC50 IC50 Sodium channel protein type X alpha subunit 6.82390874094 6.34678748622 Q9Y5Y9 Q62968 714122 328.367 Ion channel 53932 53932 IC50 IC50 Histamine H3 receptor 7.70553377384 8.1018235165 Q9Y5N1 Q9QYN8 452023 517.959 Membrane receptor 44314,47387 44314,47387 Ki,Ki Ki,Ki Histamine H3 receptor 6.26520017041 6.0 Q9Y5N1 Q9QYN8 452024 356.545 Membrane receptor 44314,47387 44314,47387 Ki,Ki Ki,Ki Histamine H3 receptor 7.42021640338 7.61083391564 Q9Y5N1 Q9QYN8 452025 342.518 Membrane receptor 44314 44314 Ki Ki Sodium channel protein type X alpha subunit 8.30102999566 7.79588001734 Q9Y5Y9 Q62968 714208 373.329 Ion channel 53932 53932 IC50 IC50 Sodium channel protein type X alpha subunit 7.7447274949 6.76955107862 Q9Y5Y9 Q62968 714209 387.355 Ion channel 53932 53932 IC50 IC50 Histamine H3 receptor 7.40011692793 6.70996538864 Q9Y5N1 Q9QYN8 452101 471.677 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 7.79048498546 6.80966830183 Q9Y5N1 Q9QYN8 452155 447.655 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 8.77989191196 7.61978875829 Q9Y5N1 Q9QYN8 452157 443.667 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 7.21968268786 6.59006687667 Q9Y5N1 Q9QYN8 452158 400.597 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 7.30016227413 6.53017798402 Q9Y5N1 Q9QYN8 452235 413.639 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 7.51004152058 6.61978875829 Q9Y5N1 Q9QYN8 452236 449.693 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 7.63078414259 6.85078088734 Q9Y5N1 Q9QYN8 452237 434.678 Membrane receptor 44314 44314 Ki Ki Histamine H3 receptor 8.11013827874 7.20971483597 Q9Y5N1 Q9QYN8 452238 482.721 Membrane receptor 44314 44314 Ki Ki Monoamine oxidase A 5.25492520842 5.25492520842 P21397 P21396 452516 379.498 Enzyme 49675 44921 IC50 IC50 Steroid 5-alpha-reductase 2 6.58502665203 5.60205999133 P31213 P31214 190596 379.492 Enzyme 16544 16544 IC50 IC50 Steroid 5-alpha-reductase 2 7.95860731484 5.52287874528 P31213 P31214 190627 441.578 Enzyme 16544 16544 IC50 IC50 Alpha-2a adrenergic receptor 6.94309514866 6.50445566245 P08913 P22909 190658 279.805 Membrane receptor 13032 13032 Ki Ki Neurokinin 1 receptor 9.80666135802 9.5376020021 P25103 P14600 381329 1210.29 Membrane receptor 35835,45287 45287 Ki,Ki Ki Vasopressin V2 receptor 8.63827216398 7.38721614328 P30518 Q00788 453484 478.583 Membrane receptor 44817 44817 IC50 IC50 Matrix metalloproteinase 13 7.92081875395 8.36653154442 P45452 P23097 453588 393.457 Enzyme 3166 4737 IC50 IC50 Vasopressin V2 receptor 8.32790214206 7.18708664336 P30518 Q00788 453594 492.61 Membrane receptor 44817 44817 IC50 IC50 Vasopressin V2 receptor 8.36653154442 7.82390874094 P30518 Q00788 453595 506.636 Membrane receptor 44817 44817 IC50 IC50 Calcitonin gene-related peptide 1 9.04959803259 8.05060999336 P06881 P01256 453737 3427.91 NA 44809,44809 44809 Ki,IC50 IC50 Calcitonin gene-related peptide 1 8.67778070527 7.69036983257 P06881 P01256 453739 3453.99 NA 44809 44809 IC50 IC50 Monoamine oxidase B 7.55284196866 8.44369749923 P27338 P19643 453850 197.224 Enzyme 44818 44818 Ki IC50 Vasopressin V2 receptor 7.6883753548 7.88605664769 P30518 Q00788 454158 449.492 Membrane receptor 44817,44817 44817 IC50,Ki IC50 Adenosine A3 receptor 6.70053912009 6.23358715289 P33765 P28647 192029 499.52 Membrane receptor 16653,15395,21026,49861 15395 Ki,Ki,Ki,IC50 Ki Adenosine A1 receptor 6.51999305704 5.58502665203 P30542 P25099 192029 499.52 Membrane receptor 3027,15395,21026 16653,15395,13048 IC50,Ki,Ki Ki,Ki,Ki Adenosine A2a receptor 7.33535802444 7.89125802789 P29274 P30543 192029 499.52 Membrane receptor 15395,21026,38739,42591,47890,49861,49861 13048,16653 Ki,Ki,Ki,Ki,Ki,Ki,IC50 Ki,Ki Neurokinin 1 receptor 8.7447274949 7.63827216398 P25103 P14600 556293 1343.37 Membrane receptor 47632 47632 Ki Ki C-X-C chemokine receptor type 4 6.96257350206 5.8416375079 P61073 O08565 454218 715.802 Membrane receptor 44811 44811 IC50 IC50 C-X-C chemokine receptor type 4 7.31875876262 7.3986196563 P61073 O08565 454219 378.598 Membrane receptor 44811,44811,44811 44811,44811 IC50,IC50,IC50 IC50,IC50 Histamine H3 receptor 8.60205999133 7.66354026615 Q9Y5N1 Q9QYN8 599975 407.936 Membrane receptor 49904 49904 Ki Ki Histamine H3 receptor 8.56863623584 7.76955107862 Q9Y5N1 Q9QYN8 454365 295.847 Membrane receptor 46449,46764,44709,46281,46281,46281,53042,53055 46281 Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki Ki C-X-C chemokine receptor type 4 8.52775866392 7.95860731484 P61073 O08565 454523 406.651 Membrane receptor 44811,44811 44811 IC50,IC50 IC50 Dopamine transporter 6.20480202641 6.43179827593 Q01959 P23977 192908 297.415 Transporter 6463,30228,31495,37434,38837,39371,45878,47532,50055,51366 45021 Ki,Ki,IC50,IC50,IC50,Ki,IC50,IC50,Ki,Ki IC50 Serotonin transporter 8.30102999566 8.33724216832 P31645 P31652 192908 297.415 Transporter 6463,30228,31495,37434,38837,39371,45878,47195,47532,50055,51128,51366 45021 Ki,Ki,IC50,IC50,IC50,Ki,IC50,IC50,IC50,Ki,IC50,Ki Ki Excitatory amino acid transporter 1 6.18045606446 6.01322826573 P43003 P24942 455730 422.475 Transporter 45442,45442,53164 45442 IC50,IC50,IC50 IC50 Serotonin transporter 8.31875876262 9.0 P31645 P31652 393973 366.496 Transporter 36227 36227 Ki Ki Vanilloid receptor 10.0200025808 9.72734644177 Q8NER1 O35433 456371 628.708 Ion channel 5440,36194,49452,53995 17091,45405,45405,53995 Ki,IC50,IC50,Ki Ki,IC50,Ki,IC50 Adenosine A3 receptor 8.92081875395 8.95860731484 P33765 P28647 194619 510.286 Membrane receptor 17361,16675,15395,20156,30254,30254,31055,31066,34814,39543,43854,45320,45320,45270,49365,49365 15395,17161,39543,45270 Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,IC50,Ki,IC50,Ki,Ki,Ki Ki,Ki,Ki,Ki Adenosine A1 receptor 7.30715308072 7.26760624018 P30542 P25099 194619 510.286 Membrane receptor 15395,17361,20156,31066,39543,45270,49365 14546,39543 Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A2a receptor 6.2924298239 7.25181197299 P29274 P30543 194619 510.286 Membrane receptor 14051,14051,14051,15395,20156,31066,39543,45270,49365 14546,39543 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Metabotropic glutamate receptor 5 8.0 7.95860731484 P41594 P31424 194729 223.27 Membrane receptor 35537 35537 Ki Ki Dihydrofolate reductase 4.49485002168 1.99567862622 P00374 Q920D2 382026 313.421 Enzyme 36076 36076 IC50 IC50 Cannabinoid CB2 receptor 7.20065945055 7.2076083105 P34972 Q9QZN9 582616 303.399 Membrane receptor 48957 48957 Ki IC50 11-beta-hydroxysteroid dehydrogenase 1 7.28399665637 6.61261017366 P28845 P16232 457593 411.458 Enzyme 46089,46089,46089 46089 IC50,IC50,IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.39794000867 5.45481663178 P36544 Q05941 195974 None Ion channel 36679,36679,45323 38731 IC50,IC50,IC50 Ki Adenosine A3 receptor 8.85387196432 9.48148606012 P33765 P28647 76361 544.731 Membrane receptor 17361,2660,16675,16675,16675,31066,36081,37136,38563,38563,38785,39543,44562,45270,47561,49365,49365 39543,45270 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A1 receptor 6.65364702555 6.6768961939 P30542 P25099 76361 544.731 Membrane receptor 17361,31066,36081,37136,38563,38785,39543,44562,45270,47561,49365 2660,39543 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Adenosine A2a receptor 5.27083521031 6.78985705753 P29274 P30543 76361 544.731 Membrane receptor 36081,37136,38563,38785,39543,44562,45270,47561,49365 2660,39543 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Diacylglycerol O-acyltransferase 1 7.82390874094 7.72124639905 O75907 Q9ERM3 458543 394.467 Enzyme 46013 46013 IC50 IC50 Diacylglycerol O-acyltransferase 1 7.82390874094 8.04575749056 O75907 Q9ERM3 458603 420.504 Enzyme 46013 46013 IC50 IC50 Angiotensin II type 2 (AT-2) receptor 5.34678748622 5.34678748622 P50052 P35351 32747 550.654 Membrane receptor 30228 12035,817 IC50 IC50,IC50 Melanocortin receptor 4 8.13005567246 8.40553575812 P32245 P70596 426001 621.024 Membrane receptor 38716,38716 38716,38716 IC50,IC50 IC50,IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 7.78515615195 7.8696662315 P36544 Q05941 600799 258.319 Ion channel 49908 49908 Ki Ki Mu opioid receptor 6.58502665203 7.19168558549 P35372 P33535 32837 435.602 Membrane receptor 45228 12391,12391 Ki IC50,IC50 Mu opioid receptor 8.62287553703 8.42943195494 P35372 P33535 197398 571.667 Membrane receptor 31329,48894 17669,17669,31475,35810,36256,36495,38119,38291,43813,43813,43813,46977,42175,47725,51376,52873 Ki,Ki Ki,Ki,Ki,Ki,Ki,IC50,Ki,IC50,Ki,Ki,IC50,IC50,Ki,Ki,Ki,Ki Adenosine A1 receptor 6.4528518013 6.64589156085 P30542 P25099 197514 375.344 Membrane receptor 16564,30783 16564 Ki,Ki Ki Adenosine A2a receptor 6.97930365742 7.01055018233 P29274 P30543 197514 375.344 Membrane receptor 16564,30783 16564 Ki,Ki Ki Dipeptidyl peptidase IV 7.91816592311 7.89279003035 P27487 P14740 460014 366.409 Enzyme 47179,47179 47179 IC50,IC50 IC50 Glucagon receptor 7.19745526906 5.85387196432 P47871 P30082 460166 559.987 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glucagon receptor 7.18095513901 5.76955107862 P47871 P30082 460167 575.987 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glucagon receptor 7.03386461205 5.56863623584 P47871 P30082 460168 559.987 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glucagon receptor 7.16432099828 5.69897000434 P47871 P30082 460169 609.539 