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Designing Focused Chemical Libraries Enriched in Protein-Protein Interaction Inhibitors using Machine-Learning Methods

  • Christelle Reynès,

    Affiliation Inserm UMR-S 973/MTi, University Paris Diderot, Paris, France

  • Hélène Host,

    Affiliations CDithem Platform/IGM, Paris, France, Inserm UMR-S 761, Institut Pasteur de Lille, Lille, France, Université Lille 2, Faculté des Sciences Pharmaceutiques et Biologiques, Lille, France

  • Anne-Claude Camproux,

    Affiliation Inserm UMR-S 973/MTi, University Paris Diderot, Paris, France

  • Guillaume Laconde,

    Affiliations CDithem Platform/IGM, Paris, France, Inserm UMR-S 761, Institut Pasteur de Lille, Lille, France, Université Lille 2, Faculté des Sciences Pharmaceutiques et Biologiques, Lille, France

  • Florence Leroux,

    Affiliations CDithem Platform/IGM, Paris, France, Inserm UMR-S 761, Institut Pasteur de Lille, Lille, France, Université Lille 2, Faculté des Sciences Pharmaceutiques et Biologiques, Lille, France

  • Anne Mazars,

    Affiliations CDithem Platform/IGM, Paris, France, UMR-S940, Hôpital St Louis, Paris, France

  • Benoit Deprez,

    Affiliations CDithem Platform/IGM, Paris, France, Inserm UMR-S 761, Institut Pasteur de Lille, Lille, France, Université Lille 2, Faculté des Sciences Pharmaceutiques et Biologiques, Lille, France

  • Robin Fahraeus,

    Affiliations CDithem Platform/IGM, Paris, France, UMR-S940, Hôpital St Louis, Paris, France

  • Bruno O. Villoutreix,

    Affiliations Inserm UMR-S 973/MTi, University Paris Diderot, Paris, France, CDithem Platform/IGM, Paris, France

  • Olivier Sperandio

    olivier.sperandio@univ-paris-diderot.fr

    Affiliations Inserm UMR-S 973/MTi, University Paris Diderot, Paris, France, CDithem Platform/IGM, Paris, France

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