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Anandamide amidohydrolase 9.22184874962 9.42021640338 O00519 P97612 382573 358.39 Enzyme 36082 36082 Ki Ki Vanilloid receptor 8.72796597782 9.1883753548 Q8NER1 O35433 198372 372.892 Ion channel 38185,38185,38185,38185,44549,50255 38185,38185,38185,38185 IC50,IC50,IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Norepinephrine transporter 5.89245087026 5.48174934869 P23975 Q9WTR4 198461 303.353 Transporter 15623,15623,15113,21665,30737,31321,31321,35284,35284,36559,47133,45958,45958,46012,46012,44983,44983,49019,49019,49267,49267 15861,13641,14202,12788,17584,6436,13096,3800,5430,4355,31903 IC50,Ki,Ki,IC50,Ki,Ki,IC50,IC50,Ki,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50 Ki,IC50,IC50,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki Dopamine transporter 6.43062609038 6.64208186242 Q01959 P23977 198461 303.353 Transporter 15623,4058,16613,15623,15113,21665,30737,31321,34825,34825,35284,36559,47133,42481,42481,45958,45958,46012,46012,44983,44983,49019,49019,49267,49267 14838,11608,13641,11191,3964,14202,4585,12788,15202,3456,3189,4972,6436,5430,14321,14321,14322,14322,4355,4998,13096,3456,12326,3800,3800,13833,15861,30380,31446,31446,31903,31903,36501,49074 IC50,IC50,Ki,Ki,Ki,IC50,Ki,IC50,Ki,IC50,IC50,Ki,IC50,IC50,IC50,IC50,Ki,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50 IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,IC50,IC50,Ki,IC50,Ki,Ki Serotonin transporter 6.41228903498 6.54363396687 P31645 P31652 198461 303.353 Transporter 16613,15623,15113,21665,30737,31321,31321,35284,35284,36559,47133,45958,45958,46012,46012,44983,44983,49019,49019,49267,49267 13641,3964,14202,12788,4972,6436,15861,5430,4355,3964,4770,3800,31446,31903,49074 Ki,Ki,Ki,IC50,Ki,Ki,IC50,IC50,Ki,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50,Ki,IC50 IC50,IC50,IC50,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki Neuropeptide Y receptor type 5 8.61978875829 8.76955107862 Q15761 Q63634 461011 400.43 Membrane receptor 47123,46791,46791 46791 Ki,IC50,IC50 IC50 Urotensin II receptor 8.09691001301 7.46852108296 Q9UKP6 P49684 461020 539.363 Membrane receptor 48952,48952 48952 Ki,IC50 IC50 Glutamate receptor ionotropic, AMPA 1 7.18708664336 7.43179827593 P42261 P19490 198912 233.609 Ion channel 14175 45271 Ki Ki Glutamate receptor ionotropic, AMPA 2 7.27490547892 6.51125251546 P42262 P19491 198912 233.609 Ion channel 14175 45271,45271 Ki Ki,IC50 Glutamate receptor ionotropic, AMPA 4 6.34582345812 6.25103713874 P48058 P19493 198912 233.609 Ion channel 14175 45271 Ki Ki Glutamate receptor ionotropic, AMPA 1 7.03621217265 5.55284196866 P42261 P19490 198946 278.06 Ion channel 14175 45271 Ki IC50 Glutamate receptor ionotropic, AMPA 1 6.41341269533 4.93930215965 P42261 P19490 198978 199.164 Ion channel 14175 45271 Ki IC50 Histamine H3 receptor 8.09691001301 7.24412514433 Q9Y5N1 Q9QYN8 339003 474.273 Membrane receptor 30729 30729 Ki Ki Glucagon receptor 7.26508899201 5.7447274949 P47871 P30082 461209 629.648 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glucagon receptor 7.12966078739 5.26760624018 P47871 P30082 461361 565.606 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glucagon receptor 7.04415492062 5.35654732351 P47871 P30082 461362 581.605 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glucagon receptor 7.18498957444 5.79588001734 P47871 P30082 461364 580.525 Membrane receptor 47089,47089 47089 IC50,IC50 IC50 Glutamate receptor ionotropic, AMPA 1 7.83268266525 7.47890920274 P42261 P19490 199497 217.155 Ion channel 14175 45271,45271 Ki Ki,IC50 Glutamate receptor ionotropic, AMPA 2 7.60032627852 7.3675910885 P42262 P19491 199497 217.155 Ion channel 14175 45271,45271 Ki Ki,IC50 Glutamate receptor ionotropic, AMPA 4 6.51570016065 5.91727396358 P48058 P19493 199497 217.155 Ion channel 14175 45271,45271 Ki Ki,IC50 Glutamate receptor ionotropic, AMPA 1 4.7328282716 6.08234499957 P42261 P19490 469283 257.266 Ion channel 45271 45271,45271 IC50 Ki,IC50 Glutamate receptor ionotropic kainate 1 8.42021640338 8.28399665637 P39086 P22756 469283 257.266 Ion channel 45271 45271 IC50 IC50 Glutamate receptor ionotropic, AMPA 1 6.7878123956 5.77729131512 P42261 P19490 199610 325.061 Ion channel 14175 45271,45271 Ki Ki,IC50 Glutamate receptor ionotropic, AMPA 2 6.75448733219 6.97881070093 P42262 P19491 199610 325.061 Ion channel 14175 45271 Ki Ki Glutamate receptor ionotropic, AMPA 4 6.01233373507 6.13194363818 P48058 P19493 199610 325.061 Ion channel 14175 45271 Ki Ki Vasopressin V1b receptor 6.8601209136 7.25181197299 P47901 P48974 572207 621.808 Membrane receptor 48483 48483 Ki Ki Phospholipase A2 group IIA 5.40893539297 4.41566877563 P14555 P14423 462520 416.55 Enzyme 42278,40039,40039 40039 IC50,IC50,IC50 IC50 Metabotropic glutamate receptor 1 6.71896663275 6.07987667371 Q13255 P23385 296377 379.515 Membrane receptor 21599 21599 IC50 IC50 Histamine H3 receptor 10.0 9.50863830617 Q9Y5N1 Q9QYN8 631571 397.512 Membrane receptor 51341 51341 Ki Ki Serotonin transporter 6.6615435064 7.54060751224 P31645 P31652 514335 467.551 Transporter 44692 44692 IC50 Ki Cannabinoid CB1 receptor 6.09799710865 6.27901425585 P21554 P20272 466039 493.992 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 7.20204035626 6.98716277529 P21554 P20272 466061 490.864 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 7.30627305108 7.08460016479 P21554 P20272 466062 504.89 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.83564714422 6.89619627904 P21554 P20272 466063 504.89 Membrane receptor 42580 42580 IC50 IC50 Cannabinoid CB1 receptor 6.54363396687 6.62525165399 P21554 P20272 466064 464.826 Membrane receptor 42580 42580 IC50 IC50 Adenosine A3 receptor 7.69897000434 6.94692155652 P33765 P28647 466130 308.293 Membrane receptor 4326,17602,4574,17615,21026,30325,31066,34841,35256,35729,37136,38739,38785,44049,42591,47890,49861,51223 14501,15395,16119 Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki Ki,Ki,Ki Adenosine A1 receptor 7.85387196432 7.9829666607 P30542 P25099 466130 308.293 Membrane receptor 3027,17615,15395,4326,21026,30325,31066,34841,35256,35729,37136,38785,44049,49861,51223 3027,9678,9748,9679,9679,14501,16119,11295,11295,11295,9748,13649,13048 IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki IC50,IC50,IC50,IC50,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Adenosine A2a receptor 7.66857388337 8.10790539731 P29274 P30543 466130 308.293 Membrane receptor 17615,4574,17274,17274,17274,17274,14051,14051,14051,4326,21026,30325,31066,34814,34841,35256,35729,37136,37208,38785,43854,45320,45320,49861,49861,51223 16119,13649,13048,14501 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,IC50,Ki,Ki,IC50,Ki Ki,Ki,Ki,Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.22184874962 7.96040937698 P36544 Q05941 427222 388.247 Ion channel 38619,38619,38619 38619,38619,38619,38619,38619,38619 IC50,IC50,IC50 IC50,Ki,IC50,Ki,IC50,Ki Adenosine A1 receptor 7.04963514562 6.53165266959 P30542 P25099 204440 344.777 Membrane receptor 17161 17161 Ki Ki Dopamine D2 receptor 7.05551732785 7.78504315112 P14416 P61169 466587 343.418 Membrane receptor 41947 47870,47870 Ki Ki,IC50 Dopamine D2 receptor 8.42021640338 8.22679036658 P14416 P61169 466588 359.418 Membrane receptor 41947 47870,47870 Ki Ki,IC50 Adenosine A1 receptor 5.87614835903 6.70333480974 P30542 P25099 204469 358.804 Membrane receptor 17161 17161 Ki Ki Adenosine A2a receptor 7.69897000434 5.19791074212 P29274 P30543 204469 358.804 Membrane receptor 17161 17161 Ki Ki P2X purinoceptor 7 7.60205999133 6.74957999769 Q99572 Q64663 467075 498.576 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.87942606879 7.02227639471 Q99572 Q64663 467076 472.969 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 5.98716277529 6.5376020021 Q99572 Q64663 467077 486.996 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.26760624018 5.39147396642 Q99572 Q64663 467078 494.008 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.50863830617 5.50723961097 Q99572 Q64663 467143 491.969 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 5.19382002602 4.98716277529 Q99572 Q64663 467144 490.985 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.10790539731 6.2076083105 Q99572 Q64663 467145 448.945 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 7.22184874962 6.90308998699 Q99572 Q64663 467209 438.953 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.95078197733 6.95860731484 Q99572 Q64663 467210 438.953 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 7.39794000867 7.24412514433 Q99572 Q64663 467211 475.973 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 7.1739251973 7.03151705145 Q99572 Q64663 467212 475.973 Ion channel 43867 43867 IC50 IC50 Adenosine A1 receptor 6.71444269099 6.85387196432 P30542 P25099 205102 560.796 Membrane receptor 17161 17161 Ki Ki Adenosine A2a receptor 6.65169513695 6.45842075605 P29274 P30543 205102 560.796 Membrane receptor 17161 17161 Ki Ki P2X purinoceptor 7 7.34678748622 6.95860731484 Q99572 Q64663 467267 463.963 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.88605664769 7.25181197299 Q99572 Q64663 467268 497.979 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 6.31875876262 5.97061622231 Q99572 Q64663 467349 516.037 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 5.77989191196 5.28483264215 Q99572 Q64663 467350 512.993 Ion channel 43867 43867 IC50 IC50 P2X purinoceptor 7 5.87614835903 5.69036983257 Q99572 Q64663 467351 459.931 Ion channel 43867 43867 IC50 IC50 Adenosine A1 receptor 9.14266750357 8.81043792696 P30542 P25099 76666 356.462 Membrane receptor 13965 13965,11377 Ki Ki,Ki P2X purinoceptor 7 6.95860731484 6.7447274949 Q99572 Q64663 467409 480.005 Ion channel 43867 43867 IC50 IC50 Histamine H1 receptor 8.06048074738 7.39794000867 P35367 P31390 34234 383.507 Membrane receptor 43952 39442 Ki IC50 Histamine H3 receptor 7.38721614328 6.8601209136 Q9Y5N1 Q9QYN8 689681 442.556 Membrane receptor 52388 52388 IC50 IC50 Hexokinase type IV 7.58502665203 7.58502665203 P35557 P17712 646012 462.625 Enzyme 51557 51557 IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 7.67778070527 7.3767507096 P28845 P16232 468242 500.553 Enzyme 43826 43826 IC50 IC50 Dopamine D1 receptor 6.93554201077 5.82973828461 P21728 P18901 468359 365.465 Membrane receptor 43771 45044 Ki Ki 11-beta-hydroxysteroid dehydrogenase 1 8.0 7.88605664769 P28845 P16232 468426 487.511 Enzyme 43826 43826 IC50 IC50 Metabotropic glutamate receptor 1 6.97881070093 7.10790539731 Q13255 P23385 296525 370.485 Membrane receptor 21599 21599 IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 7.58502665203 7.09151498112 P28845 P16232 468519 469.456 Enzyme 43826 43826 IC50 IC50 Butyrylcholinesterase 5.81875876262 7.31875876262 P06276 Q9JKC1 206406 446.495 Enzyme 21324,35447 14639 IC50,IC50 IC50 Acetylcholinesterase 9.52287874528 7.69897000434 P22303 P37136 206406 446.495 Enzyme 21324,35447,38283 14639 IC50,IC50,IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 6.52287874528 6.95860731484 P28845 P16232 468589 504.495 Enzyme 43826 43826 IC50 IC50 Adenosine A3 receptor 8.13667713988 7.00877392431 P33765 P28647 468967 361.394 Membrane receptor 45270 45270 Ki Ki Adenosine A3 receptor 8.82390874094 7.76955107862 P33765 P28647 469023 377.849 Membrane receptor 45270 45270 Ki Ki Adenosine A3 receptor 8.16749108729 8.20065945055 P33765 P28647 469024 422.3 Membrane receptor 45270 45270 Ki Ki Adenosine A3 receptor 8.60205999133 7.31875876262 P33765 P28647 469025 469.3 Membrane receptor 45270 45270 Ki Ki Adenosine A3 receptor 9.60205999133 8.73048705578 P33765 P28647 469141 526.351 Membrane receptor 45270,49365 45270,49365 Ki,Ki Ki,Ki Glutamate receptor ionotropic, AMPA 1 5.90717227054 6.22184874962 P42261 P19490 469285 255.25 Ion channel 45271,45271 45271,45271 IC50,IC50 Ki,IC50 Glutamate receptor ionotropic kainate 1 8.72124639905 8.2757241304 P39086 P22756 469285 255.25 Ion channel 45271 45271 IC50 IC50 Histamine H3 receptor 5.80594939921 5.80594939921 Q9Y5N1 Q9QYN8 469986 473.202 Membrane receptor 47344,47344 45258,45258 Ki,IC50 Ki,IC50 Vanilloid receptor 6.26841123481 6.9829666607 Q8NER1 O35433 471269 566.813 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.64975198167 6.94692155652 Q8NER1 O35433 471270 536.808 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.56224943718 7.11350927483 Q8NER1 O35433 471271 568.807 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.22914798836 7.60205999133 Q8NER1 O35433 471272 511.35 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.92081875395 7.44369749923 Q8NER1 O35433 471338 525.377 Ion channel 45022 45022 IC50 IC50 Anandamide amidohydrolase 7.71010820169 7.7447274949 O00519 P97612 471461 497.653 Enzyme 45059,45059,45059,45059 45059 IC50,IC50,IC50,IC50 IC50 Vanilloid receptor 7.20065945055 7.48148606012 Q8NER1 O35433 471495 539.403 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.52287874528 7.79588001734 Q8NER1 O35433 471496 541.376 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.73518217699 6.92445303861 Q8NER1 O35433 471498 582.471 Ion channel 45022 45022 IC50 IC50 Cannabinoid CB2 receptor 6.95467702121 7.48148606012 P34972 Q9QZN9 471531 428.458 Membrane receptor 44207,44207,45050 44207 IC50,IC50,IC50 IC50 Vanilloid receptor 7.22914798836 7.36653154442 Q8NER1 O35433 471591 499.34 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.31875876262 7.46852108296 Q8NER1 O35433 471592 527.393 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.38721614328 7.26760624018 Q8NER1 O35433 471593 543.392 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.88605664769 8.04575749056 Q8NER1 O35433 471594 513.366 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 8.69897000434 9.0 Q8NER1 O35433 471675 527.393 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 8.52287874528 8.52287874528 Q8NER1 O35433 471676 525.377 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.40893539297 7.95860731484 Q8NER1 O35433 471677 584.444 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 9.0 9.30102999566 Q8NER1 O35433 471678 486.298 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.82390874094 7.14874165128 Q8NER1 O35433 471759 439.357 Ion channel 45022,53995 45022 IC50,IC50 IC50 Vanilloid receptor 7.8210325765 8.39794000867 Q8NER1 O35433 471835 456.272 Ion channel 45022,45022 45022,45022,45022 IC50,IC50 IC50,IC50,IC50 Vanilloid receptor 6.16749108729 6.06348625752 Q8NER1 O35433 471836 456.272 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.29929628285 6.26760624018 Q8NER1 O35433 471900 470.298 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.63827216398 8.22184874962 Q8NER1 O35433 471901 415.435 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 8.04575749056 8.79588001734 Q8NER1 O35433 471902 435.853 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.19382002602 7.49485002168 Q8NER1 O35433 471903 421.827 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.36653154442 7.58502665203 Q8NER1 O35433 471904 433.473 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.63078414259 6.65560772631 Q8NER1 O35433 471969 465.472 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.2924298239 7.85387196432 Q8NER1 O35433 471970 401.408 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.13076828027 7.43179827593 Q8NER1 O35433 471971 455.38 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.02227639471 7.2757241304 Q8NER1 O35433 472034 481.281 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.90308998699 7.26760624018 Q8NER1 O35433 472035 485.313 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.16115090926 7.24412514433 Q8NER1 O35433 472128 499.296 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.68613277963 6.7166987713 Q8NER1 O35433 472239 456.272 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.75448733219 6.76955107862 Q8NER1 O35433 472241 388.274 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.85387196432 8.39794000867 Q8NER1 O35433 472308 457.26 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.48148606012 7.49485002168 Q8NER1 O35433 472309 402.3 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 8.0 8.52287874528 Q8NER1 O35433 472310 430.353 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.95860731484 9.0 Q8NER1 O35433 472311 444.38 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.50863830617 8.69897000434 Q8NER1 O35433 472312 474.363 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.01772876696 7.92081875395 Q8NER1 O35433 472386 434.365 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 8.30102999566 8.52287874528 Q8NER1 O35433 472387 466.364 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 9.0 9.30102999566 Q8NER1 O35433 472463 521.443 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 7.67778070527 8.04575749056 Q8NER1 O35433 472464 490.717 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 8.52287874528 8.69897000434 Q8NER1 O35433 472465 504.743 Ion channel 45022 45022 IC50 IC50 Vanilloid receptor 6.08618614762 5.49620931694 Q8NER1 O35433 472129 514.308 Ion channel 45022 45022 IC50 IC50 Coagulation factor X 8.63827216398 8.05700040663 P00742 Q63207 473774 543.081 Enzyme 44187,45639,45639,49374,49394 45639 IC50,IC50,Ki,IC50,IC50 Ki Histamine H3 receptor 9.22184874962 8.94981472744 Q9Y5N1 Q9QYN8 212531 316.481 Membrane receptor 30729,36041,36915,37369,38362,45718,46449,51148,53407 30729,38362 Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki Ki,Ki Histamine H3 receptor 8.91143937264 8.0 Q9Y5N1 Q9QYN8 474746 375.892 Membrane receptor 45602,45602 45602 Ki,IC50 IC50 Phospholipase A2 group IIA 5.79588001734 7.04575749056 P14555 P14423 474946 490.715 Enzyme 44657 44657 IC50 IC50 Monoamine oxidase B 5.61978875829 5.82681373159 P27338 P19643 603565 251.345 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 4.39794000867 5.06148027482 P21397 P21396 603565 251.345 Enzyme 49639 49639 Ki Ki Metabotropic glutamate receptor 4 5.34412306947 5.69250396209 Q14833 P31423 476037 294.305 Membrane receptor 44620,52028 47355 IC50,IC50 IC50 Monoamine oxidase B 5.67778070527 5.66354026615 P27338 P19643 603658 223.334 Enzyme 49639 49639 Ki Ki Monoamine oxidase A 5.01772876696 5.66354026615 P21397 P21396 603658 223.334 Enzyme 49639 49639 Ki Ki Gonadotropin-releasing hormone receptor 8.29335011796 7.56304920107 P30968 P30969 476283 522.641 Membrane receptor 46195,46195 46195,46195 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 8.05284196866 7.24452652566 P30968 P30969 476284 599.725 Membrane receptor 46195,46195 46195,46195 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.79588001734 6.99064975067 P30968 P30969 476355 494.631 Membrane receptor 46195,46195 46195,46195 IC50,IC50 IC50,IC50 Gonadotropin-releasing hormone receptor 7.73683036131 6.81875876262 P30968 P30969 476356 476.615 Membrane receptor 46195,46195,50731,50731 46195,46195,50731,50731 IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Gonadotropin-releasing hormone receptor 7.43580036564 6.08092190762 P30968 P30969 476357 475.627 Membrane receptor 46195,46195 46195 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 7.23683036131 6.26760624018 P30968 P30969 476358 475.627 Membrane receptor 46195,46195 46195 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 6.99148333035 5.22914798836 P30968 P30969 476436 476.615 Membrane receptor 46195,46195 46195 IC50,IC50 IC50 Oxytocin receptor 6.2757241304 6.43179827593 P30559 P70536 214427 459.598 Membrane receptor 52842 52842 Ki Ki Vasopressin V2 receptor 5.25181197299 4.5376020021 P30518 Q00788 214427 459.598 Membrane receptor 52842 52842 Ki Ki Vasopressin V1a receptor 5.79588001734 4.58502665203 P37288 P30560 214427 459.598 Membrane receptor 52842 52842 Ki Ki Glucagon receptor 7.25963731051 7.25181197299 P47871 P30082 99195 563.608 Membrane receptor 34824 34824 IC50 IC50 Gonadotropin-releasing hormone receptor 7.81913608199 7.46852108296 P30968 P30969 477537 442.599 Membrane receptor 46170,46170 46170 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 7.7447274949 7.10790539731 P30968 P30969 477538 456.626 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.58502665203 7.23657200644 P30968 P30969 477539 484.679 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 8.0 7.2924298239 P30968 P30969 477540 456.626 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.55562951966 7.38721614328 P30968 P30969 477604 470.652 Membrane receptor 46170,46170 46170 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 7.95860731484 7.16115090926 P30968 P30969 477759 470.652 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.99148333035 7.30980391997 P30968 P30969 477760 484.679 Membrane receptor 46170,46170 46170 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 7.5376020021 7.24412514433 P30968 P30969 477761 498.705 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.24412514433 6.92081875395 P30968 P30969 477762 498.705 Membrane receptor 46170 46170 IC50 IC50 Adenosine A3 receptor 3.93181413825 4.3767507096 P33765 P28647 215973 318.411 Membrane receptor 13586 13586 Ki Ki Gonadotropin-releasing hormone receptor 7.67778070527 6.5376020021 P30968 P30969 478233 414.546 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.48148606012 7.00877392431 P30968 P30969 478234 428.572 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.74074303006 7.55284196866 P30968 P30969 478296 428.572 Membrane receptor 46170,46170 46170 IC50,IC50 IC50 Gonadotropin-releasing hormone receptor 7.04575749056 6.07058107429 P30968 P30969 478298 429.557 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.50863830617 6.13076828027 P30968 P30969 478299 443.584 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.43179827593 6.49485002168 P30968 P30969 478357 457.61 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.56863623584 6.25963731051 P30968 P30969 478358 457.61 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.69897000434 6.92081875395 P30968 P30969 478360 473.676 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.63827216398 6.50863830617 P30968 P30969 478495 442.599 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.65757731918 6.60205999133 P30968 P30969 478496 456.626 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.42021640338 6.34678748622 P30968 P30969 478498 456.626 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.36653154442 6.45593195565 P30968 P30969 478567 456.626 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 8.00438696215 7.61978875829 P30968 P30969 478569 456.626 Membrane receptor 46170,46170,50731,50731 46170,50731,50731 IC50,IC50,IC50,IC50 IC50,IC50,IC50 Gonadotropin-releasing hormone receptor 7.92081875395 7.32790214206 P30968 P30969 478639 470.652 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.72124639905 7.21467016499 P30968 P30969 478640 470.652 Membrane receptor 46170 46170 IC50 IC50 Gonadotropin-releasing hormone receptor 7.2429919098 7.30980391997 P30968 P30969 478641 484.679 Membrane receptor 46170,46170 46170 IC50,IC50 IC50 D-amino-acid oxidase 7.44826918895 6.37263414341 P14920 O35078 478724 151.119 Enzyme 46745,42099 46745 IC50,IC50 IC50 D-amino-acid oxidase 8.52287874528 6.7447274949 P14920 O35078 478725 179.148 Enzyme 46745 46745 IC50 IC50 Oxytocin receptor 6.0 5.79588001734 P30559 P70536 210864 339.451 Membrane receptor 52842 52842 Ki Ki D-amino-acid oxidase 8.0 5.84013215291 P14920 O35078 478796 179.148 Enzyme 46745 46745 IC50 IC50 D-amino-acid oxidase 8.04575749056 6.5114492835 P14920 O35078 478936 179.148 Enzyme 46745 46745 IC50 IC50 D-amino-acid oxidase 7.48148606012 5.05948351507 P14920 O35078 478938 195.602 Enzyme 46745 46745 IC50 IC50 D-amino-acid oxidase 8.39794000867 7.39794000867 P14920 O35078 478941 195.602 Enzyme 46745 46745 IC50 IC50 D-amino-acid oxidase 7.79588001734 5.07211658967 P14920 O35078 478945 175.184 Enzyme 46745 46745 IC50 IC50 D-amino-acid oxidase 8.09691001301 5.43592602102 P14920 O35078 479020 189.211 Enzyme 46745 46745 IC50 IC50 D-amino-acid oxidase 7.49485002168 5.51130830168 P14920 O35078 479024 162.145 Enzyme 46745 46745 IC50 IC50 Niemann-Pick C1-like protein 1 7.92693598216 7.79588001734 Q9UHC9 Q6T3U3 479057 622.616 Membrane other 46716,46716 46716 IC50,IC50 IC50 Niemann-Pick C1-like protein 1 5.72809009743 4.46852108296 Q9UHC9 Q6T3U3 479058 462.582 Membrane other 46716,46716 46716 IC50,IC50 IC50 D-amino-acid oxidase 8.52287874528 8.39794000867 P14920 O35078 479090 214.581 Enzyme 46745 46745 IC50 IC50 Niemann-Pick C1-like protein 1 5.30102999566 3.95860731484 Q9UHC9 Q6T3U3 479123 516.674 Membrane other 46716,46716 46716 IC50,IC50 IC50 Adenosine A3 receptor 4.44611697336 4.81247927916 P33765 P28647 216994 272.384 Membrane receptor 13586 13586 Ki Ki Pyrimidinergic receptor P2Y6 6.6883753548 6.69897000434 Q15077 Q63371 217096 404.161 Membrane receptor 30315,31866,42212,49079,49584,51313 46909 IC50,IC50,IC50,IC50,IC50,IC50 IC50 Adenosine A2b receptor 9.09691001301 8.66 P29275 P29276 479429 410.446 Membrane receptor 46704 46704 Ki IC50 Adenosine A2a receptor 7.97881070093 7.55 P29274 P30543 479429 410.446 Membrane receptor 46704 46704 Ki IC50 Mu opioid receptor 9.58057545463 8.37973910399 P35372 P33535 36315 341.401 Membrane receptor 17097,17097,20966,31576,31889,31889,34746,34748,35613,36720,36965,36965,37230,38573,38573,46008,45005,46432,46432,46432 11348,11348 IC50,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,IC50,IC50 IC50,Ki Delta opioid receptor 7.85387196432 7.59832949244 P41143 P33533 36315 341.401 Membrane receptor 17097,17097,20966,31576,31889,31889,34746,34748,35613,36720,36965,36965,37230,38573,38573,46008,45005,46432,46432,46432 14428,10692 IC50,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,IC50,IC50 Ki,Ki Renin 9.22184874962 7.09691001301 P00797 P08424 480746 551.758 Enzyme 47217,46771,46771,48265,48265,49462,49462 53821 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 Prostanoid EP1 receptor 7.79588001734 7.89962945488 P34995 P70597 480883 381.852 Membrane receptor 46595 46595 IC50 IC50 Vanilloid receptor 6.93053302987 6.54415492062 Q8NER1 O35433 382643 361.437 Ion channel 36134,36134 36134,36134 IC50,IC50 IC50,IC50 Adenosine A2a receptor 7.21897258517 7.55284196866 P29274 P30543 219271 482.276 Membrane receptor 17274,17274,17274,17274,17274,17274 16218 Ki,Ki,Ki,Ki,Ki,Ki Ki Adenosine A2a receptor 9.0 7.82390874094 P29274 P30543 517265 424.471 Membrane receptor 45839 45839 Ki IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 8.14779603631 8.39794000867 P36544 Q05941 482512 682.8 Ion channel 36679,36679,36679,36679 39867 Ki,Ki,IC50,IC50 Ki Phospholipase A2 group IIA 4.78263572911 4.6615435064 P14555 P14423 482639 400.551 Enzyme 40039,40039 40039 IC50,IC50 IC50 Phospholipase A2 group IIA 4.93422274512 4.64716220437 P14555 P14423 482640 400.551 Enzyme 40039,40039 40039,40039 IC50,IC50 IC50,IC50 Serotonin 2a (5-HT2a) receptor 8.44369749923 8.82390874094 P28223 P14842 220775 230.306 Membrane receptor 17200 17200,17200,17200 Ki IC50,IC50,Ki Gonadotropin-releasing hormone receptor 8.22184874962 6.09691001301 P30968 P30969 220854 588.664 Membrane receptor 31350 14661 IC50 IC50 Serotonin 2a (5-HT2a) receptor 9.18708664336 9.39794000867 P28223 P14842 221517 321.155 Membrane receptor 30538 17200,17200,17200,30538,36532 Ki IC50,IC50,Ki,IC50,IC50 Adenosine A3 receptor 5.69464863055 5.3705904009 P33765 P28647 221831 414.581 Membrane receptor 15182 15333 Ki Ki Adenosine A1 receptor 4.62708799703 5.3387415027 P30542 P25099 484449 862.822 Membrane receptor 41516,41516,41516 41516,41516 Ki,Ki,Ki Ki,IC50 Cannabinoid CB1 receptor 8.72883630861 9.08092190762 P21554 P20272 486200 468.88 Membrane receptor 42092,42092 42092 Ki,IC50 Ki Cannabinoid CB1 receptor 8.71684018924 8.68613277963 P21554 P20272 486392 476.882 Membrane receptor 42092,42092 42092 Ki,IC50 Ki Cannabinoid CB1 receptor 9.44369749923 9.38721614328 P21554 P20272 486395 503.947 Membrane receptor 42092,42092 42092 Ki,IC50 Ki Serotonin 2a (5-HT2a) receptor 7.07058107429 7.07058107429 P28223 P14842 486993 439.57 Membrane receptor 42101 48248 IC50 Ki Serotonin 1a (5-HT1a) receptor 7.64401207282 8.33724216832 P08908 P19327 486993 439.57 Membrane receptor 42101,52373 48248 IC50,Ki Ki Melanocortin receptor 3 6.30980391997 6.46852108296 P41968 P32244 487109 531.105 Membrane receptor 42045 42045 Ki Ki Melanocortin receptor 4 7.34678748622 8.25963731051 P32245 P70596 487109 531.105 Membrane receptor 42045,42045 42045 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 8.52287874528 6.7447274949 P28845 P16232 487126 290.424 Enzyme 42046 42046 Ki Ki Gonadotropin-releasing hormone receptor 9.30102999566 5.92081875395 P30968 P30969 487193 545.5 Membrane receptor 45332,45332,42049 45332 Ki,IC50,Ki Ki Gonadotropin-releasing hormone receptor 8.0 7.13220055015 P30968 P30969 487202 456.626 Membrane receptor 42049,50731,50731 50731,50731 IC50,IC50,IC50 IC50,IC50 Dopamine D2 receptor 7.87289520164 7.24565166429 P14416 P61169 487274 468.486 Membrane receptor 42030 42030,42030,42030 IC50 Ki,Ki,Ki Dopamine D3 receptor 10.2218487496 8.73992861201 P35462 P19020 487274 468.486 Membrane receptor 42030 42030,42030,42030 IC50 Ki,Ki,Ki Dopamine D2 receptor 7.70114692359 6.57839607313 P14416 P61169 487543 475.692 Membrane receptor 42030 42030 IC50 Ki Dopamine D3 receptor 10.0705810743 9.03621217265 P35462 P19020 487543 475.692 Membrane receptor 42030 42030 IC50 Ki Anandamide amidohydrolase 8.25963731051 8.52287874528 O00519 P97612 488243 335.403 Enzyme 44028 44028,44028,44028 Ki IC50,Ki,Ki Adenosine A2b receptor 7.25181197299 6.73048705578 P29275 P29276 365442 304.387 Membrane receptor 31281,46210,51928,53892 16424 Ki,Ki,Ki,Ki Ki Adenosine A1 receptor 8.49485002168 9.04575749056 P30542 P25099 365442 304.387 Membrane receptor 17602,16931,17661,13965,3027,30254,30321,30325,31281,31341,34814,36623,37136,38162,38785,39088,43854,44049,46945,42133,46235,46210,51223,51928,53892 3027,1775,3214,11687,16931,13965,11377,16931,11292,11292,41516,41879,49741,51024 Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki IC50,IC50,IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,IC50,Ki,Ki,Ki Adenosine A2a receptor 6.58502665203 6.80410034759 P29274 P30543 365442 304.387 Membrane receptor 3282,14051,14051,14051,30254,30321,30325,31341,36623,37136,38785,39088,44049,46945,42133,46235,46210,51223,53892 3214,41879,49741,51024 IC50,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki,Ki IC50,Ki,Ki,Ki Anandamide amidohydrolase 9.03621217265 9.46852108296 O00519 P97612 489002 335.4 Enzyme 44028 44028,44028,44028 Ki Ki,Ki,Ki Anandamide amidohydrolase 7.79588001734 8.95860731484 O00519 P97612 489077 335.4 Enzyme 44028 44028,44028,44028 Ki IC50,Ki,Ki Anandamide amidohydrolase 6.95860731484 7.2757241304 O00519 P97612 489153 379.409 Enzyme 44028 44028,44028,44028 Ki IC50,Ki,Ki Anandamide amidohydrolase 8.52287874528 9.09691001301 O00519 P97612 489221 351.465 Enzyme 44028 44028,44028,44028 Ki Ki,Ki,Ki Dipeptidyl peptidase IV 7.95860731484 7.69466991846 P27487 P14740 643454 393.442 Enzyme 34705 34705,34705 Ki Ki,Ki D-amino-acid oxidase 8.09691001301 6.70774392864 P14920 O35078 478937 179.148 Enzyme 46745 46745 IC50 IC50 Dihydrofolate reductase 5.52287874528 5.6143937264 P00374 Q920D2 489492 327.447 Enzyme 43976 43976 IC50 IC50 Dihydrofolate reductase 4.55284196866 5.05060999336 P00374 Q920D2 489495 359.446 Enzyme 43976 43976 IC50 IC50 Adenosine A1 receptor 5.95428594106 5.74112337063 P30542 P25099 227480 389.411 Membrane receptor 15707,53892 15707 Ki,Ki Ki Adenosine A2a receptor 9.35298745295 9.30102999566 P29274 P30543 227480 389.411 Membrane receptor 15707,53080 15707 Ki,Ki Ki Dihydrofolate reductase 4.79588001734 5.69897000434 P00374 Q920D2 489750 299.394 Enzyme 43976 43976 IC50 IC50 Dihydrofolate reductase 4.52287874528 5.72124639905 P00374 Q920D2 489751 329.42 Enzyme 43976 43976 IC50 IC50 Dihydrofolate reductase 4.56863623584 5.33724216832 P00374 Q920D2 489753 359.446 Enzyme 43976 43976 IC50 IC50 C-X-C chemokine receptor type 3 9.0 8.39794000867 P49682 Q9JII9 618614 688.613 Membrane receptor 50038,50038,50038,50038,50038,50038,50038 50038 IC50,IC50,IC50,IC50,IC50,IC50,IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 8.30102999566 8.39794000867 P28845 P16232 365490 452.513 Enzyme 34818,34818,44799 34818 Ki,IC50,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 2 6.59006687667 6.44369749923 P80365 P50233 387585 470.684 Enzyme 53438 49766 IC50 IC50 11-beta-hydroxysteroid dehydrogenase 1 7.88605664769 7.04575749056 P28845 P16232 387585 470.684 Enzyme 38435,47148,53438 49766 IC50,IC50,IC50 IC50 Dihydrofolate reductase 5.58502665203 5.22548303427 P00374 Q920D2 490612 368.284 Enzyme 43976 43976 IC50 IC50 D-amino-acid oxidase 8.09691001301 6.69897000434 P14920 O35078 479023 162.145 Enzyme 46745 46745 IC50 IC50 Adenosine A1 receptor 6.86327943284 8.45311410925 P30542 P25099 82013 466.533 Membrane receptor 16931 16931,16931 Ki Ki,Ki Neurokinin 1 receptor 11.1870866434 8.13667713988 P25103 P14600 492364 1209.3 Membrane receptor 45287,49287,52184 45287,49287 Ki,Ki,Ki Ki,Ki Neurokinin 1 receptor 8.49485002168 6.15490195999 P25103 P14600 492365 1073.31 Membrane receptor 45287 45287 Ki Ki Vanilloid receptor 7.85387196432 7.52287874528 Q8NER1 O35433 492667 375.467 Ion channel 44549 44549 IC50 IC50 Adenosine A1 receptor 5.60205999133 6.04575749056 P30542 P25099 230600 394.424 Membrane receptor 15790 15790 Ki Ki Adenosine A2a receptor 8.0624693683 8.09691001301 P29274 P30543 230600 394.424 Membrane receptor 15790,15790 15790 Ki,Ki Ki Adenosine A3 receptor 7.53313237965 7.2924298239 P33765 P28647 230679 522.296 Membrane receptor 36081 16675 Ki Ki Dopamine transporter 6.09205147839 6.18045606446 Q01959 P23977 230690 297.415 Transporter 31619,49267,49267 45021 IC50,Ki,IC50 IC50 Serotonin transporter 8.55395269865 8.05551732785 P31645 P31652 230690 297.415 Transporter 31619,44579,49267,49267 45021 IC50,IC50,Ki,IC50 Ki D-amino-acid oxidase 8.30102999566 7.30102999566 P14920 O35078 479089 213.593 Enzyme 46745 46745 IC50 IC50 Dopamine D2 receptor 6.07008273386 7.46341586887 P14416 P61169 494033 391.506 Membrane receptor 45067,45067 45067,51830 IC50,IC50 Ki,Ki Cannabinoid CB1 receptor 8.49211062181 8.3767507096 P21554 P20272 494322 458.771 Membrane receptor 45084,45084 45084 Ki,Ki Ki Cannabinoid CB1 receptor 8.79843973941 8.67778070527 P21554 P20272 494323 424.326 Membrane receptor 45084,45084 45084 Ki,Ki Ki Cannabinoid CB1 receptor 8.674360993 7.61978875829 P21554 P20272 494324 439.34 Membrane receptor 45084,45084 45084 Ki,Ki Ki Cannabinoid CB1 receptor 8.55395269865 8.22914798836 P21554 P20272 494387 473.785 Membrane receptor 45084,45084 45084 Ki,Ki Ki Cannabinoid CB1 receptor 8.45015967945 8.44369749923 P21554 P20272 494389 473.785 Membrane receptor 45084,45084 45084 Ki,Ki Ki Cannabinoid CB1 receptor 8.48632519611 7.92081875395 P21554 P20272 494491 472.797 Membrane receptor 45084,45084 45084 Ki,Ki Ki Adenosine A1 receptor 6.01278077009 8.14878473178 P30542 P25099 82467 538.662 Membrane receptor 16931 16931,16931 Ki Ki,Ki Histamine H3 receptor 8.12736374745 7.4224693683 Q9Y5N1 Q9QYN8 494860 346.464 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Histamine H3 receptor 8.73184874962 8.00948500217 Q9Y5N1 Q9QYN8 494861 360.49 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Cannabinoid CB1 receptor 6.69897000434 6.66354026615 P21554 P20272 232743 409.604 Membrane receptor 44808 13682 Ki Ki Histamine H3 receptor 7.17069991412 6.42513184222 Q9Y5N1 Q9QYN8 494954 334.453 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Histamine H3 receptor 9.06878865959 8.40438696215 Q9Y5N1 Q9QYN8 495020 344.491 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Histamine H3 receptor 9.21602999566 8.405 Q9Y5N1 Q9QYN8 495021 358.518 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Histamine H3 receptor 7.80431915308 7.13860731484 Q9Y5N1 Q9QYN8 495022 360.49 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Histamine H3 receptor 9.07062319952 8.34161413287 Q9Y5N1 Q9QYN8 495078 360.49 Membrane receptor 45718,45718 45718,45718 IC50,Ki Ki,IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 8.16115090926 8.0 P36544 Q05941 495110 284.353 Ion channel 30228 6769 Ki IC50 Oxytocin receptor 9.18708664336 9.1739251973 P30559 P70536 496153 625.138 Membrane receptor 52842 52842 Ki Ki Adenosine A2a receptor 7.69924160817 7.31875876262 P29274 P30543 496613 344.411 Membrane receptor 45661,45661 45661 Ki,IC50 Ki Adenosine A2a receptor 7.94119865415 7.2076083105 P29274 P30543 496797 338.364 Membrane receptor 45867,45867,45661,45661 45867 IC50,Ki,Ki,IC50 Ki Dihydroorotate dehydrogenase 6.93181413825 7.67778070527 Q02127 Q63707 235052 296.245 Enzyme 47058 34935 IC50 IC50 Adenosine A1 receptor 6.23732143627 8.21125410008 P30542 P25099 82949 490.915 Membrane receptor 16931 16931,16931 Ki Ki,Ki Gonadotropin-releasing hormone receptor 8.37897788032 7.05063740921 P30968 P30969 476285 509.602 Membrane receptor 46195,46195 46195,46195 IC50,IC50 IC50,IC50 Cannabinoid CB1 receptor 6.37468754904 7.90657831484 P21554 P20272 498748 557.212 Membrane receptor 46331 46425 Ki Ki Cannabinoid CB2 receptor 5.3767507096 5.3767507096 P34972 Q9QZN9 498748 557.212 Membrane receptor 46425 46425 Ki Ki Cannabinoid CB1 receptor 8.97930365742 8.33992685694 P21554 P20272 498930 520.488 Membrane receptor 46260,46260,46260,46260 46260,46260,46260,46260 IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Cannabinoid CB1 receptor 8.76880100105 8.56304920107 P21554 P20272 499005 546.525 Membrane receptor 46260,46260,46260,46260 46260,46260,46260,46260 IC50,IC50,IC50,IC50 IC50,IC50,IC50,IC50 Cannabinoid CB1 receptor 7.32790214206 6.93523561307 P21554 P20272 499066 506.461 Membrane receptor 46260,46260,46260 46260,46260,46260,46260 IC50,IC50,IC50 IC50,IC50,IC50,IC50 Adenosine A1 receptor 7.16749108729 7.45593195565 P30542 P25099 500016 400.428 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.73518217699 6.60205999133 P30542 P25099 500068 494.566 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.81815641206 6.47495519296 P29274 P30543 500068 494.566 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 8.1877553032 6.35163998902 P29274 P30543 500069 529.011 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.96257350206 6.74957999769 P30542 P25099 500070 543.038 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.79317412397 6.09745322069 P29274 P30543 500070 543.038 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.64975198167 6.41341269533 P30542 P25099 500129 543.038 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.47755576649 5.76195389687 P29274 P30543 500129 543.038 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.68402965454 6.44490555142 P30542 P25099 500194 512.557 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.8416375079 6.41116827441 P29274 P30543 500194 512.557 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.63827216398 6.95467702121 P30542 P25099 500195 526.583 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.55595520408 6.10679324694 P29274 P30543 500195 526.583 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 7.64397414281 6.91364016933 P29274 P30543 500196 562.564 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.24949160515 6.33441900898 P30542 P25099 500258 576.591 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.83863199777 5.81247927916 P29274 P30543 500258 576.591 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.58335949266 6.56383735296 P30542 P25099 500260 576.591 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.51427857352 5.76955107862 P29274 P30543 500260 576.591 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.42021640338 6.45099673797 P30542 P25099 500336 524.592 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.62708799703 6.03905380427 P29274 P30543 500336 524.592 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.48412615629 5.99139982824 P29274 P30543 500402 538.619 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.99139982824 6.36051351073 P29274 P30543 500403 538.576 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 6.35359627378 7.10017949757 P30542 P25099 500404 552.602 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.95078197733 6.22914798836 P29274 P30543 500404 552.602 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 7.31515463836 6.92445303861 P29274 P30543 500476 514.984 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 5.42945706012 7.38195190329 P29274 P30543 500554 524.592 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 6.56703070913 6.16685288809 P29274 P30543 500556 522.619 Membrane receptor 46829 46829 Ki Ki Adenosine A1 receptor 5.93181413825 7.41453927049 P30542 P25099 500629 522.619 Membrane receptor 46829 46829 Ki Ki Adenosine A2a receptor 7.02456819149 6.86646109163 P29274 P30543 500629 522.619 Membrane receptor 46829 46829 Ki Ki Histamine H3 receptor 8.84948500217 9.52287874528 Q9Y5N1 Q9QYN8 500759 550.467 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.17827366176 8.30102999566 Q9Y5N1 Q9QYN8 500760 501.562 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.84948500217 9.69897000434 Q9Y5N1 Q9QYN8 500761 465.509 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 7.84201482727 7.88605664769 Q9Y5N1 Q9QYN8 500762 467.481 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.69897000434 9.39794000867 Q9Y5N1 Q9QYN8 500825 451.482 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.33889035263 8.30102999566 Q9Y5N1 Q9QYN8 501020 478.507 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Neuropeptide Y receptor type 5 8.85387196432 9.1739251973 Q15761 Q63634 501149 400.43 Membrane receptor 46791 46791 IC50 IC50 Histamine H3 receptor 7.20817394573 7.04095860768 Q9Y5N1 Q9QYN8 501765 371.473 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.5484550065 8.69897000434 Q9Y5N1 Q9QYN8 501766 369.457 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.30989437914 8.39794000867 Q9Y5N1 Q9QYN8 501767 385.5 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.30102999566 8.15490195999 Q9Y5N1 Q9QYN8 501768 371.473 Membrane receptor 46764 46764 Ki Ki Histamine H3 receptor 8.22184874962 7.2757241304 Q9Y5N1 Q9QYN8 501769 383.527 Membrane receptor 46764 46764 Ki Ki Histamine H3 receptor 8.04575749056 7.43179827593 Q9Y5N1 Q9QYN8 501834 399.526 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.5484550065 7.85387196432 Q9Y5N1 Q9QYN8 501835 371.473 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.61092437481 8.52287874528 Q9Y5N1 Q9QYN8 501836 405.481 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.5484550065 8.52287874528 Q9Y5N1 Q9QYN8 501837 405.481 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.1883753548 8.15490195999 Q9Y5N1 Q9QYN8 501838 419.538 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 7.55987911205 7.02227639471 Q9Y5N1 Q9QYN8 501912 371.473 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.46040937698 9.0 Q9Y5N1 Q9QYN8 501913 453.498 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.46040937698 9.0 Q9Y5N1 Q9QYN8 501914 487.506 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.5 8.30102999566 Q9Y5N1 Q9QYN8 501915 447.561 Membrane receptor 46764,46764,53081,53081 46764 Ki,IC50,Ki,IC50 Ki Alpha-1a adrenergic receptor 9.48148606012 9.01322826573 P35348 P43140 239828 585.726 Membrane receptor 15233 15233 Ki Ki Histamine H3 receptor 8.02047930384 8.30102999566 Q9Y5N1 Q9QYN8 501981 447.518 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.46040937698 8.39794000867 Q9Y5N1 Q9QYN8 501982 483.572 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.32878865959 8.39794000867 Q9Y5N1 Q9QYN8 501983 563.632 Membrane receptor 46764,46764 46764 Ki,IC50 Ki Histamine H3 receptor 8.61092437481 8.69897000434 Q9Y5N1 Q9QYN8 501984 444.517 Membrane receptor 46764,46764 46764 Ki,IC50 Ki 11-beta-hydroxysteroid dehydrogenase 1 8.0 4.83863199777 P28845 P16232 502044 350.394 Enzyme 46809,46809 46809 IC50,IC50 IC50 Corticotropin releasing factor receptor 1 8.92081875395 8.22184874962 P34998 P35353 520749 391.87 Membrane receptor 47072 47072,47072 IC50 IC50,IC50 Serotonin transporter 7.61798295743 9.39794000867 P31645 P31652 353739 427.487 Transporter 31450 31450 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.44369749923 6.42021640338 P36544 Q05941 83659 182.22 Ion channel 45299 6769 IC50 IC50 Adenosine A1 receptor 7.55284196866 7.78251605579 P30542 P25099 241454 385.417 Membrane receptor 3027 3027 IC50 IC50 Metabotropic glutamate receptor 4 6.46852108296 7.09691001301 Q14833 P31423 564895 264.228 Membrane receptor 47355 47355 IC50 IC50 D-amino-acid oxidase 8.39794000867 6.66756154008 P14920 O35078 244271 161.157 Enzyme 46745 46745 IC50 IC50 Dihydrofolate reductase 3.08990945441 4.60205999133 P00374 Q920D2 565100 544.602 Enzyme 47416 47416 IC50 IC50 Sodium channel protein type X alpha subunit 6.55284196866 6.36653154442 Q9Y5Y9 Q62968 507784 290.745 Ion channel 42188 42188 IC50 IC50 Sodium channel protein type X alpha subunit 6.52287874528 6.40893539297 Q9Y5Y9 Q62968 507840 372.888 Ion channel 42188 42188 IC50 IC50 Sodium channel protein type X alpha subunit 7.52287874528 7.04575749056 Q9Y5Y9 Q62968 507898 394.55 Ion channel 42188 42188 IC50 IC50 Mu opioid receptor 7.81247927916 7.82973828461 P35372 P33535 509924 808.02 Membrane receptor 42132 42132 Ki Ki Mu opioid receptor 9.79588001734 9.79588001734 P35372 P33535 510042 500.589 Membrane receptor 31329 44204 Ki Ki Delta opioid receptor 10.3767507096 10.3767507096 P41143 P33533 510042 500.589 Membrane receptor 31329 44204 Ki Ki Cannabinoid CB2 receptor 6.4300604568 7.01322826573 P34972 Q9QZN9 510046 428.462 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.20115240704 6.18708664336 P21554 P20272 510200 428.458 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 8.16376634347 8.49485002168 P34972 Q9QZN9 510200 428.458 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 5.92081875395 6.48148606012 P21554 P20272 510287 462.903 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 8.98328812226 9.39794000867 P34972 Q9QZN9 510287 462.903 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 5.85387196432 6.55284196866 P21554 P20272 510288 442.485 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 9.68925606771 9.56863623584 P34972 Q9QZN9 510288 442.485 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.14935376482 6.61978875829 P21554 P20272 510289 453.468 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 9.2760335672 9.88605664769 P34972 Q9QZN9 510289 453.468 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 8.42021640338 8.88605664769 P34972 Q9QZN9 510290 436.465 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 7.99826973395 9.42021640338 P34972 Q9QZN9 510347 418.488 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 7.59724957092 6.88605664769 P21554 P20272 510348 431.247 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.57745097999 7.95860731484 P34972 Q9QZN9 510348 431.247 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 5.63827216398 6.65757731918 P21554 P20272 510349 432.235 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 8.85166740487 9.39794000867 P34972 Q9QZN9 510349 432.235 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 8.35498269432 8.16115090926 P34972 Q9QZN9 510350 486.827 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.6757175447 6.65757731918 P21554 P20272 510407 436.891 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 9.00886438348 8.95860731484 P34972 Q9QZN9 510407 436.891 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.27257757 7.23657200644 P34972 Q9QZN9 510409 413.753 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.40483415091 7.10237290871 P34972 Q9QZN9 510411 448.198 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.06056683152 7.13667713988 P34972 Q9QZN9 510465 414.741 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.68125513524 8.50863830617 P34972 Q9QZN9 510466 469.777 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 8.40260412114 8.88605664769 P34972 Q9QZN9 510467 403.838 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 5.79588001734 6.76955107862 P21554 P20272 510468 392.812 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 9.42693598216 9.39794000867 P34972 Q9QZN9 510468 392.812 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 6.9761679027 6.88605664769 P34972 Q9QZN9 510469 455.793 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.22734644177 6.72124639905 P34972 Q9QZN9 510536 378.828 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 6.86407919673 6.5376020021 P34972 Q9QZN9 510537 423.291 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.45469464609 7.11350927483 P21554 P20272 510538 417.264 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 8.7135641989 8.88605664769 P34972 Q9QZN9 510538 417.264 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.01459419456 6.88605664769 P21554 P20272 510539 466.816 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 9.73109045246 8.88605664769 P34972 Q9QZN9 510539 466.816 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.32790214206 6.61978875829 P21554 P20272 510540 382.819 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 7.62981865525 7.34678748622 P34972 Q9QZN9 510540 382.819 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 5.98148606012 7.08092190762 P21554 P20272 510624 418.248 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 8.2931825014 8.2924298239 P34972 Q9QZN9 510624 418.248 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.01928945297 6.26760624018 P21554 P20272 510625 390.839 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB2 receptor 7.96479633913 7.79588001734 P34972 Q9QZN9 510625 390.839 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Cannabinoid CB1 receptor 6.09151498112 5.79588001734 P21554 P20272 510626 381.831 Membrane receptor 44207 44207 IC50 IC50 Cannabinoid CB2 receptor 6.70335696649 6.42021640338 P34972 Q9QZN9 510626 381.831 Membrane receptor 44207,44207 44207 IC50,IC50 IC50 Corticotropin releasing factor receptor 1 8.69897000434 8.01322826573 P34998 P35353 511234 385.46 Membrane receptor 44165 47072 Ki IC50 Norepinephrine transporter 6.14792474158 6.03621217265 P23975 Q9WTR4 609542 259.343 Transporter 31321,31321 13641,13641,14202,12788,13096 Ki,IC50 IC50,IC50,IC50,IC50,Ki Dopamine transporter 7.63827216398 7.63827216398 Q01959 P23977 609542 259.343 Transporter 31321 13641,13641,14202,12788,13096 IC50 IC50,IC50,IC50,IC50,Ki Serotonin transporter 6.22866196317 5.69897000434 P31645 P31652 609542 259.343 Transporter 31321,31321 13641,13641,14202,12788 Ki,IC50 IC50,IC50,IC50,IC50 Vanilloid receptor 8.82390874094 9.30102999566 Q8NER1 O35433 511612 478.39 Ion channel 44130,50778 44130 IC50,IC50 IC50 Sodium channel protein type X alpha subunit 7.58502665203 7.01322826573 Q9Y5Y9 Q62968 710456 386.367 Ion channel 53444 53444 IC50 IC50 Dopamine D1 receptor 7.52287874528 7.19382002602 P21728 P18901 33087 255.312 Membrane receptor 38679 11749,11749,10358,10358,10581 IC50 IC50,IC50,Ki,Ki,IC50 Adenosine A2b receptor 9.0 9.33 P29275 P29276 512447 555.42 Membrane receptor 44739 44739 Ki IC50 Adenosine A2a receptor 7.0 6.65 P29274 P30543 512447 555.42 Membrane receptor 44739 44739 Ki IC50 11-beta-hydroxysteroid dehydrogenase 1 7.4622265193 6.49569991412 P28845 P16232 512642 310.387 Enzyme 44799,44799 44799,44799 Ki,IC50 Ki,IC50 Dopamine transporter 7.33441900898 6.60024701827 Q01959 P23977 513010 303.353 Transporter 52167 35801,35801 Ki Ki,IC50 Dopamine D2 receptor 7.39147396642 7.39147396642 P14416 P61169 513629 393.565 Membrane receptor 49130 44804,47595,52843 Ki Ki,Ki,Ki Dopamine D3 receptor 8.75202673364 8.75202673364 P35462 P19020 513629 393.565 Membrane receptor 49130 44804,47595,52843 Ki Ki,Ki,Ki Dopamine D2 receptor 7.58502665203 6.62342304294 P14416 P61169 513631 393.565 Membrane receptor 49130 44804 Ki Ki Dopamine D3 receptor 9.08354605145 7.73518217699 P35462 P19020 513631 393.565 Membrane receptor 49130 44804 Ki Ki Dopamine D2 receptor 7.13977149836 6.60459010786 P14416 P61169 513723 475.692 Membrane receptor 49130,49130 44804,47595 Ki,IC50 Ki,Ki Dopamine D3 receptor 9.55339662347 9.03503521996 P35462 P19020 513723 475.692 Membrane receptor 49130,49130 44804,47595 Ki,IC50 Ki,Ki Serotonin transporter 7.22989159052 8.56523160377 P31645 P31652 514014 455.952 Transporter 44692,44692 44692,44692 IC50,IC50 Ki,Ki Serotonin transporter 7.24565435657 8.08133206599 P31645 P31652 514016 421.507 Transporter 44692,44692 44692,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.96257350206 8.22914798836 P31645 P31652 514017 421.507 Transporter 44692 44692 IC50 Ki Histamine H3 receptor 9.16909365723 8.7447274949 Q9Y5N1 Q9QYN8 514035 403.517 Membrane receptor 44709,44709 44709 IC50,Ki Ki Serotonin transporter 8.09691001301 7.48148606012 P31645 P31652 514036 428.526 Transporter 44645 44645 IC50 IC50 Serotonin transporter 7.82390874094 8.08092190762 P31645 P31652 514087 453.524 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.83268266525 7.99139982824 P31645 P31652 514088 453.524 Transporter 44692 44692 IC50 Ki Serotonin transporter 5.73048705578 6.79317412397 P31645 P31652 514089 454.509 Transporter 44692 44692 IC50 Ki Histamine H3 receptor 8.96259177968 8.63827216398 Q9Y5N1 Q9QYN8 514102 457.488 Membrane receptor 44709,44709 44709 IC50,Ki Ki Serotonin transporter 5.98885263922 6.30233483735 P31645 P31652 514155 440.482 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.55439579673 8.023650021 P31645 P31652 514156 467.551 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.48545224734 8.09908693226 P31645 P31652 514157 481.577 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.34969247687 7.94769090035 P31645 P31652 514158 481.577 Transporter 44692 44692 IC50 Ki Phospholipase A2 group IIA 7.09691001301 6.92081875395 P14555 P14423 514243 730.969 Enzyme 44657 44657 IC50 IC50 Phospholipase A2 group IIA 6.16115090926 7.09691001301 P14555 P14423 514245 504.742 Enzyme 44657 44657 IC50 IC50 Serotonin transporter 7.15739076039 8.09420411963 P31645 P31652 514269 479.561 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.15119529895 8.1390633793 P31645 P31652 514270 493.588 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.8416375079 7.70333480974 P31645 P31652 514271 521.641 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.36051351073 8.16052195263 P31645 P31652 514272 493.588 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.80683079182 8.32798079723 P31645 P31652 514336 446.517 Transporter 44692,44692 44692,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.75246383822 7.66104147384 P31645 P31652 514337 453.524 Transporter 44692,44692 44692,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.21324857785 7.12205304837 P31645 P31652 514432 455.952 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.04624030827 6.62433638604 P31645 P31652 514433 439.498 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.89645222979 8.19583862763 P31645 P31652 514505 457.488 Transporter 44692,44692 44692,44692 IC50,IC50 Ki,Ki Serotonin transporter 6.11013827874 7.15490195999 P31645 P31652 514574 441.513 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.36151074305 7.48280410205 P31645 P31652 514575 441.513 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.8601209136 7.41228903498 P31645 P31652 514661 453.524 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.98716277529 6.53985418251 P31645 P31652 514723 453.524 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.35457773065 7.90308998699 P31645 P31652 514786 414.488 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.42136079003 7.75696195131 P31645 P31652 514787 414.488 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.53610701101 7.50112338058 P31645 P31652 514788 411.444 Transporter 44692 44692,44692 IC50 Ki,Ki Serotonin transporter 6.34486156519 7.8696662315 P31645 P31652 514855 414.488 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.6143937264 8.61978875829 P31645 P31652 514934 441.513 Transporter 44692 44692 IC50 Ki Serotonin transporter 7.32790214206 7.94692155652 P31645 P31652 514935 441.513 Transporter 44692 44692 IC50 Ki Serotonin transporter 6.83564714422 7.63078414259 P31645 P31652 514936 409.496 Transporter 44692 44692 IC50 Ki Histamine H3 receptor 7.21968268786 6.42021640338 Q9Y5N1 Q9QYN8 452099 410.635 Membrane receptor 44314 44314 Ki Ki Adenosine A1 receptor 4.92081875395 4.16115090926 P30542 P25099 101593 149.153 Membrane receptor 46210 11175 Ki Ki Gonadotropin-releasing hormone receptor 8.93483311575 5.35654732351 P30968 P30969 515206 631.59 Membrane receptor 45332,45332 45332 Ki,IC50 Ki Adenosine A2a receptor 8.35834938565 7.92081875395 P29274 P30543 516457 355.366 Membrane receptor 45867,45867 45867 IC50,Ki Ki Histamine H3 receptor 7.91009488856 6.77989191196 Q9Y5N1 Q9QYN8 566679 357.287 Membrane receptor 47387 47387 Ki Ki Gonadotropin-releasing hormone receptor 6.7447274949 7.08092190762 P30968 P30969 304539 551.675 Membrane receptor 20757 20757 IC50 IC50 Gonadotropin-releasing hormone receptor 6.12493873661 6.34678748622 P30968 P30969 304541 537.649 Membrane receptor 20757 20757 IC50 IC50 Adenosine A2a receptor 9.69897000434 8.03024037369 P29274 P30543 516531 367.402 Membrane receptor 45839,45867,45867 45839,45867 Ki,IC50,Ki IC50,Ki Adenosine A2a receptor 7.86571101406 7.49485002168 P29274 P30543 516533 324.337 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 7.85387196432 7.52287874528 P29274 P30543 516535 423.468 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.12668290053 7.67778070527 P29274 P30543 516613 352.39 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 7.45402590456 7.16749108729 P29274 P30543 516614 354.363 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 7.40782466298 7.08618614762 P29274 P30543 516615 368.39 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.48348927766 8.0 P29274 P30543 516690 393.442 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.01077278332 7.69897000434 P29274 P30543 516692 351.406 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.65182180563 8.15490195999 P29274 P30543 516777 406.484 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.14878473178 7.85387196432 P29274 P30543 516778 395.458 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.53631481848 8.82390874094 P29274 P30543 516844 393.442 Membrane receptor 45867,45867 45867 IC50,Ki Ki Adenosine A2a receptor 8.18941185911 8.0 P29274 P30543 516846 407.469 Membrane receptor 45867,45867 45867 IC50,Ki Ki Vasopressin V2 receptor 8.53174312876 7.72124639905 P30518 Q00788 516898 547.983 Membrane receptor 45841,45841 45841 Ki,IC50 Ki Dopamine transporter 5.49485002168 4.69897000434 Q01959 P23977 516936 246.348 Transporter 45878 45878 IC50 IC50 Serotonin transporter 6.49485002168 7.55284196866 P31645 P31652 516936 246.348 Transporter 45878 45878 IC50 IC50 Serotonin transporter 7.01322826573 6.79588001734 P31645 P31652 516938 282.377 Transporter 45878 45878 IC50 IC50 Serotonin transporter 7.49485002168 7.95860731484 P31645 P31652 516939 276.397 Transporter 45878 45878 IC50 IC50 Adenosine A2a receptor 8.69897000434 7.3767507096 P29274 P30543 516976 406.481 Membrane receptor 45839 45839 Ki IC50 Serotonin transporter 7.09151498112 6.79588001734 P31645 P31652 517016 262.371 Transporter 45878 45878 IC50 IC50 Dopamine transporter 5.25656863485 5.69897000434 Q01959 P23977 517018 298.403 Transporter 45878 45878 IC50 IC50 Serotonin transporter 7.88605664769 7.60205999133 P31645 P31652 517018 298.403 Transporter 45878 45878 IC50 IC50 Histamine H3 receptor 8.7135641989 8.22184874962 Q9Y5N1 Q9QYN8 514805 407.481 Membrane receptor 44709,44709 44709 IC50,Ki Ki Oxytocin receptor 8.09691001301 8.05060999336 P30559 P70536 256008 554.766 Membrane receptor 44053 12711 Ki IC50 Acyl coenzyme A:cholesterol acyltransferase 1 7.45593195565 7.45593195565 P35610 O70536 518245 499.687 Enzyme 45920 48377 IC50 IC50 Cannabinoid CB1 receptor 8.27719789836 8.56066730617 P21554 P20272 113285 386.567 Membrane receptor 30590,37904,46331,48965 30590 Ki,Ki,Ki,IC50 Ki Vanilloid receptor 9.18708664336 8.31875876262 Q8NER1 O35433 436070 381.351 Ion channel 38526 38526 IC50 IC50 Fructose-1,6-bisphosphatase 5.85387196432 4.69897000434 P09467 P19112 519883 391.361 Enzyme 47053 47053 IC50 IC50 Corticotropin releasing factor receptor 1 8.32790214206 7.77860338703 P34998 P35353 519943 399.487 Membrane receptor 47072 47072,47072 IC50 IC50,IC50 Corticotropin releasing factor receptor 1 8.69897000434 7.74248719398 P34998 P35353 520017 3826.36 Membrane receptor 47071,47072 47072,47072 IC50,IC50 IC50,IC50 Fructose-1,6-bisphosphatase 5.82390874094 5.15490195999 P09467 P19112 520087 337.271 Enzyme 47053,49142 47053 IC50,IC50 IC50 Fructose-1,6-bisphosphatase 6.09691001301 5.90308998699 P09467 P19112 520088 351.298 Enzyme 47053,49142 47053 IC50,IC50 IC50 Fructose-1,6-bisphosphatase 5.95860731484 5.39794000867 P09467 P19112 520253 397.389 Enzyme 47053 47053 IC50 IC50 Corticotropin releasing factor receptor 1 8.34678748622 7.55204022734 P34998 P35353 520543 340.423 Membrane receptor 47071 47071,47071 IC50 IC50,IC50 Peroxisome proliferator-activated receptor alpha 7.36062319952 5.64589156085 Q07869 P37230 520672 437.508 Transcription Factor 47054,47054 47054 IC50,IC50 IC50 Corticotropin releasing factor receptor 1 8.46852108296 7.65757731918 P34998 P35353 520682 369.461 Membrane receptor 47072 47072,47072 IC50 IC50,IC50 Corticotropin releasing factor receptor 1 7.81815641206 8.06177560656 P34998 P35353 520691 413.513 Membrane receptor 47072 47072,47072 IC50 IC50,IC50 Fructose-1,6-bisphosphatase 5.30102999566 4.39794000867 P09467 P19112 520816 385.314 Enzyme 47053 47053 IC50 IC50 Androgen Receptor 9.09691001301 8.31875876262 P10275 P15207 520894 291.733 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 9.52287874528 7.85387196432 P10275 P15207 520895 291.733 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 9.52287874528 9.69897000434 P10275 P15207 520896 359.731 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 9.69897000434 7.72124639905 P10275 P15207 520897 359.731 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 8.63827216398 8.95860731484 P10275 P15207 520898 359.731 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 9.52287874528 8.85387196432 P10275 P15207 520899 359.731 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 9.15490195999 8.43179827593 P10275 P15207 520965 333.813 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 8.0 5.7447274949 P10275 P15207 520966 290.748 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 8.72124639905 7.35654732351 P10275 P15207 520967 304.775 Transcription Factor 47060 47060 Ki IC50 Androgen Receptor 7.76955107862 5.95506845385 P10275 P15207 520969 331.8 Transcription Factor 47060 47060 Ki IC50 Monoglyceride lipase 4.61978875829 4.61978875829 Q99685 Q8R431 567478 311.358 Enzyme 47831 47831 IC50 IC50 Metabotropic glutamate receptor 1 6.77728352885 7.48148606012 Q13255 P23385 359617 359.446 Membrane receptor 35368 31805 IC50 IC50 Histamine H3 receptor 9.02287874528 10.15490196 Q9Y5N1 Q9QYN8 436369 336.514 Membrane receptor 44506,44506 38812,44506 Ki,Ki Ki,Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.93930215965 7.75696195131 P36544 Q05941 522471 266.341 Ion channel 46997 46997 IC50 Ki Neuronal acetylcholine receptor protein alpha-7 subunit 5.3705904009 7.96259177968 P36544 Q05941 522472 280.367 Ion channel 46997,49457 46997,49457 IC50,IC50 Ki,Ki Neuronal acetylcholine receptor protein alpha-7 subunit 6.49485002168 9.61978875829 P36544 Q05941 522690 319.404 Ion channel 46997 46997 IC50 Ki Dopamine D3 receptor 8.85387196432 8.20830935098 P35462 P19020 52338 247.376 Membrane receptor 2331,42030,44689 42030,44804,47595,52843 Ki,IC50,Ki Ki,Ki,Ki,Ki Serotonin 1a (5-HT1a) receptor 7.32790214206 6.3456537789 P08908 P19327 52338 247.376 Membrane receptor 2331 12028,12058 Ki Ki,Ki Dopamine D2 receptor 7.40011692793 6.60094412076 P14416 P61169 52338 247.376 Membrane receptor 42030 12058,2331,42030,44804,47595,52843 IC50 Ki,Ki,Ki,Ki,Ki,Ki Dopamine D2 receptor 6.84771165562 6.84771165562 P14416 P61169 261089 393.565 Membrane receptor 5330,38128,38128 42030 Ki,Ki,IC50 Ki Dopamine D3 receptor 8.80687540165 8.80687540165 P35462 P19020 261089 393.565 Membrane receptor 5330,38128,38128 42030 Ki,Ki,IC50 Ki Nitric-oxide synthase, brain 4.81530856918 5.20065945055 P29475 P29476 523284 235.329 Enzyme 46991 46991 IC50 IC50 Nitric-oxide synthase, brain 5.39794000867 5.88605664769 P29475 P29476 523285 249.355 Enzyme 46991 46991 IC50 IC50 Nitric-oxide synthase, brain 4.91364016933 5.48148606012 P29475 P29476 523286 373.923 Enzyme 46991 46991 IC50 IC50 Nitric-oxide synthase, brain 6.15490195999 7.0 P29475 P29476 523287 371.495 Enzyme 46991 46991 IC50 IC50 Neuronal acetylcholine receptor protein alpha-7 subunit 5.34969247687 7.2924298239 P36544 Q05941 523295 189.257 Ion channel 46997 46997 IC50 Ki Nitric-oxide synthase, brain 5.3767507096 5.95860731484 P29475 P29476 523358 387.949 Enzyme 46991 46991 IC50 IC50 Nitric-oxide synthase, brain 6.15490195999 7.0 P29475 P29476 523359 372.48 Enzyme 46991,46991,50330 46991,46991,50330,50330 IC50,IC50,IC50 IC50,IC50,IC50,Ki Nitric-oxide synthase, brain 5.18045606446 5.5376020021 P29475 P29476 523360 372.48 Enzyme 46991 46991 IC50 IC50 Nitric-oxide synthase, brain 5.52287874528 6.15490195999 P29475 P29476 523361 385.478 Enzyme 46991 46991 IC50 IC50